Page last updated: 2024-09-04

l 741626 and piperidines

l 741626 has been researched along with piperidines in 47 studies

Compound Research Comparison

Studies
(l 741626)
Trials
(l 741626)
Recent Studies (post-2010)
(l 741626)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
7603340,2355,22114,545

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (4.26)18.2507
2000's24 (51.06)29.6817
2010's20 (42.55)24.3611
2020's1 (2.13)2.80

Authors

AuthorsStudies
Bowery, BJ; Bristow, L; Emms, F; Freedman, S; Kulagowski, J; Patel, S; Razzaque, Z; Seabrook, GR1
Brown, NA; McAllister, G; Milligan, G; Pillai, G; Seabrook, GR1
Dekeyne, A; Girardon, S; Millan, MJ; Monneyron, S1
Audinot, V; Cussac, D; Dubuffet, T; Gobert, A; Lavielle, G; Lejeune, F; Millan, MJ; Newman-Tancredi, A; Rivet, JM1
Brocco, M; Dekeyne, A; Dubuffet, T; Lavielle, G; Millan, MJ; Rivet, JM1
Fushiki, T; Imaizumi, M; Takeda, M1
Henry, BL; LaHoste, GJ; Marshall, JF1
Canales, JJ; Iversen, SD1
Bergeron, J; Courtney, C; McConkey, M; Melch, M; Shrikhande, A; Smith, D; Wong, SK1
Chapman, KL; Hutson, PH; Marston, D; Patel, S; Ragan, CI1
Chaperon, F; Neijt, HC; Tricklebank, MD; Unger, L1
Doleviczényi, Z; Halmos, G; Kittel, A; Lendvai, B; Répássy, G; Vizi, ES; Zelles, T1
Hattori, K; Isosaka, T; Iyo, M; Kohsaka, S; Maekawa, M; Sato, T; Uchino, S; Yagi, T; Yuasa, S1
Brotchie, JM; Millan, MJ; Visanji, NP1
Brotchie, JM; Crossman, AR; Hill, MP; McGuire, SG; Millan, MJ; Ravenscroft, P; Rochat, C1
Grundt, P; Husband, SL; Luedtke, RR; Newman, AH; Taylor, M1
Calinski, DM; Collins, GT; Grundt, P; Newman, AH; Woods, JH1
Bugert, P; Klüter, H; Schedel, A; Schloss, P1
Abe, M; Egashira, N; Fujiwara, M; Iwasaki, K; Matsushita, M; Mishima, K; Nishimura, R; Oishi, R; Okuno, R1
Loiseau, F; Millan, MJ1
Breier, M; Chang, WL; Ko, D; Swerdlow, NR; Weber, M1
Han, P; Whelan, PJ1
Chang, WL; Durbin, JP; Luedtke, RR; Mach, RH; Park, PE; Swerdlow, NR; Weber, M1
Arnt, J; Bétry, C; Etievant, A; Haddjeri, N1
Gross, G; Jongen-Rêlo, AL; Schoemaker, H; Unger, L; van Gaalen, MM1
Georgiou, J; Lee, FJ; Liu, F; Mansuy, IM; Michalon, A; Nath, A; Roder, JC; Saab, BJ; Wang, M1
Fan, X; Hess, EJ; Xu, M1
Achat-Mendes, C; Cao, J; Grundt, P; Newman, AH; Platt, DM; Spealman, RD1
Arai, Y; Kikuchi, T; Mitazaki, S; Nakagawasai, O; Nakaya, K; Niijima, F; Onogi, H; Sato, A; Tadano, T; Tan-No, K1
Breier, MR; Chang, WL; Swerdlow, NR; Yang, A1
Fone, KC; Ingallinesi, M; Loiseau, F; Marsden, CA; Millan, MJ; Watson, DJ1
Bernedo, VE; Chen, R; Kilb, W; Kolbaev, SN; Luhmann, HJ; Moser, J; Sharopov, S; Werhahn, KJ1
Ansah, OB; Pertovaara, A; Viisanen, H1
Dankoski, EC; Fish, EW; Han, JE; Hodge, CW; Krouse, MC; Malanga, CJ; Philpot, BD; Riday, TT; Walsh, PL; Wightman, RM1
Baladi, MG; France, CP; Newman, AH1
Bentley, TA; France, CP; Grenier, AE; Serafine, KM1
Davoodi, N; Langlois, X; te Riele, P1
Di Ciano, P; Diaz, J; Khaled, MA; Le Foll, B; Pushparaj, A1
Bentley, TA; France, CP; Kilborn, DJ; Koek, W; Serafine, KM1
Dulawa, SC; Ho, EV; Klenotich, SJ; McMurray, MS; Server, CH1
Newton, CL; Strange, PG; Wood, MD1
Jones, SR; McGinnis, MM; Siciliano, CA1
Cho, J; Kim, G; Kim, M; Lee, S; Won, C1
Barrett, AC; Butler, P; Caine, SB; Negus, SS; Thomsen, M1
Branco, RC; Foster, SL; Manvich, DF; Miller, GW; Newman, AH; Paladini, CA; Petko, AK; Porter-Stransky, KA; Stout, KA; Weinshenker, D1
Baumann, MH; Humburg, BA; Jordan, CJ; Newman, AH; Schindler, CW; Shaik, AB; Thorndike, EB; Xi, ZX1
King, MA; Lewis, MH; Maletz, S; Muehlmann, AM1

Other Studies

47 other study(ies) available for l 741626 and piperidines

ArticleYear
Antagonism of the effects of (+)-PD 128907 on midbrain dopamine neurones in rat brain slices by a selective D2 receptor antagonist L-741,626.
    British journal of pharmacology, 1996, Volume: 119, Issue:7

    Topics: Animals; Benzopyrans; Cloning, Molecular; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Electrophysiology; Indoles; Male; Mesencephalon; Neurons; Oxazines; Patch-Clamp Techniques; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Spiperone

1996
Human D2 and D4 dopamine receptors couple through betagamma G-protein subunits to inwardly rectifying K+ channels (GIRK1) in a Xenopus oocyte expression system: selective antagonism by L-741,626 and L-745,870 respectively.
    Neuropharmacology, 1998, Volume: 37, Issue:8

    Topics: Dopamine Antagonists; Dopamine D2 Receptor Antagonists; GTP-Binding Proteins; Humans; Indoles; Ion Channel Gating; Membrane Potentials; Oocytes; Patch-Clamp Techniques; Piperidines; Potassium Channel Blockers; Pyridines; Pyrroles; Receptors, Dopamine D4

1998
Discriminative stimulus properties of the dopamine D3 receptor agonists, PD128,907 and 7-OH-DPAT: a comparative characterization with novel ligands at D3 versus D2 receptors.
    Neuropharmacology, 2000, Feb-14, Volume: 39, Issue:4

    Topics: 2-Naphthylamine; Animals; Benzopyrans; Dioxins; Discrimination Learning; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Furans; Generalization, Psychological; Humans; Indoles; Ligands; Male; Oxazines; Piperazines; Piperidines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Stereoisomerism; Tetrahydronaphthalenes

2000
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: I. Receptorial, electrophysiological and neurochemical profile compared with GR218,231 and L741,626.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: Animals; Benzopyrans; Brain; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Activation; Guanosine 5'-O-(3-Thiotriphosphate); Indoles; Male; Mitogen-Activated Protein Kinases; Norepinephrine; Oxazines; Piperidines; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Serotonin; Sulfones; Tetrahydronaphthalenes

2000
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: II. Functional and behavioral profile compared with GR218,231 and L741,626.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: Animals; Behavior, Animal; Benzopyrans; Body Temperature; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Indoles; Male; Mice; Motor Activity; Oxazines; Piperidines; Psychotropic Drugs; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D3; Sulfones; Tetrahydronaphthalenes

2000
Effects of oil intake in the conditioned place preference test in mice.
    Brain research, 2000, Jul-07, Volume: 870, Issue:1-2

    Topics: Animals; Behavior, Animal; Benzazepines; Brain Chemistry; Conditioning, Psychological; Corn Oil; Dopamine Antagonists; Eating; Haloperidol; Indoles; Male; Mice; Piperidines; Receptors, Dopamine D1; Reward; Space Perception; Sulpiride

2000
Dopamine D1 receptors synergize with D2, but not D3 or D4, receptors in the striatum without the involvement of action potentials.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Sep-01, Volume: 20, Issue:17

    Topics: Action Potentials; Amphetamine; Animals; Corpus Striatum; Dopamine Antagonists; Genes, fos; Indans; Indoles; Male; Piperidines; Proto-Oncogene Proteins c-fos; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor Cross-Talk; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4; Tetrodotoxin

2000
Psychomotor-activating effects mediated by dopamine D(2) and D(3) receptors in the nucleus accumbens.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 67, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Benzopyrans; Bromocriptine; Grooming; Indoles; Motor Activity; Naphthalenes; Nucleus Accumbens; Oxazines; Piperidines; Pyrrolidines; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3

2000
Fully automated radioligand binding filtration assay for membrane-bound receptors.
    BioTechniques, 2002, Volume: 33, Issue:4

    Topics: Animals; Automation; Binding, Competitive; CHO Cells; Cricetinae; Filtration; Haloperidol; Indoles; Piperidines; Radioligand Assay; Receptors, Dopamine; Reproducibility of Results; Time Factors

2002
Pharmacological and functional characterisation of dopamine D4 receptors in the rat retina.
    Neuropharmacology, 2003, Volume: 44, Issue:8

    Topics: Animals; Binding Sites; Cyclic AMP; Darkness; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Indoles; Male; Piperidines; Pyridines; Pyrroles; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Retina; Spiperone

2003
Evidence for regulation of body temperature in rats by dopamine D2 receptor and possible influence of D1 but not D3 and D4 receptors.
    Neuropharmacology, 2003, Volume: 44, Issue:8

    Topics: Animals; Aporphines; Benzazepines; Benzopyrans; Body Temperature Regulation; Dopamine Agonists; Dopamine Antagonists; Hypothermia; Indoles; Oxazines; Piperazines; Piperidines; Pyridines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4

2003
D2 autoreceptor inhibition reveals oxygen-glucose deprivation-induced release of dopamine in guinea-pig cochlea.
    Neuroscience, 2005, Volume: 132, Issue:3

    Topics: Animals; Cochlea; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Drug Interactions; Electric Stimulation; Glucose; Guinea Pigs; Hypoxia; In Vitro Techniques; Indoles; Male; Neurons; Nomifensine; Piperidines; Receptors, Dopamine D2; Sulpiride; Tetrodotoxin; Time Factors; Tritium

2005
Fyn is required for haloperidol-induced catalepsy in mice.
    The Journal of biological chemistry, 2006, Mar-17, Volume: 281, Issue:11

    Topics: Animals; Anti-Dyskinesia Agents; Antipsychotic Agents; Blotting, Western; Calcium; Catalepsy; Cells, Cultured; Dopamine; Genotype; Haloperidol; Immunoblotting; Immunohistochemistry; Immunoprecipitation; In Situ Hybridization; Indoles; Mice; Neurons; Phosphorylation; Piperidines; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-fyn; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Time Factors; Tyrosine

2006
Actions at sites other than D(3) receptors mediate the effects of BP897 on l-DOPA-induced hyperactivity in monoamine-depleted rats.
    Experimental neurology, 2006, Volume: 202, Issue:1

    Topics: Adrenergic Uptake Inhibitors; Animals; Behavior, Animal; Biogenic Monoamines; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Hyperkinesis; Indoles; Levodopa; Male; Motor Activity; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Reserpine; Time Factors

2006
Antiparkinsonian effects of the novel D3/D2 dopamine receptor agonist, S32504, in MPTP-lesioned marmosets: Mediation by D2, not D3, dopamine receptors.
    Movement disorders : official journal of the Movement Disorder Society, 2006, Volume: 21, Issue:12

    Topics: Analysis of Variance; Animals; Antiparkinson Agents; Behavior, Animal; Callithrix; Disease Models, Animal; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Indoles; Levodopa; Motor Activity; MPTP Poisoning; Oxazines; Piperidines; Receptors, Dopamine D2; Receptors, Dopamine D3; Time Factors

2006
Analogues of the dopamine D2 receptor antagonist L741,626: Binding, function, and SAR.
    Bioorganic & medicinal chemistry letters, 2007, Feb-01, Volume: 17, Issue:3

    Topics: Cell Line; Dopamine Antagonists; Humans; Indoles; Ligands; Piperidines; Protein Binding; Receptors, Dopamine D2; Structure-Activity Relationship; Transfection

2007
Food restriction alters N'-propyl-4,5,6,7-tetrahydrobenzothiazole-2,6-diamine dihydrochloride (pramipexole)-induced yawning, hypothermia, and locomotor activity in rats: evidence for sensitization of dopamine D2 receptor-mediated effects.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 325, Issue:2

    Topics: Animals; Benzamides; Benzothiazoles; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Food; Hypothermia; Indoles; Male; Motor Activity; Penile Erection; Physostigmine; Piperazines; Piperidines; Pramipexole; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Yawning

2008
The dopamine agonism on ADP-stimulated platelets is mediated through D2-like but not D1-like dopamine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 378, Issue:4

    Topics: Adenosine Diphosphate; Antigens, CD; Benzazepines; Clozapine; Collagen Type IV; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Epinephrine; Flow Cytometry; Humans; Indoles; Methylphenidate; P-Selectin; Piperidines; Platelet Activation; Platelet Adhesiveness; Platelet Aggregation; Platelet Membrane Glycoproteins; Platelet-Rich Plasma; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Tetraspanin 30

2008
Aripiprazole inhibits marble-burying behavior via 5-hydroxytryptamine (5-HT)1A receptor-independent mechanisms.
    European journal of pharmacology, 2008, Sep-11, Volume: 592, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Anxiety; Aripiprazole; Behavior, Animal; Benzodiazepines; Catalepsy; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Ketanserin; Male; Mice; Mice, Inbred ICR; Olanzapine; Piperazines; Piperidines; Postural Balance; Psychomotor Performance; Pyridines; Quinolones; Quinpirole; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Blockade of dopamine D(3) receptors in frontal cortex, but not in sub-cortical structures, enhances social recognition in rats: similar actions of D(1) receptor agonists, but not of D(2) antagonists.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2009, Volume: 19, Issue:1

    Topics: Animals; Benzazepines; Benzopyrans; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indoles; Male; Microinjections; Nitriles; Piperidines; Prefrontal Cortex; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D3; Recognition, Psychology; Social Behavior; Tetrahydroisoquinolines

2009
Heritable strain differences in sensitivity to the startle gating-disruptive effects of D2 but not D3 receptor stimulation.
    Behavioural pharmacology, 2008, Volume: 19, Issue:8

    Topics: Acoustic Stimulation; Analysis of Variance; Animals; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gait Disorders, Neurologic; Indoles; Male; Neural Inhibition; Nucleus Accumbens; Piperidines; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sensory Gating

2008
Modulation of AMPA currents by D(1)-like but not D(2)-like receptors in spinal motoneurons.
    Neuroscience, 2009, Feb-18, Volume: 158, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Newborn; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Excitatory Amino Acid Agonists; In Vitro Techniques; Indoles; Ion Channel Gating; Membrane Potentials; Mice; Motor Neurons; Patch-Clamp Techniques; Piperidines; Receptors, Dopamine D1; Receptors, Dopamine D2; Spinal Cord

2009
Using prepulse inhibition to detect functional D3 receptor antagonism: effects of WC10 and WC44.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 93, Issue:2

    Topics: Animals; Antipsychotic Agents; Apomorphine; Benzothiazoles; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Piperazines; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Startle

2009
Bifeprunox and aripiprazole suppress in vivo VTA dopaminergic neuronal activity via D2 and not D3 dopamine autoreceptor activation.
    Neuroscience letters, 2009, Aug-21, Volume: 460, Issue:1

    Topics: Action Potentials; Analysis of Variance; Animals; Antipsychotic Agents; Aripiprazole; Benzoxazoles; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Drug Interactions; Indoles; Male; Neurons; Piperazines; Piperidines; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Sulfones; Tetrahydronaphthalenes; Ventral Tegmental Area

2009
Amphetamine decreases behavioral inhibition by stimulation of dopamine D2, but not D3, receptors.
    Behavioural pharmacology, 2009, Volume: 20, Issue:5-6

    Topics: Amphetamine; Animals; Cell Line, Transformed; Central Nervous System Stimulants; Choice Behavior; Conditioning, Operant; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Humans; Indoles; Inhibition, Psychological; Male; Nitriles; Piperidines; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydroisoquinolines

2009
NCS-1 in the dentate gyrus promotes exploration, synaptic plasticity, and rapid acquisition of spatial memory.
    Neuron, 2009, Sep-10, Volume: 63, Issue:5

    Topics: Animals; Cell Membrane; Dentate Gyrus; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Exploratory Behavior; In Vitro Techniques; Indoles; Learning; Long-Term Potentiation; Maze Learning; Memory; Mice; Mice, Transgenic; Models, Neurological; Motor Activity; Neuronal Calcium-Sensor Proteins; Neuropeptides; Neuropsychological Tests; Piperidines; Rats; Receptors, Dopamine D2; Recognition, Psychology; Space Perception; Time Factors

2009
D2 dopamine receptor subtype-mediated hyperactivity and amphetamine responses in a model of ADHD.
    Neurobiology of disease, 2010, Volume: 37, Issue:1

    Topics: Amphetamine; Animals; Attention Deficit Disorder with Hyperactivity; Benzopyrans; Corpus Striatum; Dihydroxyphenylalanine; Disease Models, Animal; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Extracellular Space; Indoles; Locomotion; Mice; Mice, Knockout; Mice, Mutant Strains; Piperidines; Pyridines; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4

2010
Dopamine D3 and D2 receptor mechanisms in the abuse-related behavioral effects of cocaine: studies with preferential antagonists in squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 334, Issue:2

    Topics: Animals; Behavior, Animal; Benzamides; Benzimidazoles; Benzopyrans; Cocaine-Related Disorders; Discrimination Learning; Dopamine D2 Receptor Antagonists; Indoles; Oxazines; Piperidines; Pyridines; Receptors, Dopamine D2; Receptors, Dopamine D3; Saimiri

2010
p-Hydroxyamphetamine causes prepulse inhibition disruptions in mice: contribution of dopamine neurotransmission.
    Behavioural brain research, 2010, Dec-25, Volume: 214, Issue:2

    Topics: Animals; Benzazepines; Clozapine; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Indoles; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Oxidopamine; p-Hydroxyamphetamine; Piperazines; Piperidines; Pyridines; Pyrroles; Reflex, Startle; Salicylamides; Sensory Gating; Sympathomimetics; Synaptic Transmission

2010
Disparate effects of pramipexole on locomotor activity and sensorimotor gating in Sprague-Dawley rats.
    Pharmacology, biochemistry, and behavior, 2011, Volume: 99, Issue:4

    Topics: Animals; Benzothiazoles; Data Interpretation, Statistical; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Motor Activity; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Reflex, Startle; Sensory Gating

2011
Selective blockade of dopamine D3 receptors enhances while D2 receptor antagonism impairs social novelty discrimination and novel object recognition in rats: a key role for the prefrontal cortex.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2012, Volume: 37, Issue:3

    Topics: Animals; Benzopyrans; Discrimination, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Mice; Mice, Knockout; Microinjections; Piperidines; Prefrontal Cortex; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Recognition, Psychology

2012
Dopaminergic modulation of low-Mg²⁺-induced epileptiform activity in the intact hippocampus of the newborn mouse in vitro.
    Journal of neuroscience research, 2012, Volume: 90, Issue:10

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Benzazepines; Data Interpretation, Statistical; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Epilepsy; Hippocampus; Indoles; Magnesium Deficiency; Mice; Mice, Inbred C57BL; Nitriles; Piperidines; Quinpirole; Receptors, Dopamine D2; Synapses; Tetrahydroisoquinolines

2012
The role of the dopamine D2 receptor in descending control of pain induced by motor cortex stimulation in the neuropathic rat.
    Brain research bulletin, 2012, Nov-01, Volume: 89, Issue:3-4

    Topics: Analysis of Variance; Animals; Deep Brain Stimulation; Disease Models, Animal; Dopamine Antagonists; Functional Laterality; Hot Temperature; Indoles; Male; Motor Cortex; Motor Neurons; Nociceptors; Pain; Pain Measurement; Peripheral Nervous System Diseases; Piperidines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Reflex; Spinal Cord

2012
Pathway-specific dopaminergic deficits in a mouse model of Angelman syndrome.
    The Journal of clinical investigation, 2012, Volume: 122, Issue:12

    Topics: Angelman Syndrome; Animals; Benzazepines; Cocaine; Disease Models, Animal; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dopaminergic Neurons; Electric Stimulation; Female; Indoles; Male; Mice; Mice, Inbred C57BL; Motor Activity; Piperidines; Raclopride; Receptors, Dopamine D1; Reward; Self Stimulation; Substantia Nigra; Synaptic Transmission; Ubiquitin-Protein Ligases; Ventral Tegmental Area

2012
Feeding condition and the relative contribution of different dopamine receptor subtypes to the discriminative stimulus effects of cocaine in rats.
    Psychopharmacology, 2014, Volume: 231, Issue:3

    Topics: Animals; Apomorphine; Benzamides; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Electroshock; Food Deprivation; Indoles; Lisuride; Male; Piperidines; Pyridines; Quinpirole; Raclopride; Rats, Sprague-Dawley; Reinforcement, Psychology

2014
Eating high fat chow and the behavioral effects of direct-acting and indirect-acting dopamine receptor agonists in female rats.
    Behavioural pharmacology, 2014, Volume: 25, Issue:4

    Topics: Aging; Animals; Body Temperature; Body Weight; Cocaine; Diet, High-Fat; Dietary Fats; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Eating; Female; Hypothermia; Indoles; Insulin Resistance; Motor Activity; Piperidines; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2; Yawning

2014
Examining dopamine D3 receptor occupancy by antipsychotic drugs via [3H]7-OH-DPAT ex vivo autoradiography and its cross-validation via c-fos immunohistochemistry in the rat brain.
    European journal of pharmacology, 2014, Oct-05, Volume: 740

    Topics: Animals; Antipsychotic Agents; Autoradiography; Benzodiazepines; Clozapine; Dopamine Antagonists; Haloperidol; Indoles; Islands of Calleja; Male; Nitriles; Olanzapine; Piperidines; Proto-Oncogene Proteins c-fos; Radiography; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydroisoquinolines; Tetrahydronaphthalenes

2014
Dopamine D3 receptors in the basolateral amygdala and the lateral habenula modulate cue-induced reinstatement of nicotine seeking.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:13

    Topics: Animals; Autoradiography; Basolateral Nuclear Complex; Conditioning, Operant; Cues; Dopamine Antagonists; Drug-Seeking Behavior; Extinction, Psychological; Habenula; Indoles; Iodine Isotopes; Male; Nicotine; Nicotinic Agonists; Nitriles; Piperidines; Rats; Rats, Long-Evans; Receptors, Dopamine D3; Reinforcement, Psychology; Self Administration; Tetrahydroisoquinolines; Tetrahydronaphthalenes

2014
Drinking sucrose or saccharin enhances sensitivity of rats to quinpirole-induced yawning.
    European journal of pharmacology, 2015, Oct-05, Volume: 764

    Topics: Administration, Oral; Animals; Behavior, Animal; Benzamides; Dietary Sucrose; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drinking; Drug Administration Schedule; Drug Interactions; Indoles; Male; Non-Nutritive Sweeteners; Piperidines; Pyridines; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D3; Saccharin; Yawning

2015
Dopamine D2/3 receptor antagonism reduces activity-based anorexia.
    Translational psychiatry, 2015, Aug-04, Volume: 5

    Topics: Amisulpride; Animals; Anorexia Nervosa; Benzodiazepines; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Eating; Female; Indoles; Mice; Mice, Inbred BALB C; Motor Activity; Nitriles; Olanzapine; Piperidines; Receptors, Dopamine D3; Salicylamides; Sulpiride; Tetrahydroisoquinolines; Weight Loss

2015
Examining the Effects of Sodium Ions on the Binding of Antagonists to Dopamine D2 and D3 Receptors.
    PloS one, 2016, Volume: 11, Issue:7

    Topics: Animals; Binding, Competitive; Biphenyl Compounds; Cell Line, Tumor; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Indans; Indoles; Ions; Ligands; Molecular Structure; Mutation; Nitriles; Piperazines; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Sf9 Cells; Sodium; Spodoptera; Tetrahydroisoquinolines

2016
Dopamine D3 autoreceptor inhibition enhances cocaine potency at the dopamine transporter.
    Journal of neurochemistry, 2016, Volume: 138, Issue:6

    Topics: Animals; Autoreceptors; Cocaine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Synergism; Female; Indoles; Male; Mice; Mice, Inbred C57BL; Nitriles; Piperidines; Raclopride; Receptors, Dopamine D2; Receptors, Tumor Necrosis Factor, Member 25; Sex Characteristics; Tetrahydroisoquinolines

2016
Dopamine D3 receptor-modulated neuroprotective effects of lisuride.
    Neuropharmacology, 2017, 05-01, Volume: 117

    Topics: Animals; ATPases Associated with Diverse Cellular Activities; Biphenyl Compounds; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Indoles; Lisuride; Male; Metalloendopeptidases; Mice; Mitochondria; Neuroprotective Agents; Oxidopamine; Piperazines; Piperidines; Primary Cell Culture; Receptors, Dopamine D3; Tyrosine 3-Monooxygenase

2017
Effects of Acute and Chronic Treatments with Dopamine D
    The Journal of pharmacology and experimental therapeutics, 2017, Volume: 362, Issue:1

    Topics: Aminopyridines; Animals; Benzamides; Choice Behavior; Cocaine; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Tolerance; Food; Indoles; Ligands; Male; Morpholines; Piperidines; Pyridines; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology

2017
Selective D
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:8

    Topics: Action Potentials; Animals; Benzamides; Central Nervous System Sensitization; Cocaine; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Mice; Motor Activity; Neurons; Nucleus Accumbens; Piperidines; Pyridines; Receptors, Dopamine D2; Receptors, Dopamine D3

2019
Newly Developed Dopamine D
    The Journal of pharmacology and experimental therapeutics, 2019, Volume: 371, Issue:3

    Topics: Animals; Blood Pressure; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Heart Rate; Indoles; Male; Nitriles; Oxycodone; Piperazines; Piperidines; Rats; Rats, Long-Evans; Receptors, Dopamine D3; Tetrahydroisoquinolines

2019
Pharmacological targeting of striatal indirect pathway neurons improves subthalamic nucleus dysfunction and reduces repetitive behaviors in C58 mice.
    Behavioural brain research, 2020, 08-05, Volume: 391

    Topics: Adenosine; Animals; Autism Spectrum Disorder; Basal Ganglia; Behavior, Animal; Benzamides; Compulsive Behavior; Corpus Striatum; Disease Models, Animal; Indoles; Male; Mice; Mice, Inbred Strains; Neural Pathways; Neurons; Phenethylamines; Piperidines; Pyrazoles; Stereotyped Behavior; Subthalamic Nucleus

2020