l 741626 has been researched along with piperidines in 47 studies
Studies (l 741626) | Trials (l 741626) | Recent Studies (post-2010) (l 741626) | Studies (piperidines) | Trials (piperidines) | Recent Studies (post-2010) (piperidines) |
---|---|---|---|---|---|
76 | 0 | 33 | 40,235 | 5,221 | 14,545 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (4.26) | 18.2507 |
2000's | 24 (51.06) | 29.6817 |
2010's | 20 (42.55) | 24.3611 |
2020's | 1 (2.13) | 2.80 |
Authors | Studies |
---|---|
Bowery, BJ; Bristow, L; Emms, F; Freedman, S; Kulagowski, J; Patel, S; Razzaque, Z; Seabrook, GR | 1 |
Brown, NA; McAllister, G; Milligan, G; Pillai, G; Seabrook, GR | 1 |
Dekeyne, A; Girardon, S; Millan, MJ; Monneyron, S | 1 |
Audinot, V; Cussac, D; Dubuffet, T; Gobert, A; Lavielle, G; Lejeune, F; Millan, MJ; Newman-Tancredi, A; Rivet, JM | 1 |
Brocco, M; Dekeyne, A; Dubuffet, T; Lavielle, G; Millan, MJ; Rivet, JM | 1 |
Fushiki, T; Imaizumi, M; Takeda, M | 1 |
Henry, BL; LaHoste, GJ; Marshall, JF | 1 |
Canales, JJ; Iversen, SD | 1 |
Bergeron, J; Courtney, C; McConkey, M; Melch, M; Shrikhande, A; Smith, D; Wong, SK | 1 |
Chapman, KL; Hutson, PH; Marston, D; Patel, S; Ragan, CI | 1 |
Chaperon, F; Neijt, HC; Tricklebank, MD; Unger, L | 1 |
Doleviczényi, Z; Halmos, G; Kittel, A; Lendvai, B; Répássy, G; Vizi, ES; Zelles, T | 1 |
Hattori, K; Isosaka, T; Iyo, M; Kohsaka, S; Maekawa, M; Sato, T; Uchino, S; Yagi, T; Yuasa, S | 1 |
Brotchie, JM; Millan, MJ; Visanji, NP | 1 |
Brotchie, JM; Crossman, AR; Hill, MP; McGuire, SG; Millan, MJ; Ravenscroft, P; Rochat, C | 1 |
Grundt, P; Husband, SL; Luedtke, RR; Newman, AH; Taylor, M | 1 |
Calinski, DM; Collins, GT; Grundt, P; Newman, AH; Woods, JH | 1 |
Bugert, P; Klüter, H; Schedel, A; Schloss, P | 1 |
Abe, M; Egashira, N; Fujiwara, M; Iwasaki, K; Matsushita, M; Mishima, K; Nishimura, R; Oishi, R; Okuno, R | 1 |
Loiseau, F; Millan, MJ | 1 |
Breier, M; Chang, WL; Ko, D; Swerdlow, NR; Weber, M | 1 |
Han, P; Whelan, PJ | 1 |
Chang, WL; Durbin, JP; Luedtke, RR; Mach, RH; Park, PE; Swerdlow, NR; Weber, M | 1 |
Arnt, J; Bétry, C; Etievant, A; Haddjeri, N | 1 |
Gross, G; Jongen-Rêlo, AL; Schoemaker, H; Unger, L; van Gaalen, MM | 1 |
Georgiou, J; Lee, FJ; Liu, F; Mansuy, IM; Michalon, A; Nath, A; Roder, JC; Saab, BJ; Wang, M | 1 |
Fan, X; Hess, EJ; Xu, M | 1 |
Achat-Mendes, C; Cao, J; Grundt, P; Newman, AH; Platt, DM; Spealman, RD | 1 |
Arai, Y; Kikuchi, T; Mitazaki, S; Nakagawasai, O; Nakaya, K; Niijima, F; Onogi, H; Sato, A; Tadano, T; Tan-No, K | 1 |
Breier, MR; Chang, WL; Swerdlow, NR; Yang, A | 1 |
Fone, KC; Ingallinesi, M; Loiseau, F; Marsden, CA; Millan, MJ; Watson, DJ | 1 |
Bernedo, VE; Chen, R; Kilb, W; Kolbaev, SN; Luhmann, HJ; Moser, J; Sharopov, S; Werhahn, KJ | 1 |
Ansah, OB; Pertovaara, A; Viisanen, H | 1 |
Dankoski, EC; Fish, EW; Han, JE; Hodge, CW; Krouse, MC; Malanga, CJ; Philpot, BD; Riday, TT; Walsh, PL; Wightman, RM | 1 |
Baladi, MG; France, CP; Newman, AH | 1 |
Bentley, TA; France, CP; Grenier, AE; Serafine, KM | 1 |
Davoodi, N; Langlois, X; te Riele, P | 1 |
Di Ciano, P; Diaz, J; Khaled, MA; Le Foll, B; Pushparaj, A | 1 |
Bentley, TA; France, CP; Kilborn, DJ; Koek, W; Serafine, KM | 1 |
Dulawa, SC; Ho, EV; Klenotich, SJ; McMurray, MS; Server, CH | 1 |
Newton, CL; Strange, PG; Wood, MD | 1 |
Jones, SR; McGinnis, MM; Siciliano, CA | 1 |
Cho, J; Kim, G; Kim, M; Lee, S; Won, C | 1 |
Barrett, AC; Butler, P; Caine, SB; Negus, SS; Thomsen, M | 1 |
Branco, RC; Foster, SL; Manvich, DF; Miller, GW; Newman, AH; Paladini, CA; Petko, AK; Porter-Stransky, KA; Stout, KA; Weinshenker, D | 1 |
Baumann, MH; Humburg, BA; Jordan, CJ; Newman, AH; Schindler, CW; Shaik, AB; Thorndike, EB; Xi, ZX | 1 |
King, MA; Lewis, MH; Maletz, S; Muehlmann, AM | 1 |
47 other study(ies) available for l 741626 and piperidines
Article | Year |
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Antagonism of the effects of (+)-PD 128907 on midbrain dopamine neurones in rat brain slices by a selective D2 receptor antagonist L-741,626.
Topics: Animals; Benzopyrans; Cloning, Molecular; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electrophysiology; Indoles; Male; Mesencephalon; Neurons; Oxazines; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Spiperone | 1996 |
Human D2 and D4 dopamine receptors couple through betagamma G-protein subunits to inwardly rectifying K+ channels (GIRK1) in a Xenopus oocyte expression system: selective antagonism by L-741,626 and L-745,870 respectively.
Topics: Dopamine Antagonists; Dopamine D2 Receptor Antagonists; GTP-Binding Proteins; Humans; Indoles; Ion Channel Gating; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Piperidines; Potassium Channel Blockers; Pyridines; Pyrroles; Receptors, Dopamine D4 | 1998 |
Discriminative stimulus properties of the dopamine D3 receptor agonists, PD128,907 and 7-OH-DPAT: a comparative characterization with novel ligands at D3 versus D2 receptors.
Topics: 2-Naphthylamine; Animals; Benzopyrans; Dioxins; Discrimination Learning; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Furans; Generalization, Psychological; Humans; Indoles; Ligands; Male; Oxazines; Piperazines; Piperidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Stereoisomerism; Tetrahydronaphthalenes | 2000 |
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: I. Receptorial, electrophysiological and neurochemical profile compared with GR218,231 and L741,626.
Topics: Animals; Benzopyrans; Brain; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Activation; Guanosine 5'-O-(3-Thiotriphosphate); Indoles; Male; Mitogen-Activated Protein Kinases; Norepinephrine; Oxazines; Piperidines; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Serotonin; Sulfones; Tetrahydronaphthalenes | 2000 |
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: II. Functional and behavioral profile compared with GR218,231 and L741,626.
Topics: Animals; Behavior, Animal; Benzopyrans; Body Temperature; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Indoles; Male; Mice; Motor Activity; Oxazines; Piperidines; Psychotropic Drugs; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D3; Sulfones; Tetrahydronaphthalenes | 2000 |
Effects of oil intake in the conditioned place preference test in mice.
Topics: Animals; Behavior, Animal; Benzazepines; Brain Chemistry; Conditioning, Psychological; Corn Oil; Dopamine Antagonists; Eating; Haloperidol; Indoles; Male; Mice; Piperidines; Receptors, Dopamine D1; Reward; Space Perception; Sulpiride | 2000 |
Dopamine D1 receptors synergize with D2, but not D3 or D4, receptors in the striatum without the involvement of action potentials.
Topics: Action Potentials; Amphetamine; Animals; Corpus Striatum; Dopamine Antagonists; Genes, fos; Indans; Indoles; Male; Piperidines; Proto-Oncogene Proteins c-fos; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor Cross-Talk; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Tetrodotoxin | 2000 |
Psychomotor-activating effects mediated by dopamine D(2) and D(3) receptors in the nucleus accumbens.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzopyrans; Bromocriptine; Grooming; Indoles; Motor Activity; Naphthalenes; Nucleus Accumbens; Oxazines; Piperidines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3 | 2000 |
Fully automated radioligand binding filtration assay for membrane-bound receptors.
Topics: Animals; Automation; Binding, Competitive; CHO Cells; Cricetinae; Filtration; Haloperidol; Indoles; Piperidines; Radioligand Assay; Receptors, Dopamine; Reproducibility of Results; Time Factors | 2002 |
Pharmacological and functional characterisation of dopamine D4 receptors in the rat retina.
Topics: Animals; Binding Sites; Cyclic AMP; Darkness; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Indoles; Male; Piperidines; Pyridines; Pyrroles; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Retina; Spiperone | 2003 |
Evidence for regulation of body temperature in rats by dopamine D2 receptor and possible influence of D1 but not D3 and D4 receptors.
Topics: Animals; Aporphines; Benzazepines; Benzopyrans; Body Temperature Regulation; Dopamine Agonists; Dopamine Antagonists; Hypothermia; Indoles; Oxazines; Piperazines; Piperidines; Pyridines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4 | 2003 |
D2 autoreceptor inhibition reveals oxygen-glucose deprivation-induced release of dopamine in guinea-pig cochlea.
Topics: Animals; Cochlea; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Drug Interactions; Electric Stimulation; Glucose; Guinea Pigs; Hypoxia; In Vitro Techniques; Indoles; Male; Neurons; Nomifensine; Piperidines; Receptors, Dopamine D2; Sulpiride; Tetrodotoxin; Time Factors; Tritium | 2005 |
Fyn is required for haloperidol-induced catalepsy in mice.
Topics: Animals; Anti-Dyskinesia Agents; Antipsychotic Agents; Blotting, Western; Calcium; Catalepsy; Cells, Cultured; Dopamine; Genotype; Haloperidol; Immunoblotting; Immunohistochemistry; Immunoprecipitation; In Situ Hybridization; Indoles; Mice; Neurons; Phosphorylation; Piperidines; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-fyn; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Time Factors; Tyrosine | 2006 |
Actions at sites other than D(3) receptors mediate the effects of BP897 on l-DOPA-induced hyperactivity in monoamine-depleted rats.
Topics: Adrenergic Uptake Inhibitors; Animals; Behavior, Animal; Biogenic Monoamines; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Hyperkinesis; Indoles; Levodopa; Male; Motor Activity; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Reserpine; Time Factors | 2006 |
Antiparkinsonian effects of the novel D3/D2 dopamine receptor agonist, S32504, in MPTP-lesioned marmosets: Mediation by D2, not D3, dopamine receptors.
Topics: Analysis of Variance; Animals; Antiparkinson Agents; Behavior, Animal; Callithrix; Disease Models, Animal; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Indoles; Levodopa; Motor Activity; MPTP Poisoning; Oxazines; Piperidines; Receptors, Dopamine D2; Receptors, Dopamine D3; Time Factors | 2006 |
Analogues of the dopamine D2 receptor antagonist L741,626: Binding, function, and SAR.
Topics: Cell Line; Dopamine Antagonists; Humans; Indoles; Ligands; Piperidines; Protein Binding; Receptors, Dopamine D2; Structure-Activity Relationship; Transfection | 2007 |
Food restriction alters N'-propyl-4,5,6,7-tetrahydrobenzothiazole-2,6-diamine dihydrochloride (pramipexole)-induced yawning, hypothermia, and locomotor activity in rats: evidence for sensitization of dopamine D2 receptor-mediated effects.
Topics: Animals; Benzamides; Benzothiazoles; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Food; Hypothermia; Indoles; Male; Motor Activity; Penile Erection; Physostigmine; Piperazines; Piperidines; Pramipexole; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Yawning | 2008 |
The dopamine agonism on ADP-stimulated platelets is mediated through D2-like but not D1-like dopamine receptors.
Topics: Adenosine Diphosphate; Antigens, CD; Benzazepines; Clozapine; Collagen Type IV; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Epinephrine; Flow Cytometry; Humans; Indoles; Methylphenidate; P-Selectin; Piperidines; Platelet Activation; Platelet Adhesiveness; Platelet Aggregation; Platelet Membrane Glycoproteins; Platelet-Rich Plasma; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetraspanin 30 | 2008 |
Aripiprazole inhibits marble-burying behavior via 5-hydroxytryptamine (5-HT)1A receptor-independent mechanisms.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Anxiety; Aripiprazole; Behavior, Animal; Benzodiazepines; Catalepsy; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Ketanserin; Male; Mice; Mice, Inbred ICR; Olanzapine; Piperazines; Piperidines; Postural Balance; Psychomotor Performance; Pyridines; Quinolones; Quinpirole; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
Blockade of dopamine D(3) receptors in frontal cortex, but not in sub-cortical structures, enhances social recognition in rats: similar actions of D(1) receptor agonists, but not of D(2) antagonists.
Topics: Animals; Benzazepines; Benzopyrans; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indoles; Male; Microinjections; Nitriles; Piperidines; Prefrontal Cortex; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D3; Recognition, Psychology; Social Behavior; Tetrahydroisoquinolines | 2009 |
Heritable strain differences in sensitivity to the startle gating-disruptive effects of D2 but not D3 receptor stimulation.
Topics: Acoustic Stimulation; Analysis of Variance; Animals; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gait Disorders, Neurologic; Indoles; Male; Neural Inhibition; Nucleus Accumbens; Piperidines; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sensory Gating | 2008 |
Modulation of AMPA currents by D(1)-like but not D(2)-like receptors in spinal motoneurons.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Newborn; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Agonists; In Vitro Techniques; Indoles; Ion Channel Gating; Membrane Potentials; Mice; Motor Neurons; Patch-Clamp Techniques; Piperidines; Receptors, Dopamine D1; Receptors, Dopamine D2; Spinal Cord | 2009 |
Using prepulse inhibition to detect functional D3 receptor antagonism: effects of WC10 and WC44.
Topics: Animals; Antipsychotic Agents; Apomorphine; Benzothiazoles; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Piperazines; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Startle | 2009 |
Bifeprunox and aripiprazole suppress in vivo VTA dopaminergic neuronal activity via D2 and not D3 dopamine autoreceptor activation.
Topics: Action Potentials; Analysis of Variance; Animals; Antipsychotic Agents; Aripiprazole; Benzoxazoles; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Indoles; Male; Neurons; Piperazines; Piperidines; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulfones; Tetrahydronaphthalenes; Ventral Tegmental Area | 2009 |
Amphetamine decreases behavioral inhibition by stimulation of dopamine D2, but not D3, receptors.
Topics: Amphetamine; Animals; Cell Line, Transformed; Central Nervous System Stimulants; Choice Behavior; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Humans; Indoles; Inhibition, Psychological; Male; Nitriles; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydroisoquinolines | 2009 |
NCS-1 in the dentate gyrus promotes exploration, synaptic plasticity, and rapid acquisition of spatial memory.
Topics: Animals; Cell Membrane; Dentate Gyrus; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Exploratory Behavior; In Vitro Techniques; Indoles; Learning; Long-Term Potentiation; Maze Learning; Memory; Mice; Mice, Transgenic; Models, Neurological; Motor Activity; Neuronal Calcium-Sensor Proteins; Neuropeptides; Neuropsychological Tests; Piperidines; Rats; Receptors, Dopamine D2; Recognition, Psychology; Space Perception; Time Factors | 2009 |
D2 dopamine receptor subtype-mediated hyperactivity and amphetamine responses in a model of ADHD.
Topics: Amphetamine; Animals; Attention Deficit Disorder with Hyperactivity; Benzopyrans; Corpus Striatum; Dihydroxyphenylalanine; Disease Models, Animal; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Extracellular Space; Indoles; Locomotion; Mice; Mice, Knockout; Mice, Mutant Strains; Piperidines; Pyridines; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4 | 2010 |
Dopamine D3 and D2 receptor mechanisms in the abuse-related behavioral effects of cocaine: studies with preferential antagonists in squirrel monkeys.
Topics: Animals; Behavior, Animal; Benzamides; Benzimidazoles; Benzopyrans; Cocaine-Related Disorders; Discrimination Learning; Dopamine D2 Receptor Antagonists; Indoles; Oxazines; Piperidines; Pyridines; Receptors, Dopamine D2; Receptors, Dopamine D3; Saimiri | 2010 |
p-Hydroxyamphetamine causes prepulse inhibition disruptions in mice: contribution of dopamine neurotransmission.
Topics: Animals; Benzazepines; Clozapine; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Indoles; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Oxidopamine; p-Hydroxyamphetamine; Piperazines; Piperidines; Pyridines; Pyrroles; Reflex, Startle; Salicylamides; Sensory Gating; Sympathomimetics; Synaptic Transmission | 2010 |
Disparate effects of pramipexole on locomotor activity and sensorimotor gating in Sprague-Dawley rats.
Topics: Animals; Benzothiazoles; Data Interpretation, Statistical; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Motor Activity; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Reflex, Startle; Sensory Gating | 2011 |
Selective blockade of dopamine D3 receptors enhances while D2 receptor antagonism impairs social novelty discrimination and novel object recognition in rats: a key role for the prefrontal cortex.
Topics: Animals; Benzopyrans; Discrimination, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Mice; Mice, Knockout; Microinjections; Piperidines; Prefrontal Cortex; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Recognition, Psychology | 2012 |
Dopaminergic modulation of low-Mg²⁺-induced epileptiform activity in the intact hippocampus of the newborn mouse in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Data Interpretation, Statistical; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Epilepsy; Hippocampus; Indoles; Magnesium Deficiency; Mice; Mice, Inbred C57BL; Nitriles; Piperidines; Quinpirole; Receptors, Dopamine D2; Synapses; Tetrahydroisoquinolines | 2012 |
The role of the dopamine D2 receptor in descending control of pain induced by motor cortex stimulation in the neuropathic rat.
Topics: Analysis of Variance; Animals; Deep Brain Stimulation; Disease Models, Animal; Dopamine Antagonists; Functional Laterality; Hot Temperature; Indoles; Male; Motor Cortex; Motor Neurons; Nociceptors; Pain; Pain Measurement; Peripheral Nervous System Diseases; Piperidines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reflex; Spinal Cord | 2012 |
Pathway-specific dopaminergic deficits in a mouse model of Angelman syndrome.
Topics: Angelman Syndrome; Animals; Benzazepines; Cocaine; Disease Models, Animal; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dopaminergic Neurons; Electric Stimulation; Female; Indoles; Male; Mice; Mice, Inbred C57BL; Motor Activity; Piperidines; Raclopride; Receptors, Dopamine D1; Reward; Self Stimulation; Substantia Nigra; Synaptic Transmission; Ubiquitin-Protein Ligases; Ventral Tegmental Area | 2012 |
Feeding condition and the relative contribution of different dopamine receptor subtypes to the discriminative stimulus effects of cocaine in rats.
Topics: Animals; Apomorphine; Benzamides; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Electroshock; Food Deprivation; Indoles; Lisuride; Male; Piperidines; Pyridines; Quinpirole; Raclopride; Rats, Sprague-Dawley; Reinforcement, Psychology | 2014 |
Eating high fat chow and the behavioral effects of direct-acting and indirect-acting dopamine receptor agonists in female rats.
Topics: Aging; Animals; Body Temperature; Body Weight; Cocaine; Diet, High-Fat; Dietary Fats; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Eating; Female; Hypothermia; Indoles; Insulin Resistance; Motor Activity; Piperidines; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2; Yawning | 2014 |
Examining dopamine D3 receptor occupancy by antipsychotic drugs via [3H]7-OH-DPAT ex vivo autoradiography and its cross-validation via c-fos immunohistochemistry in the rat brain.
Topics: Animals; Antipsychotic Agents; Autoradiography; Benzodiazepines; Clozapine; Dopamine Antagonists; Haloperidol; Indoles; Islands of Calleja; Male; Nitriles; Olanzapine; Piperidines; Proto-Oncogene Proteins c-fos; Radiography; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2014 |
Dopamine D3 receptors in the basolateral amygdala and the lateral habenula modulate cue-induced reinstatement of nicotine seeking.
Topics: Animals; Autoradiography; Basolateral Nuclear Complex; Conditioning, Operant; Cues; Dopamine Antagonists; Drug-Seeking Behavior; Extinction, Psychological; Habenula; Indoles; Iodine Isotopes; Male; Nicotine; Nicotinic Agonists; Nitriles; Piperidines; Rats; Rats, Long-Evans; Receptors, Dopamine D3; Reinforcement, Psychology; Self Administration; Tetrahydroisoquinolines; Tetrahydronaphthalenes | 2014 |
Drinking sucrose or saccharin enhances sensitivity of rats to quinpirole-induced yawning.
Topics: Administration, Oral; Animals; Behavior, Animal; Benzamides; Dietary Sucrose; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drinking; Drug Administration Schedule; Drug Interactions; Indoles; Male; Non-Nutritive Sweeteners; Piperidines; Pyridines; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D3; Saccharin; Yawning | 2015 |
Dopamine D2/3 receptor antagonism reduces activity-based anorexia.
Topics: Amisulpride; Animals; Anorexia Nervosa; Benzodiazepines; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Eating; Female; Indoles; Mice; Mice, Inbred BALB C; Motor Activity; Nitriles; Olanzapine; Piperidines; Receptors, Dopamine D3; Salicylamides; Sulpiride; Tetrahydroisoquinolines; Weight Loss | 2015 |
Examining the Effects of Sodium Ions on the Binding of Antagonists to Dopamine D2 and D3 Receptors.
Topics: Animals; Binding, Competitive; Biphenyl Compounds; Cell Line, Tumor; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Indans; Indoles; Ions; Ligands; Molecular Structure; Mutation; Nitriles; Piperazines; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Sf9 Cells; Sodium; Spodoptera; Tetrahydroisoquinolines | 2016 |
Dopamine D3 autoreceptor inhibition enhances cocaine potency at the dopamine transporter.
Topics: Animals; Autoreceptors; Cocaine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Synergism; Female; Indoles; Male; Mice; Mice, Inbred C57BL; Nitriles; Piperidines; Raclopride; Receptors, Dopamine D2; Receptors, Tumor Necrosis Factor, Member 25; Sex Characteristics; Tetrahydroisoquinolines | 2016 |
Dopamine D3 receptor-modulated neuroprotective effects of lisuride.
Topics: Animals; ATPases Associated with Diverse Cellular Activities; Biphenyl Compounds; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Indoles; Lisuride; Male; Metalloendopeptidases; Mice; Mitochondria; Neuroprotective Agents; Oxidopamine; Piperazines; Piperidines; Primary Cell Culture; Receptors, Dopamine D3; Tyrosine 3-Monooxygenase | 2017 |
Effects of Acute and Chronic Treatments with Dopamine D
Topics: Aminopyridines; Animals; Benzamides; Choice Behavior; Cocaine; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Tolerance; Food; Indoles; Ligands; Male; Morpholines; Piperidines; Pyridines; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology | 2017 |
Selective D
Topics: Action Potentials; Animals; Benzamides; Central Nervous System Sensitization; Cocaine; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Mice; Motor Activity; Neurons; Nucleus Accumbens; Piperidines; Pyridines; Receptors, Dopamine D2; Receptors, Dopamine D3 | 2019 |
Newly Developed Dopamine D
Topics: Animals; Blood Pressure; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Heart Rate; Indoles; Male; Nitriles; Oxycodone; Piperazines; Piperidines; Rats; Rats, Long-Evans; Receptors, Dopamine D3; Tetrahydroisoquinolines | 2019 |
Pharmacological targeting of striatal indirect pathway neurons improves subthalamic nucleus dysfunction and reduces repetitive behaviors in C58 mice.
Topics: Adenosine; Animals; Autism Spectrum Disorder; Basal Ganglia; Behavior, Animal; Benzamides; Compulsive Behavior; Corpus Striatum; Disease Models, Animal; Indoles; Male; Mice; Mice, Inbred Strains; Neural Pathways; Neurons; Phenethylamines; Piperidines; Pyrazoles; Stereotyped Behavior; Subthalamic Nucleus | 2020 |