Page last updated: 2024-09-05

lasofoxifene and palbociclib

lasofoxifene has been researched along with palbociclib in 1 studies

Compound Research Comparison

Studies
(lasofoxifene)
Trials
(lasofoxifene)
Recent Studies (post-2010)
(lasofoxifene)
Studies
(palbociclib)
Trials
(palbociclib)
Recent Studies (post-2010) (palbociclib)
881424911126864

Protein Interaction Comparison

ProteinTaxonomylasofoxifene (IC50)palbociclib (IC50)
Chain B, Cell division protein kinase 6Homo sapiens (human)0.015
Chain B, Cell division protein kinase 6Homo sapiens (human)0.015
Cyclin-T1Homo sapiens (human)1.5085
Cyclin-KHomo sapiens (human)1.207
Cyclin-dependent kinase 1Homo sapiens (human)9.8
Cyclin-dependent kinase 4Homo sapiens (human)0.0109
G2/mitotic-specific cyclin-B1Homo sapiens (human)9.8
Cyclin-A2Homo sapiens (human)2.2042
AcetylcholinesteraseMus musculus (house mouse)0.021
G1/S-specific cyclin-D1Homo sapiens (human)0.0115
G1/S-specific cyclin-E1Homo sapiens (human)9.15
Cyclin-dependent kinase 2Homo sapiens (human)4.1887
G1/S-specific cyclin-D2Homo sapiens (human)0.0127
G1/S-specific cyclin-D3Homo sapiens (human)0.0194
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)3.48
Cyclin-dependent kinase 9Homo sapiens (human)1.1821
Tyrosine-protein kinase JAK3Homo sapiens (human)0.0631
Cyclin-dependent kinase 6Homo sapiens (human)0.018

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Chang, YF; Fanning, SW; Green, B; Greene, GL; Greene, ME; Komm, B; Kurleto, JD; Lainé, M; Phung, L1

Other Studies

1 other study(ies) available for lasofoxifene and palbociclib

ArticleYear
Lasofoxifene as a potential treatment for therapy-resistant ER-positive metastatic breast cancer.
    Breast cancer research : BCR, 2021, 05-12, Volume: 23, Issue:1

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Disease Models, Animal; Estrogen Receptor alpha; Female; Fulvestrant; Humans; MCF-7 Cells; Mice; Mutation; Neoplasm Metastasis; Piperazines; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Pyridines; Pyrrolidines; Receptors, Estrogen; Selective Estrogen Receptor Modulators; Tetrahydronaphthalenes; Treatment Outcome

2021