Page last updated: 2024-09-05

lapatinib and cyclizine

lapatinib has been researched along with cyclizine in 2 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(cyclizine)
Trials
(cyclizine)
Recent Studies (post-2010) (cyclizine)
1,9193051,4423003941

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)cyclizine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.021
Muscarinic acetylcholine receptor M2Homo sapiens (human)1.158
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.852
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.633
Alpha-2A adrenergic receptorHomo sapiens (human)1.551
Cytochrome P450 2D6Homo sapiens (human)6.2175
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.675
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.748
Alpha-1D adrenergic receptorHomo sapiens (human)1.215
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.225
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.021
Histamine H1 receptorHomo sapiens (human)0.038
D(3) dopamine receptorHomo sapiens (human)2.992
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.373
Sodium-dependent dopamine transporter Homo sapiens (human)0.763

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ekins, S; Williams, AJ; Xu, JJ1
Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR1

Other Studies

2 other study(ies) available for lapatinib and cyclizine

ArticleYear
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
    Bioorganic & medicinal chemistry, 2019, 07-15, Volume: 27, Issue:14

    Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility

2019