Page last updated: 2024-09-05

lapatinib and pd 173955

lapatinib has been researched along with pd 173955 in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(pd 173955)
Trials
(pd 173955)
Recent Studies (post-2010) (pd 173955)
1,9193051,44229013

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)pd 173955 (IC50)
Tyrosine-protein kinase ABL1Homo sapiens (human)0.0193
Carbonic anhydrase 2Homo sapiens (human)0.028
Tyrosine-protein kinase LckHomo sapiens (human)0.5889
NucleophosminHomo sapiens (human)2.75
Platelet-derived growth factor receptor betaHomo sapiens (human)0.9199
Dihydrofolate reductaseEscherichia coli K-120.028
Breakpoint cluster region proteinHomo sapiens (human)0.002
Fibroblast growth factor receptor 1Homo sapiens (human)0.8379
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.5928
Platelet-derived growth factor receptor alphaHomo sapiens (human)1.66
Cyclin-dependent kinase 2Homo sapiens (human)0.028
Ephrin type-A receptor 2Homo sapiens (human)0.0079
ALK tyrosine kinase receptorHomo sapiens (human)2.75

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ciceri, P; Davis, MI; Herrgard, S; Hocker, M; Hunt, JP; Pallares, G; Treiber, DK; Wodicka, LM; Zarrinkar, PP1

Other Studies

1 other study(ies) available for lapatinib and pd 173955

ArticleYear
Comprehensive analysis of kinase inhibitor selectivity.
    Nature biotechnology, 2011, Oct-30, Volume: 29, Issue:11

    Topics: Catalysis; Drug Design; Enzyme Stability; High-Throughput Screening Assays; Humans; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Signal Transduction; Substrate Specificity

2011