Page last updated: 2024-09-03

lestaurtinib and staurosporine aglycone

lestaurtinib has been researched along with staurosporine aglycone in 2 studies

Compound Research Comparison

Studies
(lestaurtinib)
Trials
(lestaurtinib)
Recent Studies (post-2010)
(lestaurtinib)
Studies
(staurosporine aglycone)
Trials
(staurosporine aglycone)
Recent Studies (post-2010) (staurosporine aglycone)
12412637390175

Protein Interaction Comparison

ProteinTaxonomylestaurtinib (IC50)staurosporine aglycone (IC50)
B2 bradykinin receptorCavia porcellus (domestic guinea pig)8
Serine/threonine-protein kinase D3Homo sapiens (human)2.45
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.83
Beta-lactamaseEscherichia coli K-128
Protein kinase C gamma typeHomo sapiens (human)2.45
Protein kinase C beta typeHomo sapiens (human)2.45
Zinc finger protein GLI1Homo sapiens (human)1.8
Zinc finger protein GLI2Homo sapiens (human)2.7
Malate dehydrogenaseThermus thermophilus8
Cyclin-dependent kinase 4Homo sapiens (human)0.83
Protein kinase C alpha typeHomo sapiens (human)2.45
Chymotrypsinogen BHomo sapiens (human)10
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)8
G1/S-specific cyclin-D1Homo sapiens (human)0.83
Protein kinase C eta typeHomo sapiens (human)2.45
G1/S-specific cyclin-E1Homo sapiens (human)0.83
Cyclin-dependent kinase 2Homo sapiens (human)0.83
Protein kinase C iota typeHomo sapiens (human)2.45
Tyrosine-protein kinase JAK3Homo sapiens (human)0.061
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)0.1083
Protein kinase C epsilon typeHomo sapiens (human)2.45
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)0.0935
Protein kinase C theta typeHomo sapiens (human)2.45
Protein kinase C zeta typeHomo sapiens (human)2.45
Protein kinase C delta typeHomo sapiens (human)2.45
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)0.184
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)0.184
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)0.184
Serine/threonine-protein kinase D1Homo sapiens (human)2.45
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)0.0787
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)0.184

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hudkins, RL; Miknyoczki, SJ; Ruggeri, BA; Singh, J1
Courts, C; Gallala, H; Janzen, V; Kraus, D; Nowak, M; Perner, S; Probstmeier, R; Veit, N; Winter, J1

Reviews

1 review(s) available for lestaurtinib and staurosporine aglycone

ArticleYear
Role of neurotrophin-trk interactions in oncology: the anti-tumor efficacy of potent and selective trk tyrosine kinase inhibitors in pre-clinical tumor models.
    Current medicinal chemistry, 1999, Volume: 6, Issue:9

    Topics: Animals; Antineoplastic Agents; Carbazoles; Disease Models, Animal; Drug Design; Female; Furans; Humans; Indole Alkaloids; Indoles; Mice; Nerve Growth Factors; Nerve Tissue Proteins; Protein-Tyrosine Kinases; Signal Transduction

1999

Other Studies

1 other study(ies) available for lestaurtinib and staurosporine aglycone

ArticleYear
Staurosporine analogs promote distinct patterns of process outgrowth and polyploidy in small cell lung carcinoma cells.
    Tumour biology : the journal of the International Society for Oncodevelopmental Biology and Medicine, 2015, Volume: 36, Issue:4

    Topics: Carbazoles; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Furans; Humans; Indole Alkaloids; Polyploidy; Signal Transduction; Small Cell Lung Carcinoma; Staurosporine

2015