Page last updated: 2024-09-05

lapatinib and purvalanol b

lapatinib has been researched along with purvalanol b in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(purvalanol b)
Trials
(purvalanol b)
Recent Studies (post-2010) (purvalanol b)
1,9193051,44231013

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)purvalanol b (IC50)
G2/mitotic-specific cyclin-B2Homo sapiens (human)0.006
G1/S-specific cyclin-E2Homo sapiens (human)0.009
Cyclin-dependent kinase 1Saccharomyces cerevisiae S288C1.2
Insulin receptorHomo sapiens (human)2.2
Tyrosine-protein kinase LckHomo sapiens (human)0.006
Cyclin-dependent kinase 1Homo sapiens (human)0.006
G2/mitotic-specific cyclin-B1Homo sapiens (human)0.006
G2/mitotic-specific cyclin-BMarthasterias glacialis (spiny starfish)0.006
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)3.8
Cyclin-A2Homo sapiens (human)0.006
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)3.8
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)3.8
G1/S-specific cyclin-E1Homo sapiens (human)0.009
Cyclin-dependent kinase 2Homo sapiens (human)0.0072
Mitogen-activated protein kinase 3 Homo sapiens (human)3.3165
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.006
Cyclin-A1Homo sapiens (human)0.006
Cyclin-dependent-like kinase 5 Homo sapiens (human)0.006
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)0.006
Cdc2Patiria pectinifera0.15
G2/mitotic-specific cyclin-B3Homo sapiens (human)0.006
Cyclin-dependent kinase 1Oryzias latipes (Japanese medaka)0.006

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

1 other study(ies) available for lapatinib and purvalanol b

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013