Page last updated: 2024-09-03

lestaurtinib and panobinostat

lestaurtinib has been researched along with panobinostat in 2 studies

Compound Research Comparison

Studies
(lestaurtinib)
Trials
(lestaurtinib)
Recent Studies (post-2010)
(lestaurtinib)
Studies
(panobinostat)
Trials
(panobinostat)
Recent Studies (post-2010) (panobinostat)
124126367895593

Protein Interaction Comparison

ProteinTaxonomylestaurtinib (IC50)panobinostat (IC50)
Histone deacetylase 8Schistosoma mansoni0.45
Histone deacetylase 3Homo sapiens (human)0.2031
Bromodomain-containing protein 4Homo sapiens (human)0.005
Cytochrome P450 3A5Homo sapiens (human)0.0033
Histone deacetylase 4Homo sapiens (human)0.3792
Histone deacetylase 1Homo sapiens (human)0.181
Histone deacetylase 7Homo sapiens (human)0.9434
Histone deacetylase 2Homo sapiens (human)0.2527
Polyamine deacetylase HDAC10Homo sapiens (human)0.007
Histone deacetylase 11 Homo sapiens (human)0.8396
Histone deacetylase 8Homo sapiens (human)0.46
Histone deacetylase 6Homo sapiens (human)0.2307
Histone deacetylase 9Homo sapiens (human)0.5825
Histone deacetylase 5Homo sapiens (human)0.3424
Histone deacetylase Plasmodium falciparum (malaria parasite P. falciparum)0.0025
Nuclear receptor corepressor 2Homo sapiens (human)0.002

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Evans, L1
Chen, E; Debnath, A; Ehrenkaufer, GM; Kangussu-Marcolino, MM; Singh, U1

Other Studies

2 other study(ies) available for lestaurtinib and panobinostat

ArticleYear
The American Society of Hematology--46th Annual Meeting and Exposition. HDAC, Flt and farnesyl transferase inhibitors.
    IDrugs : the investigational drugs journal, 2005, Volume: 8, Issue:1

    Topics: Alkyl and Aryl Transferases; Carbazoles; Farnesyltranstransferase; fms-Like Tyrosine Kinase 3; Furans; Hematology; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Hydroxamic Acids; Indoles; Panobinostat; Proto-Oncogene Proteins; Quinolones; Receptor Protein-Tyrosine Kinases; Societies, Medical; United States

2005
Identification of plicamycin, TG02, panobinostat, lestaurtinib, and GDC-0084 as promising compounds for the treatment of central nervous system infections caused by the free-living amebae Naegleria, Acanthamoeba and Balamuthia.
    International journal for parasitology. Drugs and drug resistance, 2019, Volume: 11

    Topics: Acanthamoeba; Amebiasis; Amoebozoa; Antiprotozoal Agents; Carbazoles; Cell Culture Techniques; Central Nervous System Protozoal Infections; Culture Media; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Enzyme Inhibitors; Furans; Heterocyclic Compounds, 4 or More Rings; Inhibitory Concentration 50; Naegleria; Oxazines; Panobinostat; Plicamycin; Pyrimidines

2019