Page last updated: 2024-09-05

lapatinib and su 5402

lapatinib has been researched along with su 5402 in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(su 5402)
Trials
(su 5402)
Recent Studies (post-2010) (su 5402)
1,9193051,442191077

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)su 5402 (IC50)
Epidermal growth factor receptorHomo sapiens (human)0.1867
Platelet-derived growth factor receptor betaHomo sapiens (human)0.2675
Fibroblast growth factor receptor 1Homo sapiens (human)2.0262
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.1867
Fibroblast growth factor receptor 1Mus musculus (house mouse)10
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.1136
Vascular endothelial growth factor receptor 1Mus musculus (house mouse)0.4
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.02

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, G; Chen, S; Chen, Y; Ding, J; Meng, L; Tong, L; Wang, J; Wang, X; Xie, Y; Yang, C1

Other Studies

1 other study(ies) available for lapatinib and su 5402

ArticleYear
Discovery and bioactivity of 4-(2-arylpyrido[3',2':3,4]pyrrolo[1,2-f][1,2,4]triazin-4-yl) morpholine derivatives as novel PI3K inhibitors.
    Bioorganic & medicinal chemistry letters, 2012, Jan-01, Volume: 22, Issue:1

    Topics: Antineoplastic Agents; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Drug Design; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Furans; Humans; Inhibitory Concentration 50; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Pyrimidines

2012