levocabastine has been researched along with neurotensin in 40 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (7.50) | 18.7374 |
1990's | 15 (37.50) | 18.2507 |
2000's | 16 (40.00) | 29.6817 |
2010's | 6 (15.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Garcia-Marin, L; Jensen, RT; Leyton, J; Moody, TW | 1 |
Bonnin, J; Caput, D; Chalon, P; Delpech, B; Ferrara, P; Guillemot, M; Kaghad, M; Le Fur, G; Vita, N | 1 |
Botto, JM; Coppola, T; Guillemare, E; Mazella, J; Sarret, P; Vincent, JP | 1 |
Botto, JM; Chabry, J; Mazella, J; Sarret, P; Vincent, JP | 1 |
Barroso, S; Kitabgi, P; Labbé-Jullié, C; Martinez, J; Richard, F | 1 |
Gendron, L; Giddings, AM; Gilmour, BP; Longpre, JM; Olepu, S; Runyon, SP; Sarret, P; Thomas, JB; Warner, KR; Wiethe, RW; Zhang, Y | 1 |
Campbell, AD; Erwin, VG; Jones, BC | 1 |
Leysen, JE; Schotte, A | 1 |
Harris, E; Pettibone, DJ; Robinson, FM; Totaro, JA | 1 |
Laduron, PM; Leysen, JE; Schotte, A | 1 |
Erwin, VG; Radcliffe, RA | 1 |
Campbell, AD; Erwin, VG | 1 |
Botto, JM; Mazella, J; Sarret, P; Vincent, JP | 1 |
Alonso, R; Beaudet, A; Faure, MP; Nouel, D; Quirion, R; St Pierre, JA | 1 |
Botto, JM; Guillemare, E; Mazella, J; Vincent, JP | 1 |
Cusack, B; Groshan, K; Richelson, E; Tyler, BM | 1 |
Forgez, P; Lombet, A; Rostène, W; Yamada, M | 1 |
Bédard, PJ; Di Paolo, T; Falardeau, P; Goulet, M; Grondin, R; Morissette, M; Rostène, W | 1 |
Laissue, JA; Reubi, JC; Schaer, JC; Waser, B | 1 |
Costentin, J; Dubuc, I; Remande, S | 1 |
Matthews, RT | 1 |
Trudeau, LE | 1 |
López Ordieres, MG; Rodríguez de Lores Arnaiz, G | 1 |
Asselin, ML; Coquerel, A; Costentin, J; Dubuc, I | 1 |
Botto, JM; Dal Farra, C; Mazella, J; Navarro, V; Sarret, P; Vincent, JP | 1 |
Azriel, Y; Burcher, E | 1 |
Greengard, P; Higashi, H; Maeda, H; Matsuyama, S; Nishi, A | 1 |
Fukui, R; Higashi, H; Matsuyama, S; Nishi, A | 1 |
Ohinata, K; Yamauchi, R; Yoshikawa, M | 1 |
Beaudet, A; Gallo-Payet, N; Gendron, L; Payet, MD; Perron, A; Sarret, P | 1 |
Beaudet, A; Gendron, L; Perron, A; Sarret, P; Stroh, T | 1 |
Beaudet, A; Esdaile, MJ; Martinez, J; Perron, A; Sarret, P; Stroh, T | 1 |
Bredeloux, P; Costentin, J; Dubuc, I | 1 |
Baudisson, S; Beaudet, N; Belleville, K; Dansereau, MA; Ezzoubaa, F; Martinez, J; Richelson, E; Roussy, G; Sarret, P | 1 |
Barbut, D; Boules, M; Liang, Y; Richelson, E; Shaw, A | 1 |
Abderrahmani, A; Béraud-Dufour, S; Brau, F; Coppola, T; Mazella, J; Noel, J; Waeber, G | 1 |
Arnaiz, GR; Ordieres, MG; Rosin, C | 1 |
Hugel, S; Kadiri, N; Rodeau, JL; Schlichter, R | 1 |
Bogdański, P; Krauss, H; Maćkowiak, P; Nowak, D; Piątek, J | 1 |
Boules, M; Richelson, E; Smith, KE; Williams, K | 1 |
40 other study(ies) available for levocabastine and neurotensin
Article | Year |
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Neurotensin causes tyrosine phosphorylation of focal adhesion kinase in lung cancer cells.
Topics: Binding, Competitive; Cell Division; Cytochalasin D; Dose-Response Relationship, Drug; Focal Adhesion Kinase 1; Focal Adhesion Protein-Tyrosine Kinases; Humans; Lung Neoplasms; Neurotensin; Nucleic Acid Synthesis Inhibitors; Peptide Fragments; Phosphorylation; Piperidines; Protein-Tyrosine Kinases; Pyrazoles; Quinolines; Receptors, Neurotensin; Tumor Cells, Cultured; Tyrosine | 2002 |
Molecular cloning of a levocabastine-sensitive neurotensin binding site.
Topics: Amino Acid Sequence; Animals; Cell Line; Chlorocebus aethiops; Hypothalamus; Molecular Sequence Data; Piperidines; Rats; Receptors, Neurotensin; RNA, Messenger; Sequence Homology, Amino Acid; Tissue Distribution | 1996 |
Structure, functional expression, and cerebral localization of the levocabastine-sensitive neurotensin/neuromedin N receptor from mouse brain.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; Histamine H1 Antagonists; Humans; Mice; Molecular Sequence Data; Neurotensin; Peptide Fragments; Piperidines; Rats; Receptors, Neurotensin; RNA, Messenger; Structure-Activity Relationship; Tissue Distribution; Xenopus laevis | 1996 |
Stable expression of the mouse levocabastine-sensitive neurotensin receptor in HEK 293 cell line: binding properties, photoaffinity labeling, and internalization mechanism.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Cell Line; Endocytosis; Gene Expression Regulation; Humans; Iodine Radioisotopes; Kinetics; Mice; Molecular Sequence Data; Neurotensin; Peptides; Photoaffinity Labels; Piperidines; Protein Binding; Receptors, Neurotensin; Signal Transduction; Transfection | 1998 |
Agonism, inverse agonism, and neutral antagonism at the constitutively active human neurotensin receptor 2.
Topics: Amino Acid Sequence; Animals; COS Cells; Histamine H1 Antagonists; Humans; Molecular Sequence Data; Neurotensin; Piperidines; Pyrazoles; Quinolines; Receptors, Neurotensin; Sequence Homology, Amino Acid; Transfection | 2001 |
Identification of 1-({[1-(4-fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane carboxylic acid as a selective nonpeptide neurotensin receptor type 2 compound.
Topics: Analgesics; Animals; Calcium; CHO Cells; Cricetulus; Cyclohexanecarboxylic Acids; Drug Partial Agonism; Pyrazoles; Radioligand Assay; Rats; Receptors, Neurotensin; Structure-Activity Relationship | 2014 |
Regional characterization of brain neurotensin receptor subtypes in LS and SS mice.
Topics: Alcohol Drinking; Animals; Binding, Competitive; Brain; Chlorpheniramine; Haloperidol; Histamine H1 Antagonists; Male; Mice; Mice, Inbred Strains; Neurotensin; Piperidines; Receptors, Neurotensin; Receptors, Neurotransmitter; Sleep Stages; Species Specificity | 1991 |
Further characterization of neurotensin binding in the rat brain: levocabastine-displaceable neurotensin binding sites are not histamine-H1 receptors.
Topics: Animals; Binding Sites; Brain; Guinea Pigs; Neurotensin; Piperidines; Rats; Receptors, Histamine H1 | 1989 |
Heterogeneity of [3H]neurotensin bindings: studies with dynorphin, L-156,903 and levocabastine.
Topics: Animals; Binding Sites; Brain; Brain Chemistry; Dynorphins; Female; In Vitro Techniques; Male; Neurotensin; Oligopeptides; Phenothiazines; Piperidines; Rats; Rats, Inbred Strains | 1988 |
Evidence for a displaceable non-specific [3H]neurotensin binding site in rat brain.
Topics: Animals; Binding, Competitive; Brain; Cats; Dogs; Guinea Pigs; Humans; In Vitro Techniques; Mice; Neurotensin; Piperidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Neurotensin; Receptors, Neurotransmitter | 1986 |
Characterization of neurotensin-stimulated phosphoinositide hydrolysis in brain regions of long sleep and short sleep mice.
Topics: Animals; Brain; Calcium; Carbachol; Cerebellum; Dose-Response Relationship, Drug; Hippocampus; Histamine H1 Antagonists; Hydrolysis; Inositol; Inositol Phosphates; Kinetics; Membrane Lipids; Mesencephalon; Mice; Mice, Inbred Strains; Neurotensin; Nucleus Accumbens; Organ Specificity; Phosphatidylinositols; Phospholipids; Piperidines; Receptors, Neurotensin; Second Messenger Systems; Sleep | 1993 |
Chronic ethanol administration downregulates neurotensin receptors in long- and short-sleep mice.
Topics: Animals; Benzamides; Benzazepines; Down-Regulation; Ethanol; Histamine H1 Antagonists; Kinetics; Male; Membranes; Mesencephalon; Mice; Mice, Inbred Strains; Neural Pathways; Neurotensin; Piperidines; Pyrrolidines; Receptors, Dopamine D1; Receptors, Neurotensin; Receptors, Neurotransmitter; Sleep; Species Specificity | 1993 |
Identification and expression of a variant isoform of the levocabastine-sensitive neurotensin receptor in the mouse central nervous system.
Topics: Amino Acid Sequence; Animals; Base Sequence; Brain; Cloning, Molecular; COS Cells; DNA, Complementary; Gene Expression; Genetic Variation; Mice; Molecular Sequence Data; Neurotensin; Piperidines; Receptors, Neurotensin | 1997 |
Differential binding profile and internalization process of neurotensin via neuronal and glial receptors.
Topics: Animals; Animals, Newborn; Binding Sites; Cells, Cultured; Cerebral Cortex; Coculture Techniques; Endocytosis; GTP-Binding Proteins; Mesencephalon; Nerve Tissue Proteins; Neuroglia; Neurons; Neurotensin; Piperidines; Protein Binding; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Signal Transduction; Tegmentum Mesencephali; Tyrosine 3-Monooxygenase | 1997 |
Effects of SR 48692 on neurotensin-induced calcium-activated chloride currents in the Xenopus oocyte expression system: agonist-like activity on the levocabastine-sensitive neurotensin receptor and absence of antagonist effect on the levocabastine insensi
Topics: Animals; Calcium; Chlorides; Electric Conductivity; Female; Mice; Neurotensin; Oocytes; Piperidines; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin | 1997 |
In vivo studies with low doses of levocabastine and diphenhydramine, but not pyrilamine, antagonize neurotensin-mediated antinociception.
Topics: Animals; Body Temperature Regulation; Diphenhydramine; Drug Evaluation, Preclinical; Histamine H1 Antagonists; Male; Mice; Neurotensin; Pain; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley | 1998 |
Distinct functional characteristics of levocabastine sensitive rat neurotensin NT2 receptor expressed in Chinese hamster ovary cells.
Topics: Animals; Calcium; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Neurotensin; Oligopeptides; Piperidines; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin; Signal Transduction; Transfection | 1998 |
Neurotensin receptors and dopamine transporters: effects of MPTP lesioning and chronic dopaminergic treatments in monkeys.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Adamantane; Animals; Autoradiography; Binding Sites; Carrier Proteins; Caudate Nucleus; Denervation; Dopamine; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Down-Regulation; Imidazoles; In Situ Hybridization; Macaca fascicularis; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Neurotensin; Piperidines; Putamen; Receptors, Dopamine; Receptors, Neurotensin; RNA, Messenger; Substantia Nigra | 1999 |
Neurotensin receptors in human neoplasms: high incidence in Ewing's sarcomas.
Topics: Animals; Bone Neoplasms; Humans; Neoplasm Proteins; Neoplasms; Neurotensin; Organ Specificity; Peptide Fragments; Piperidines; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin; RNA, Messenger; RNA, Neoplasm; Sarcoma, Ewing | 1999 |
The partial agonist properties of levocabastine in neurotensin-induced analgesia.
Topics: Analgesia; Analgesics; Animals; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Male; Mice; Neurotensin; Pain; Pain Threshold; Piperidines; Pyrilamine; Receptors, Neurotensin | 1999 |
Neurotensin depolarizes cholinergic and a subset of non-cholinergic septal/diagonal band neurons by stimulating neurotensin-1 receptors.
Topics: Action Potentials; Adamantane; Animals; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Male; Membrane Potentials; Neurons; Neurotensin; Patch-Clamp Techniques; Piperidines; Prosencephalon; Receptors, Neurotensin; Tetrodotoxin | 1999 |
Neurotensin regulates intracellular calcium in ventral tegmental area astrocytes: evidence for the involvement of multiple receptors.
Topics: Adamantane; Animals; Animals, Newborn; Astrocytes; Calcium; Cells, Cultured; Estrenes; Gadolinium; Imidazoles; Neurotensin; Peptide Fragments; Piperidines; Pyrrolidinones; Rats; Receptors, Neurotensin; Thapsigargin; Type C Phospholipases; Ventral Tegmental Area | 2000 |
Neurotensin inhibits neuronal Na+,K+-ATPase activity through high affinity peptide receptor.
Topics: Animals; Cerebral Cortex; Heating; In Vitro Techniques; Intracellular Membranes; Male; Neurotensin; Piperidines; Rats; Rats, Wistar; Receptors, Neurotensin; Sodium-Potassium-Exchanging ATPase; Synaptosomes | 2000 |
Localization of neurotensin NTS2 receptors in rat brain, using.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Brain Chemistry; Histamine H1 Antagonists; Male; Neurotensin; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin | 2001 |
Involvement of the neurotensin receptor subtype NTR3 in the growth effect of neurotensin on cancer cell lines.
Topics: Animals; Cell Membrane; CHO Cells; Cholic Acids; Colonic Neoplasms; Cricetinae; Drug Resistance, Neoplasm; Electrophoresis, Polyacrylamide Gel; Humans; Kinetics; Male; Neurotensin; Pancreatic Neoplasms; Piperidines; Prostatic Neoplasms; Protein Binding; Protein Structure, Tertiary; Receptors, Neurotensin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Transfection; Tumor Cells, Cultured | 2001 |
Characterization and autoradiographic localization of neurotensin binding sites in human sigmoid colon.
Topics: Adult; Aged; Autoradiography; Binding, Competitive; Colon, Sigmoid; Dose-Response Relationship, Drug; Enteric Nervous System; Female; Histamine H1 Antagonists; Humans; In Vitro Techniques; Iodine Radioisotopes; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Neurotensin; Peptide Fragments; Phenanthrolines; Piperidines; Protease Inhibitors; Receptors, Neurotensin; Tetrodotoxin | 2001 |
Neurotensin regulates DARPP-32 thr34 phosphorylation in neostriatal neurons by activation of dopamine D1-type receptors.
Topics: Animals; Cobalt; Dopamine; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Excitatory Amino Acid Antagonists; Glutamine; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Phosphorylation; Piperidines; Pyrazoles; Quinolines; Receptors, Dopamine D1; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin | 2002 |
Regulation of DARPP-32 Thr75 phosphorylation by neurotensin in neostriatal neurons: involvement of glutamate signalling.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Anesthetics, Local; Animals; Benzazepines; Dizocilpine Maleate; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamic Acid; Histamine H1 Antagonists; Immunoblotting; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neostriatum; Nerve Tissue Proteins; Neurons; Neurotensin; Phosphoproteins; Piperidines; Pyrazoles; Quinolines; Raclopride; Receptors, Neurotensin; Signal Transduction; Tetrodotoxin; Threonine; Time Factors | 2003 |
Beta-lactotensin and neurotensin rapidly reduce serum cholesterol via NT2 receptor.
Topics: Animals; Cholesterol; Dopamine Antagonists; Male; Mice; Mice, Inbred ICR; Neurotensin; Oligopeptides; Piperidines; Raclopride; Receptors, Neurotensin | 2003 |
Low-affinity neurotensin receptor (NTS2) signaling: internalization-dependent activation of extracellular signal-regulated kinases 1/2.
Topics: Animals; Base Sequence; Calcium; CHO Cells; Cricetinae; DNA Primers; Enzyme Activation; Histamine H1 Antagonists; Kinetics; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Neurotensin; Piperidines; Rats; Receptors, Neurotensin; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Transfection | 2004 |
Identification and functional characterization of a 5-transmembrane domain variant isoform of the NTS2 neurotensin receptor in rat central nervous system.
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Western; Brain; Cell Line; Central Nervous System; CHO Cells; COS Cells; Cricetinae; Densitometry; Dimerization; DNA, Complementary; Dose-Response Relationship, Drug; Epitopes; Immunoblotting; Immunohistochemistry; Immunoprecipitation; Inhibitory Concentration 50; Ligands; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Molecular Sequence Data; Neurotensin; Peptides; Piperidines; Protein Binding; Protein Isoforms; Protein Structure, Tertiary; Rats; Receptors, Neurotensin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Homology, Amino Acid; Signal Transduction; Spinal Cord; Time Factors; Tissue Distribution; Transfection | 2005 |
Potent spinal analgesia elicited through stimulation of NTS2 neurotensin receptors.
Topics: Analgesics; Animals; Ganglia, Spinal; Hot Temperature; In Vitro Techniques; Injections, Spinal; Lumbar Vertebrae; Models, Animal; Neurotensin; Pain; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Spinal Cord; Tail | 2005 |
Interactions between NTS2 neurotensin and opioid receptors on two nociceptive responses assessed on the hot plate test in mice.
Topics: Analgesia; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Histamine H1 Antagonists, Non-Sedating; Injections, Intraventricular; Ligands; Male; Mice; Morphine; Neurotensin; Pain Threshold; Piperidines; Pyrazoles; Quinolines; Reaction Time; Receptors, Neurotensin; Receptors, Opioid | 2006 |
Evidence for a role of NTS2 receptors in the modulation of tonic pain sensitivity.
Topics: Animals; Formaldehyde; Histamine H1 Antagonists, Non-Sedating; Inflammation; Male; Neurotensin; Pain; Peptide Fragments; Piperidines; Posterior Horn Cells; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Spinal Nerves; Time Factors | 2009 |
NT69L, a novel analgesic, shows synergy with morphine.
Topics: Analgesics; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Synergism; Hot Temperature; Male; Morphine; Neurotensin; Pain; Pain Measurement; Peptide Fragments; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Time Factors | 2009 |
Neurotensin is a regulator of insulin secretion in pancreatic beta-cells.
Topics: Animals; Calcium Signaling; Cell Line; Cyclic AMP-Dependent Protein Kinases; Cytoprotection; Enzyme Activation; Insulin; Insulin Secretion; Insulin-Secreting Cells; Neurotensin; Piperidines; Protein Kinase C-alpha; Protein Kinase C-epsilon; Pyrazoles; Quinolines; Rats; Receptors, Neurotensin | 2010 |
Neurotensin decreases high affinity [3H]-ouabain binding to cerebral cortex membranes.
Topics: Animals; Cerebral Cortex; Male; Neurotensin; Ouabain; Piperidines; Protein Binding; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin | 2011 |
Neurotensin inhibits background K+ channels and facilitates glutamatergic transmission in rat spinal cord dorsal horn.
Topics: Animals; Benzophenanthridines; Excitatory Postsynaptic Potentials; Glutamic Acid; Neurotensin; Oligopeptides; Patch-Clamp Techniques; Pertussis Toxin; Piperidines; Posterior Horn Cells; Potassium Channels; Pyrazoles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Neurotensin; Signal Transduction; Synapses; Synaptic Transmission | 2011 |
In vivo investigations of neurotensin receptors in adipocytes, hepatocytes and enterocytes of rat.
Topics: Adipocytes; Adipose Tissue; Animals; Antigen-Antibody Reactions; Cell Membrane; Enterocytes; Hepatocytes; Histamine H1 Antagonists, Non-Sedating; Intestine, Small; Iodine Radioisotopes; Isotope Labeling; Liver; Male; Neurotensin; Piperidines; Pyrazoles; Quinolines; Rats; Rats, Wistar; Receptors, Neurotensin | 2011 |
NTS1 and NTS2 mediate analgesia following neurotensin analog treatment in a mouse model for visceral pain.
Topics: Acetic Acid; Analgesia; Analysis of Variance; Animals; Behavior, Animal; Histamine H1 Antagonists; Mice; Mice, Knockout; Neurotensin; Pain; Pain Measurement; Peptide Fragments; Piperidines; Receptors, Neurotensin | 2012 |