Page last updated: 2024-09-05

lapatinib and cl 387785

lapatinib has been researched along with cl 387785 in 2 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(cl 387785)
Trials
(cl 387785)
Recent Studies (post-2010) (cl 387785)
1,9193051,44234014

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)cl 387785 (IC50)
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)0.001
Epidermal growth factor receptorHomo sapiens (human)0.0456
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.1952
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)0.012
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)0.2

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Da Settimo, F; La Motta, C; Martinelli, A; Nerini, E; Sartini, S; Tuccinardi, T1
Abou El Ella, DA; Aly, RM; El-Motwally, AM; Ibrahim, DA1

Other Studies

2 other study(ies) available for lapatinib and cl 387785

ArticleYear
Computational studies of epidermal growth factor receptor: docking reliability, three-dimensional quantitative structure-activity relationship analysis, and virtual screening studies.
    Journal of medicinal chemistry, 2009, Feb-26, Volume: 52, Issue:4

    Topics: Computational Biology; Computer Simulation; Databases, Protein; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Protein Binding; Quantitative Structure-Activity Relationship

2009
Molecular design and synthesis of certain new quinoline derivatives having potential anticancer activity.
    European journal of medicinal chemistry, 2015, Sep-18, Volume: 102

    Topics: Antineoplastic Agents; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; ErbB Receptors; Humans; MCF-7 Cells; Molecular Structure; Protein Kinase Inhibitors; Quinolines; Structure-Activity Relationship

2015