Page last updated: 2024-09-02

l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide and clonidine

l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide has been researched along with clonidine in 2 studies

Compound Research Comparison

Studies
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Trials
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Recent Studies (post-2010)
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Studies
(clonidine)
Trials
(clonidine)
Recent Studies (post-2010) (clonidine)
1387213,6922,0441,394

Protein Interaction Comparison

ProteinTaxonomyl-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide (IC50)clonidine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.101
Alpha-2B adrenergic receptorHomo sapiens (human)0.0353
Alpha-2C adrenergic receptorHomo sapiens (human)0.0115
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)5.365
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0173
Alpha-1D adrenergic receptorHomo sapiens (human)1.21
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)5.365
Alpha-2A adrenergic receptorBos taurus (cattle)0.002
NischarinRattus norvegicus (Norway rat)0.3662

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bennett, GW; Elliott, JM; Heal, DJ; Marsden, CA; Stoodley, N; Youdim, MB1
Dettmar, PW; Fortune, D; Lynn, AG; Metcalf, G; Tulloch, IF1

Other Studies

2 other study(ies) available for l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide and clonidine

ArticleYear
Behavioural and biochemical evidence for the release of noradrenaline in mouse brain by TRH and some of its biologically stable analogues.
    Neuropharmacology, 1987, Volume: 26, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Apomorphine; Behavior, Animal; Brain; Clonidine; Hypothalamus; Male; Mice; Mice, Inbred C57BL; Motor Activity; Norepinephrine; Pyrrolidonecarboxylic Acid; Thyrotropin-Releasing Hormone

1987
Neuropharmacological evaluation of RX 77368--a stabilised analogue of thyrotropin-releasing hormone (TRH).
    Regulatory peptides, 1982, Volume: 3, Issue:3-4

    Topics: Adult; Animals; Body Temperature; Clonidine; Electroencephalography; Humans; Male; Motor Activity; Pyrrolidonecarboxylic Acid; Rats; Reserpine; Sleep; Thyrotropin-Releasing Hormone; Tremorine

1982