Page last updated: 2024-09-05

lapatinib and melatonin

lapatinib has been researched along with melatonin in 2 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(melatonin)
Trials
(melatonin)
Recent Studies (post-2010) (melatonin)
1,9193051,44223,2681,4519,627

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)melatonin (IC50)
MyeloperoxidaseHomo sapiens (human)3
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)3.3323
Metabotropic glutamate receptor 1Rattus norvegicus (Norway rat)0.0004
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0005
Melatonin receptor type 1AHomo sapiens (human)0.0025
Melatonin receptor type 1BHomo sapiens (human)0.0035

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Ekins, S; Williams, AJ; Xu, JJ1
Cheng, H; Li, L; Liu, P; Liu, Y; Liu, Z; Rui, C; Sang, X; Tao, Z1

Other Studies

2 other study(ies) available for lapatinib and melatonin

ArticleYear
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Induction of EnR stress by Melatonin enhances the cytotoxic effect of Lapatinib in HER2-positive breast cancer.
    Cancer letters, 2021, 10-10, Volume: 518

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; DNA Damage; Endoplasmic Reticulum Stress; Female; Humans; Lapatinib; Melatonin; Mice; Mice, Nude; Protein Kinase Inhibitors; Receptor, ErbB-2; Unfolded Protein Response

2021