Page last updated: 2024-09-03

lestaurtinib and chir 99021

lestaurtinib has been researched along with chir 99021 in 1 studies

Compound Research Comparison

Studies
(lestaurtinib)
Trials
(lestaurtinib)
Recent Studies (post-2010)
(lestaurtinib)
Studies
(chir 99021)
Trials
(chir 99021)
Recent Studies (post-2010) (chir 99021)
12412632721258

Protein Interaction Comparison

ProteinTaxonomylestaurtinib (IC50)chir 99021 (IC50)
G2/mitotic-specific cyclin-B2Homo sapiens (human)8.8
Cyclin-dependent kinase 1Homo sapiens (human)8.8
G2/mitotic-specific cyclin-B1Homo sapiens (human)8.8
Glycogen synthase kinase-3 alphaHomo sapiens (human)0.0089
Glycogen synthase kinase-3 betaHomo sapiens (human)0.0133
G2/mitotic-specific cyclin-B3Homo sapiens (human)8.8

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Abagyan, R; Balboni, B; Cavalli, A; Demuro, S; Di Martino, RMC; Giabbai, B; Girotto, S; Ortega, JA; Russo, D; Sauvey, C; Shi, D; Storici, P; Tripathi, SK1

Other Studies

1 other study(ies) available for lestaurtinib and chir 99021

ArticleYear
ARN25068, a versatile starting point towards triple GSK-3β/FYN/DYRK1A inhibitors to tackle tau-related neurological disorders.
    European journal of medicinal chemistry, 2022, Feb-05, Volume: 229

    Topics: Binding Sites; Drug Evaluation, Preclinical; Dyrk Kinases; Glycogen Synthase Kinase 3 beta; Humans; Microtubules; Models, Molecular; Neurofibrillary Tangles; Neuroprotective Agents; Phosphorylation; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-fyn; Structure-Activity Relationship; tau Proteins; Tauopathies

2022