Page last updated: 2024-09-02

l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide and carbachol

l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide has been researched along with carbachol in 5 studies

Compound Research Comparison

Studies
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Trials
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Recent Studies (post-2010)
(l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
1387213,91881968

Protein Interaction Comparison

ProteinTaxonomyl-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19903 (60.00)18.7374
1990's2 (40.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Garrick, T; Heymann-Mönnikes, I; Livingston, EH; Sierra, A; Taché, Y; Weiner, H1
Maeda-Hagiwara, M; Taché, Y1
Garrick, T; Sierra, A; Taché, Y; Veiseh, A; Weiner, H1
Garrick, T; Taché, Y; Veiseh, A; Weiner, H1
LePard, KJ; Mohammed, JR; Stephens, RL1

Other Studies

5 other study(ies) available for l-pyroglutamyl-l-histidyl-3,3-dimethylprolinamide and carbachol

ArticleYear
Bombesin microinjected into the dorsal vagal complex inhibits TRH-stimulated gastric contractility in rats.
    Brain research, 1990, Nov-19, Volume: 533, Issue:2

    Topics: Animals; Bombesin; Carbachol; Cisterna Magna; Gastrointestinal Motility; Injections; Male; Microinjections; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Stomach; Thyrotropin-Releasing Hormone; Vagus Nerve

1990
Central nervous system action of TRH to stimulate gastric emptying in rats.
    Regulatory peptides, 1987, Volume: 17, Issue:4

    Topics: Animals; Atropine; Carbachol; Gastric Emptying; Injections, Intravenous; Injections, Intraventricular; Male; Pyrrolidonecarboxylic Acid; Rats; Thyrotropin-Releasing Hormone

1987
Corticotropin-releasing factor acts centrally to suppress stimulated gastric contractility in the rat.
    Regulatory peptides, 1988, Volume: 21, Issue:1-2

    Topics: Animals; Atropine; Carbachol; Cisterna Magna; Corticotropin-Releasing Hormone; Deoxyglucose; Gastrointestinal Motility; Injections, Intravenous; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Reference Values; Thyrotropin-Releasing Hormone

1988
Corticotropin-releasing factor acts on the brain to reduce gastric contractility.
    Psychotherapy and psychosomatics, 1987, Volume: 48, Issue:1-4

    Topics: Animals; Brain; Carbachol; Corticotropin-Releasing Hormone; Deoxyglucose; Dose-Response Relationship, Drug; Gastric Emptying; Injections, Intraventricular; Pyrrolidonecarboxylic Acid; Rats; Stomach; Thyrotropin-Releasing Hormone

1987
Gastric ECL-cell hyperplasia produces enhanced basal and stimulated gastric acid output but not gastric erosion formation in the rat.
    General pharmacology, 1997, Volume: 28, Issue:3

    Topics: Animals; Carbachol; Enterochromaffin Cells; Female; Gastric Acid; Gastric Mucosa; Histamine; Hyperplasia; Indomethacin; Pentagastrin; Pyrrolidonecarboxylic Acid; Ranitidine; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Stress, Physiological; Thyrotropin-Releasing Hormone

1997