Page last updated: 2024-09-02

l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide and ketanserin

l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide has been researched along with ketanserin in 3 studies

Compound Research Comparison

Studies
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Trials
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Recent Studies (post-2010)
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Studies
(ketanserin)
Trials
(ketanserin)
Recent Studies (post-2010) (ketanserin)
138723,094335283

Protein Interaction Comparison

ProteinTaxonomyl-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide (IC50)ketanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0021
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.015
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.015
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.265
5-hydroxytryptamine receptor 1BHomo sapiens (human)6.5
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0184
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0027
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.29
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.015
D(2) dopamine receptorRattus norvegicus (Norway rat)1.8
Synaptic vesicular amine transporterHomo sapiens (human)0.18
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.001

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19901 (33.33)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clarke, KA; Parker, AJ; Stirk, GC1
Taché, Y; Yoneda, M2

Other Studies

3 other study(ies) available for l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide and ketanserin

ArticleYear
Potentiation of motoneurone excitability by combined administration of 5-HT agonist and TRH analogue.
    Neuropeptides, 1985, Volume: 6, Issue:3

    Topics: Animals; Anterior Horn Cells; Drug Synergism; Female; Fenclonine; Ketanserin; Methoxydimethyltryptamines; Methysergide; Motor Neurons; Piperidines; Pyrrolidonecarboxylic Acid; Rats; Serotonin; Stimulation, Chemical; Thyrotropin-Releasing Hormone

1985
Serotonin enhances gastric acid response to TRH analogue in dorsal vagal complex through 5-HT2 receptors in rats.
    The American journal of physiology, 1995, Volume: 269, Issue:1 Pt 2

    Topics: Animals; Drug Synergism; Gastric Acid; Globus Pallidus; Ketanserin; Male; Medulla Oblongata; Microinjections; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thyrotropin-Releasing Hormone; Vagus Nerve

1995
Potentiating interactions between medullary serotonin and thyrotropin-releasing hormone-induced gastric erosions in rats.
    Neuroscience letters, 1993, Oct-29, Volume: 161, Issue:2

    Topics: Animals; Cold Temperature; Indomethacin; Injections; Injections, Intravenous; Ketanserin; Male; Medulla Oblongata; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Restraint, Physical; Serotonin; Stomach Ulcer; Stress, Psychological; Thyrotropin-Releasing Hormone

1993