labetalol and urapidil

labetalol has been researched along with urapidil in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19906 (40.00)18.7374
1990's2 (13.33)18.2507
2000's4 (26.67)29.6817
2010's3 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Johans, C; Kinnunen, PK; Söderlund, T; Suomalainen, P1
Lombardo, F; Obach, RS; Waters, NJ1
Campillo, NE; Guerra, A; Páez, JA1
Bellera, CL; Bruno-Blanch, LE; Castro, EA; Duchowicz, PR; Goodarzi, M; Ortiz, EV; Pesce, G; Talevi, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
van Zwieten, PA2
Prichard, BN; Van Zwieten, PA1
Dollery, CT; Warren, JB1
Doyle, AE1
Holzmann, A; Loupal, G; Stackl, W1
Bacher, S; Beck, A; Kraupp, O; Raberger, G; Skoda, H1
Heintz, B; Kirsten, D; Kirsten, R; Nelson, K1
Arcega, JM; Bernardo, M; Blanch, J; Faulí, A; Gomar, C; Imaz, ML; Martínez-Pallí, G; Navinés, R; Santos, P1

Reviews

4 review(s) available for labetalol and urapidil

ArticleYear
Basic pharmacology of alpha-adrenoceptor antagonists and hybrid drugs.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Chemical Phenomena; Chemistry; Humans; Ketanserin; Labetalol; Piperazines

1988
The usefulness of alpha-adrenoceptor blockade in the treatment of hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Humans; Hypertension; Indoramin; Labetalol; Piperazines; Prazosin

1988
Do hybrid drugs offer an additional benefit over pure alpha 1-blockade for hypertensive patients?
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Humans; Hypertension; Ketanserin; Labetalol; Piperazines

1988
Clinical pharmacokinetics of vasodilators. Part II.
    Clinical pharmacokinetics, 1998, Volume: 35, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Alprostadil; Amrinone; Carbazoles; Carvedilol; Enoximone; Female; Humans; Iloprost; Imidazoles; Indoramin; Isosorbide Dinitrate; Labetalol; Milrinone; Molsidomine; Nitroglycerin; Nitroprusside; Oxyfedrine; Pentaerythritol Tetranitrate; Phosphodiesterase Inhibitors; Piperazines; Prazosin; Pregnancy; Propanolamines; Pyridones; Theophylline; Trapidil; Vasodilator Agents

1998

Trials

1 trial(s) available for labetalol and urapidil

ArticleYear
Comparative hemodynamic effects of urapidil and labetalol after electroconvulsive therapy.
    The journal of ECT, 2001, Volume: 17, Issue:4

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Adult; Aged; Dose-Response Relationship, Drug; Electroconvulsive Therapy; Electroencephalography; Female; Heart Rate; Humans; Hypertension; Labetalol; Male; Middle Aged; Piperazines

2001

Other Studies

10 other study(ies) available for labetalol and urapidil

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Surface activity profiling of drugs applied to the prediction of blood-brain barrier permeability.
    Journal of medicinal chemistry, 2004, Mar-25, Volume: 47, Issue:7

    Topics: Blood-Brain Barrier; Lipid Bilayers; Micelles; Permeability; Pharmaceutical Preparations; Structure-Activity Relationship; Surface Properties

2004
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Prediction of drug intestinal absorption by new linear and non-linear QSPR.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:1

    Topics: Humans; Intestinal Absorption; Linear Models; Molecular Conformation; Nonlinear Dynamics; Permeability; Pharmaceutical Preparations; Probability; Quantitative Structure-Activity Relationship; Thermodynamics

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Hybrid or multifactorial drugs in antihypertensive treatment.
    Journal of hypertension, 1990, Volume: 8, Issue:8

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Antihypertensive Agents; Drug Combinations; Humans; Hypertension; Labetalol; Piperazines; Serotonin Antagonists; Vasodilator Agents

1990
An antihypertensive drug with polyfactor mechanism of action: urapidil.
    Annales francaises d'anesthesie et de reanimation, 1989, Volume: 8, Issue:5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain Chemistry; Cats; Humans; Ketanserin; Labetalol; Piperazines; Rats; Receptors, Adrenergic; Receptors, Serotonin

1989
Intracavernous injection of vasoactive drugs in the rabbit.
    Urological research, 1988, Volume: 16, Issue:6

    Topics: Animals; Cavernous Sinus; Injections; Labetalol; Male; Papaverine; Penile Erection; Phenoxybenzamine; Phentolamine; Piperazines; Prostaglandins E; Rabbits; Vasoconstrictor Agents; Vasodilator Agents

1988
Characterization of vasodilators by comparison of their effects on blood pressure, counterregulation and myocardial oxygen demand in conscious normotensive dogs.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Blood Pressure; Dihydralazine; Dogs; Female; Heart Rate; Isosorbide Dinitrate; Labetalol; Male; Molsidomine; Myocardium; Oxygen Consumption; Piperazines; Prazosin; Pyridazines; Renin; Sydnones; Vasodilator Agents

1985