Page last updated: 2024-09-05

lapatinib and ag 538

lapatinib has been researched along with ag 538 in 1 studies

Compound Research Comparison

Studies
(lapatinib)
Trials
(lapatinib)
Recent Studies (post-2010)
(lapatinib)
Studies
(ag 538)
Trials
(ag 538)
Recent Studies (post-2010) (ag 538)
1,9193051,44230015

Protein Interaction Comparison

ProteinTaxonomylapatinib (IC50)ag 538 (IC50)
integrase, partialHuman immunodeficiency virus 14.0628
lens epithelium-derived growth factor p75Homo sapiens (human)4.0628
alkaline phosphatase, intestinalHomo sapiens (human)3.545
alkaline phosphatase, tissue-nonspecific isozyme isoform 1 preproproteinHomo sapiens (human)9.49
intestinal alkaline phosphatase precursorMus musculus (house mouse)3.6945
alkaline phosphatase, germ cell type preproproteinHomo sapiens (human)5.59
Epidermal growth factor receptorHomo sapiens (human)2.3603
Insulin-like growth factor 1 receptorHomo sapiens (human)0.061
DNA-(apurinic or apyrimidinic site) endonucleaseHomo sapiens (human)0.28
large T antigenBetapolyomavirus macacae0.82

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, G; Chen, S; Chen, Y; Ding, J; Meng, L; Tong, L; Wang, J; Wang, X; Xie, Y; Yang, C1

Other Studies

1 other study(ies) available for lapatinib and ag 538

ArticleYear
Discovery and bioactivity of 4-(2-arylpyrido[3',2':3,4]pyrrolo[1,2-f][1,2,4]triazin-4-yl) morpholine derivatives as novel PI3K inhibitors.
    Bioorganic & medicinal chemistry letters, 2012, Jan-01, Volume: 22, Issue:1

    Topics: Antineoplastic Agents; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Drug Design; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Furans; Humans; Inhibitory Concentration 50; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Pyrimidines

2012