Page last updated: 2024-09-04

leucine thiorphan and substance p

leucine thiorphan has been researched along with substance p in 4 studies

Compound Research Comparison

Studies
(leucine thiorphan)
Trials
(leucine thiorphan)
Recent Studies (post-2010)
(leucine thiorphan)
Studies
(substance p)
Trials
(substance p)
Recent Studies (post-2010) (substance p)
60017,2892772,010

Protein Interaction Comparison

ProteinTaxonomyleucine thiorphan (IC50)substance p (IC50)
Substance-P receptorRattus norvegicus (Norway rat)0.0005
Substance-K receptorRattus norvegicus (Norway rat)0.2
Substance-K receptorHomo sapiens (human)0.2455
Substance-P receptorHomo sapiens (human)0.0011
Neuromedin-K receptorHomo sapiens (human)0.125
Substance-K receptorMesocricetus auratus (golden hamster)0.148

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19904 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Borson, DB; Nadel, JA; Sekizawa, K; Tamaoki, J1
Borson, DB; Graf, PD; Kohrogi, H; Nadel, JA; Sekizawa, K1
Borson, DB; Djokic, TD; Nadel, JA; Sekizawa, K1
Borson, DB; Djokic, TD; Dusser, DJ; Graf, PD; Nadel, JA; Sekizawa, K1

Other Studies

4 other study(ies) available for leucine thiorphan and substance p

ArticleYear
Enkephalinase inhibitor potentiates substance P- and electrically induced contraction in ferret trachea.
    Journal of applied physiology (Bethesda, Md. : 1985), 1987, Volume: 63, Issue:4

    Topics: Airway Resistance; Amino Acids, Sulfur; Animals; Electric Stimulation; Ferrets; In Vitro Techniques; Metalloendopeptidases; Neprilysin; Substance P; Thiorphan; Tiopronin; Trachea

1987
Neutral endopeptidase inhibitors potentiate substance P- and capsaicin-induced cough in awake guinea pigs.
    The Journal of clinical investigation, 1988, Volume: 82, Issue:6

    Topics: Animals; Capsaicin; Cough; Drug Synergism; Glycopeptides; Guinea Pigs; Male; Neprilysin; Substance P; Thiorphan

1988
Neutral endopeptidase inhibitors potentiate substance P-induced contraction in gut smooth muscle.
    The American journal of physiology, 1989, Volume: 256, Issue:1 Pt 1

    Topics: Animals; Drug Synergism; Duodenum; Endopeptidases; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Female; Ferrets; Glycopeptides; Ileum; Intestines; Male; Muscle Contraction; Protease Inhibitors; Rats; Substance P; Thiorphan

1989
Inhibitors of neutral endopeptidase potentiate electrically and capsaicin-induced noncholinergic contraction in guinea pig bronchi.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Bronchi; Capsaicin; Electric Stimulation; Glycopeptides; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Neprilysin; Substance P; Thiorphan

1989