Page last updated: 2024-09-05

lapatinib and eliprodil

lapatinib has been researched along with eliprodil in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(eliprodil)
Trials
(eliprodil)
Recent Studies (post-2010) (eliprodil)
1,9193051,442104323

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)eliprodil (IC50)
N-methyl-D-aspartate receptor Sus scrofa (pig)0.0826
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)3.3
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)3.3
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)1.4
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)3.3
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)1.4

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

1 other study(ies) available for lapatinib and eliprodil

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013