Page last updated: 2024-09-05

lapatinib and fosbretabulin

lapatinib has been researched along with fosbretabulin in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(fosbretabulin)
Trials
(fosbretabulin)
Recent Studies (post-2010) (fosbretabulin)
1,9193051,4424970320

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)fosbretabulin (IC50)
Tubulin polymerization-promoting proteinHomo sapiens (human)1.016
Tubulin alpha-1A chainSus scrofa (pig)1.82
Tubulin beta chainSus scrofa (pig)1.9428
Tubulin beta-4A chainHomo sapiens (human)1.663
Tubulin beta chainHomo sapiens (human)1.663
ATP-dependent translocase ABCB1Homo sapiens (human)0.009
Tubulin alpha-3C chainHomo sapiens (human)1.663
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)1.08
Delta-type opioid receptorMus musculus (house mouse)1.005
Delta-type opioid receptorRattus norvegicus (Norway rat)0.81
Mu-type opioid receptorMus musculus (house mouse)1.2
Tubulin alpha-1B chainHomo sapiens (human)1.663
Tubulin alpha-4A chainHomo sapiens (human)1.663
Tubulin beta-4B chainHomo sapiens (human)1.663
Vesicular acetylcholine transporterTetronarce californica (Pacific electric ray)1.8
Tubulin beta-3 chainHomo sapiens (human)1.5801
Tubulin beta-2A chainHomo sapiens (human)1.663
Beta-tubulin Leishmania donovani1.95
Tubulin beta-8 chainHomo sapiens (human)1.663
Tubulin beta-2B chainBos taurus (cattle)1.4484
Tubulin alpha-3E chainHomo sapiens (human)1.663
Tubulin alpha-1A chainHomo sapiens (human)1.663
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)1.4928
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)1.4037
Tubulin alpha-1C chainHomo sapiens (human)1.663
Tubulin beta-6 chainHomo sapiens (human)1.663
Tubulin beta-2B chainHomo sapiens (human)1.663
Tubulin beta-1 chainHomo sapiens (human)1.6366

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bailey-Downs, LC; Bastian, A; Disch, BC; Dybdal-Hargreaves, NF; Gangjee, A; Hamel, E; Ihnat, M; Mooberry, SL; Raghavan, S; Rohena, CC; Thorpe, JE; Zhang, X1

Other Studies

1 other study(ies) available for lapatinib and fosbretabulin

ArticleYear
The design and discovery of water soluble 4-substituted-2,6-dimethylfuro[2,3-d]pyrimidines as multitargeted receptor tyrosine kinase inhibitors and microtubule targeting antitumor agents.
    Bioorganic & medicinal chemistry, 2014, Jul-15, Volume: 22, Issue:14

    Topics: Aniline Compounds; Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Female; HeLa Cells; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Microtubules; Neoplasms, Experimental; Protein Kinase Inhibitors; Pyrimidines; Receptor Protein-Tyrosine Kinases; Solubility; Structure-Activity Relationship; Water

2014