Page last updated: 2024-09-05

lapatinib and pd168393

lapatinib has been researched along with pd168393 in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(pd168393)
Trials
(pd168393)
Recent Studies (post-2010) (pd168393)
1,9193051,44261033

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)pd168393 (IC50)
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)1.0702
Epidermal growth factor receptorHomo sapiens (human)0.0143
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.0334
Tyrosine-protein kinase FynHomo sapiens (human)0.1543
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.073
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)0.0011
Tyrosine-protein kinase BlkHomo sapiens (human)5.47
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)0.5757
Tyrosine-protein kinase JAK3Homo sapiens (human)3.14
Tyrosine-protein kinase BTKHomo sapiens (human)5.83
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)0.0047

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Da Settimo, F; La Motta, C; Martinelli, A; Nerini, E; Sartini, S; Tuccinardi, T1

Other Studies

1 other study(ies) available for lapatinib and pd168393

ArticleYear
Computational studies of epidermal growth factor receptor: docking reliability, three-dimensional quantitative structure-activity relationship analysis, and virtual screening studies.
    Journal of medicinal chemistry, 2009, Feb-26, Volume: 52, Issue:4

    Topics: Computational Biology; Computer Simulation; Databases, Protein; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Protein Binding; Quantitative Structure-Activity Relationship

2009