Page last updated: 2024-09-05

lapatinib and doxazosin

lapatinib has been researched along with doxazosin in 2 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(doxazosin)
Trials
(doxazosin)
Recent Studies (post-2010) (doxazosin)
1,9193051,4421,372439283

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)doxazosin (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.544
Interstitial collagenaseHomo sapiens (human)5.749
Beta-2 adrenergic receptorHomo sapiens (human)2.748
Angiotensin-converting enzymeOryctolagus cuniculus (rabbit)2.2155
Alpha-1D adrenergic receptorHomo sapiens (human)0.0034
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.544
Sodium-dependent serotonin transporterHomo sapiens (human)2.688
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.368
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0007
Sodium-dependent dopamine transporter Homo sapiens (human)0.188
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.4022
Nuclear receptor subfamily 3 group C member 3 Bos taurus (cattle)2.2155

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Battastini, AM; Coelho, BP; de Quadros, AH; Gaelzer, MM; Gonçalves, CA; Guerra, MC; Guma, FC; Hoppe, JB; Salbego, CG; Setton-Avruj, P; Terra, SR; Usach, V1

Reviews

1 review(s) available for lapatinib and doxazosin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

1 other study(ies) available for lapatinib and doxazosin

ArticleYear
Phosphatidylinositol 3-Kinase/AKT Pathway Inhibition by Doxazosin Promotes Glioblastoma Cells Death, Upregulation of p53 and Triggers Low Neurotoxicity.
    PloS one, 2016, Volume: 11, Issue:4

    Topics: Animals; Antineoplastic Agents; Apoptosis; Astrocytes; Brain Neoplasms; Caspase 3; Cell Line, Tumor; Cell Proliferation; Chromones; Doxazosin; Enzyme Activation; G1 Phase Cell Cycle Checkpoints; Glioblastoma; Glycogen Synthase Kinase 3 beta; Hippocampus; Humans; Lapatinib; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Quinazolines; Rats; Rats, Wistar; Tumor Suppressor Protein p53

2016