Page last updated: 2024-09-05

lapatinib and megestrol acetate

lapatinib has been researched along with megestrol acetate in 3 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(megestrol acetate)
Trials
(megestrol acetate)
Recent Studies (post-2010) (megestrol acetate)
1,9193051,442933228173

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)megestrol acetate (IC50)
Bile salt export pumpHomo sapiens (human)10
Glucocorticoid receptorHomo sapiens (human)0.019
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)0.019
Cytochrome P450 2C9 Homo sapiens (human)10
Androgen receptorRattus norvegicus (Norway rat)0.03
Glycine receptor subunit betaRattus norvegicus (Norway rat)0.019
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)0.019
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)0.019

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Audhuy, B; El-Hariry, I; Gardner, JP; Gore, M; Harper, P; Hawkins, R; Machiels, JP; Pétavy, F; Ravaud, A; Rolland, F; Schöffski, P; von der Maase, H; Zantl, N1
Brown, C; De Souza, P; Fox, P; Gebski, V; Hudson, M; Lee, CK; Lord, S1

Trials

2 trial(s) available for lapatinib and megestrol acetate

ArticleYear
Lapatinib versus hormone therapy in patients with advanced renal cell carcinoma: a randomized phase III clinical trial.
    Journal of clinical oncology : official journal of the American Society of Clinical Oncology, 2008, May-10, Volume: 26, Issue:14

    Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Agents, Hormonal; Carcinoma, Renal Cell; Disease-Free Survival; ErbB Receptors; Female; Humans; Immunohistochemistry; Kidney Neoplasms; Lapatinib; Male; Megestrol Acetate; Middle Aged; Prospective Studies; Protein Kinase Inhibitors; Quinazolines; Tamoxifen

2008
Markers of systemic inflammation predict survival in patients with advanced renal cell cancer.
    British journal of cancer, 2013, Jul-09, Volume: 109, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Biomarkers, Tumor; Carcinoma, Renal Cell; Female; Humans; Inflammation; Kaplan-Meier Estimate; Kidney Neoplasms; Lapatinib; Leukocyte Count; Male; Megestrol Acetate; Middle Aged; Platelet Count; Prognosis; Quinazolines; Serum Albumin; Tamoxifen; Young Adult

2013

Other Studies

1 other study(ies) available for lapatinib and megestrol acetate

ArticleYear
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012