Page last updated: 2024-08-25

lecimibide and urea

lecimibide has been researched along with urea in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (75.00)18.2507
2000's3 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Harte, RA; Jackson, B; Suckling, KE; Yeaman, SJ2
Brogdon, B; Lai, CM; Pieniaszek, HJ; Quon, CY1
Billheimer, JT; Gillies, PJ; Higley, CA; Johnson, AL; Maduskuie, TP; Pennev, P; Robinson, CS; Wexler, RR; Wilde, RG1
Connell, JM; Crouse, JR; Gillies, PJ; Hainer, JW; Hunt, TL; Jenkins, RM; Livak, KJ; Shand, DL; Terry, JG; Zyruk, H1
Barrett, PH; Billheimer, JT; Gillies, PJ; Huff, MW; Telford, DE1
Anderson, M; Bousley, RF; Hamelehle, KL; Homan, R; Julian, TN; Krause, BR; Picard, JA; Rashidbaigi, ZA; Sliskovic, DR; Stanfield, RL1
Botham, KM; Hoang, VQ; Pearce, NJ; Suckling, KE1
Barrett, PH; Burnett, JR; Huff, MW; Kleinstiver, SJ; Telford, DE; Wilcox, LJ1
Chao, YS; Detmers, PA; Hernandez, M; Kim, D; Montenegro, J; Sparrow, C; Steiner, M; Wright, SD1
Horiuchi, S; Miyazaki, A1
Brown, WJ; Schmidt, JA1

Reviews

1 review(s) available for lecimibide and urea

ArticleYear
[ACAT inhibitors].
    Nihon rinsho. Japanese journal of clinical medicine, 2001, Volume: 59 Suppl 3

    Topics: Anilides; Animals; Arteriosclerosis; Benzofurans; Cholesterol Esters; Cyclohexanes; Dioxanes; Endothelium, Vascular; Humans; Hyperlipidemias; Imidazoles; Intestine, Small; Liver; Organ Specificity; Phenylurea Compounds; Sterol O-Acyltransferase; Urea

2001

Trials

1 trial(s) available for lecimibide and urea

ArticleYear
Effect of the acyl-CoA:cholesterol acyltransferase inhibitor DuP 128 on cholesterol absorption and serum cholesterol in humans.
    Clinical pharmacology and therapeutics, 1994, Volume: 56, Issue:1

    Topics: Adult; Base Sequence; Carbon Radioisotopes; Cholesterol; Humans; Imidazoles; Intestinal Absorption; Male; Molecular Sequence Data; Sterol O-Acyltransferase; Tritium; Urea

1994

Other Studies

10 other study(ies) available for lecimibide and urea

ArticleYear
Effect of membrane environment on inhibition of acyl-CoA:cholesterol acyltransferase by a range of synthetic inhibitors.
    Biochimica et biophysica acta, 1995, Oct-05, Volume: 1258, Issue:3

    Topics: Anilides; Animals; Cholesterol; Detergents; Enzyme Inhibitors; Esterification; Imidazoles; Liposomes; Male; Microsomes, Liver; Oleic Acid; Oleic Acids; Phenylurea Compounds; Phosphatidylcholines; Rats; Rats, Wistar; Solubility; Sterol O-Acyltransferase; Tumor Cells, Cultured; Urea

1995
Determination of DuP 128, an ACAT inhibitor and its sulphoxide and sulphone metabolites in human plasma by liquid chromatography.
    Journal of pharmaceutical and biomedical analysis, 1994, Volume: 12, Issue:9

    Topics: Administration, Oral; Anticholesteremic Agents; Chromatography, High Pressure Liquid; Fluorescence; Humans; Imidazoles; Male; Sterol O-Acyltransferase; Sulfones; Sulfoxides; Urea

1994
Acyl CoA:cholesterol acyltransferase (ACAT) inhibitors: synthesis and structure-activity relationship studies of a new series of trisubstituted imidazoles.
    Journal of medicinal chemistry, 1994, Oct-14, Volume: 37, Issue:21

    Topics: Animals; Anticholesteremic Agents; Cholesterol; Cricetinae; Imidazoles; Male; Mesocricetus; Microsomes, Liver; Molecular Structure; Rats; Sterol O-Acyltransferase; Structure-Activity Relationship; Urea

1994
Inhibition of hepatic ACAT decreases ApoB secretion in miniature pigs fed a cholesterol-free diet.
    Arteriosclerosis and thrombosis : a journal of vascular biology, 1994, Volume: 14, Issue:9

    Topics: Animals; Apolipoproteins B; Cholesterol; Cholesterol, Dietary; Cholesterol, LDL; Imidazoles; Kinetics; Lipoproteins, VLDL; Liver; Sterol O-Acyltransferase; Swine; Swine, Miniature; Triglycerides; Urea

1994
Inhibitors of acyl-CoA: cholesterol O-acyl transferase (ACAT) as hypocholesterolemic agents. 6. The first water-soluble ACAT inhibitor with lipid-regulating activity.
    Journal of medicinal chemistry, 1994, Mar-04, Volume: 37, Issue:5

    Topics: Absorption; Animals; Anticholesteremic Agents; Biological Availability; Carbamates; Cholesterol; Cholesterol Esters; Hydrogen-Ion Concentration; Hypercholesterolemia; Imidazoles; Lipids; Liver; Microsomes, Liver; Phenylurea Compounds; Rats; Solubility; Sterol O-Acyltransferase; Urea; Water

1994
The regulation of bile acid synthesis in cultured hamster hepatocytes.
    Biochemical Society transactions, 1993, Volume: 21 ( Pt 3), Issue:3

    Topics: Animals; Bile Acids and Salts; Cells, Cultured; Chenodeoxycholic Acid; Cholestyramine Resin; Cholic Acid; Cholic Acids; Cricetinae; Hydroxycholesterols; Imidazoles; Lipoproteins, LDL; Liver; Lovastatin; Male; Mesocricetus; Mevalonic Acid; Taurocholic Acid; Urea

1993
Differences in the potency of ACAT inhibitors in two assay systems.
    Biochemical Society transactions, 1993, Volume: 21 ( Pt 3), Issue:3

    Topics: Acyl Coenzyme A; Anilides; Animals; Carbon Radioisotopes; Imidazoles; Indicators and Reagents; Kinetics; Male; Microsomes, Liver; Radioisotope Dilution Technique; Rats; Rats, Sprague-Dawley; Sterol O-Acyltransferase; Urea

1993
Inhibition of cholesterol esterification by DuP 128 decreases hepatic apolipoprotein B secretion in vivo: effect of dietary fat and cholesterol.
    Biochimica et biophysica acta, 1998, Jul-31, Volume: 1393, Issue:1

    Topics: Animals; Anticholesteremic Agents; Apolipoproteins B; Cholesterol, Dietary; Dietary Fats; Down-Regulation; Enzyme Inhibitors; Imidazoles; Intestines; Lipoproteins, VLDL; Liver; Sterol O-Acyltransferase; Swine; Swine, Miniature; Urea

1998
Intestinal absorption of cholesterol is mediated by a saturable, inhibitable transporter.
    Biochimica et biophysica acta, 2000, Jul-19, Volume: 1486, Issue:2-3

    Topics: Animals; Anticholesteremic Agents; Bile Acids and Salts; Binding Sites; Biological Transport; Cholesterol, Dietary; Cricetinae; Dogs; Down-Regulation; Enzyme Inhibitors; Imidazoles; Intestinal Absorption; Intestinal Mucosa; Male; Mesocricetus; Mice; Microvilli; Molecular Structure; Rats; Saponins; Simvastatin; Species Specificity; Spirostans; Structure-Activity Relationship; Tritium; Urea

2000
Use of acyltransferase inhibitors to block vesicular traffic between the ER and Golgi complex.
    Methods in enzymology, 2005, Volume: 404

    Topics: 1-Acylglycerophosphocholine O-Acyltransferase; Acyltransferases; Anilides; Animals; Cells, Cultured; COP-Coated Vesicles; Endoplasmic Reticulum; Golgi Apparatus; Imidazoles; Intracellular Membranes; Protein Transport; Rats; Sterol O-Acyltransferase; Urea

2005