Page last updated: 2024-09-04

l 741626 and cocaine

l 741626 has been researched along with cocaine in 7 studies

Compound Research Comparison

Studies
(l 741626)
Trials
(l 741626)
Recent Studies (post-2010)
(l 741626)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
7603332,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomyl 741626 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's7 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dankoski, EC; Fish, EW; Han, JE; Hodge, CW; Krouse, MC; Malanga, CJ; Philpot, BD; Riday, TT; Walsh, PL; Wightman, RM1
Baladi, MG; France, CP; Newman, AH1
Bentley, TA; France, CP; Grenier, AE; Serafine, KM1
Jones, SR; McGinnis, MM; Siciliano, CA1
Barrett, AC; Butler, P; Caine, SB; Negus, SS; Thomsen, M1
Branco, RC; Foster, SL; Manvich, DF; Miller, GW; Newman, AH; Paladini, CA; Petko, AK; Porter-Stransky, KA; Stout, KA; Weinshenker, D1
Baumann, MH; Humburg, BA; Jordan, CJ; Newman, AH; Schindler, CW; Shaik, AB; Thorndike, EB; Xi, ZX1

Other Studies

7 other study(ies) available for l 741626 and cocaine

ArticleYear
Pathway-specific dopaminergic deficits in a mouse model of Angelman syndrome.
    The Journal of clinical investigation, 2012, Volume: 122, Issue:12

    Topics: Angelman Syndrome; Animals; Benzazepines; Cocaine; Disease Models, Animal; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dopaminergic Neurons; Electric Stimulation; Female; Indoles; Male; Mice; Mice, Inbred C57BL; Motor Activity; Piperidines; Raclopride; Receptors, Dopamine D1; Reward; Self Stimulation; Substantia Nigra; Synaptic Transmission; Ubiquitin-Protein Ligases; Ventral Tegmental Area

2012
Feeding condition and the relative contribution of different dopamine receptor subtypes to the discriminative stimulus effects of cocaine in rats.
    Psychopharmacology, 2014, Volume: 231, Issue:3

    Topics: Animals; Apomorphine; Benzamides; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Electroshock; Food Deprivation; Indoles; Lisuride; Male; Piperidines; Pyridines; Quinpirole; Raclopride; Rats, Sprague-Dawley; Reinforcement, Psychology

2014
Eating high fat chow and the behavioral effects of direct-acting and indirect-acting dopamine receptor agonists in female rats.
    Behavioural pharmacology, 2014, Volume: 25, Issue:4

    Topics: Aging; Animals; Body Temperature; Body Weight; Cocaine; Diet, High-Fat; Dietary Fats; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Eating; Female; Hypothermia; Indoles; Insulin Resistance; Motor Activity; Piperidines; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2; Yawning

2014
Dopamine D3 autoreceptor inhibition enhances cocaine potency at the dopamine transporter.
    Journal of neurochemistry, 2016, Volume: 138, Issue:6

    Topics: Animals; Autoreceptors; Cocaine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Synergism; Female; Indoles; Male; Mice; Mice, Inbred C57BL; Nitriles; Piperidines; Raclopride; Receptors, Dopamine D2; Receptors, Tumor Necrosis Factor, Member 25; Sex Characteristics; Tetrahydroisoquinolines

2016
Effects of Acute and Chronic Treatments with Dopamine D
    The Journal of pharmacology and experimental therapeutics, 2017, Volume: 362, Issue:1

    Topics: Aminopyridines; Animals; Benzamides; Choice Behavior; Cocaine; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Tolerance; Food; Indoles; Ligands; Male; Morpholines; Piperidines; Pyridines; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology

2017
Selective D
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2019, Volume: 44, Issue:8

    Topics: Action Potentials; Animals; Benzamides; Central Nervous System Sensitization; Cocaine; Dopamine; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Mice; Motor Activity; Neurons; Nucleus Accumbens; Piperidines; Pyridines; Receptors, Dopamine D2; Receptors, Dopamine D3

2019
Newly Developed Dopamine D
    The Journal of pharmacology and experimental therapeutics, 2019, Volume: 371, Issue:3

    Topics: Animals; Blood Pressure; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Heart Rate; Indoles; Male; Nitriles; Oxycodone; Piperazines; Piperidines; Rats; Rats, Long-Evans; Receptors, Dopamine D3; Tetrahydroisoquinolines

2019