lapatinib has been researched along with d 4476 in 1 studies
Studies (lapatinib) | Trials (lapatinib) | Recent Studies (post-2010) (lapatinib) | Studies (d 4476) | Trials (d 4476) | Recent Studies (post-2010) (d 4476) |
---|---|---|---|---|---|
1,919 | 305 | 1,442 | 18 | 0 | 13 |
Protein | Taxonomy | lapatinib (IC50) | d 4476 (IC50) |
---|---|---|---|
TGF-beta receptor type-1 | Homo sapiens (human) | 0.5 | |
Casein kinase II subunit alpha | Schizosaccharomyces pombe 972h- | 0.2 | |
Casein kinase I isoform alpha | Homo sapiens (human) | 0.3 | |
Casein kinase I isoform delta | Homo sapiens (human) | 0.2678 | |
Casein kinase I isoform epsilon | Homo sapiens (human) | 0.319 | |
Casein kinase I isoform gamma-2 | Homo sapiens (human) | 0.3 | |
Casein kinase I isoform delta | Rattus norvegicus (Norway rat) | 0.3267 | |
Serine/threonine-protein kinase D1 | Homo sapiens (human) | 9.1 | |
Mitogen-activated protein kinase 14 | Homo sapiens (human) | 4.977 | |
Casein kinase I isoform gamma-1 | Homo sapiens (human) | 0.3 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ | 1 |
1 other study(ies) available for lapatinib and d 4476
Article | Year |
---|---|
Identification of potent Yes1 kinase inhibitors using a library screening approach.
Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship | 2013 |