Page last updated: 2024-09-03

l 703606 and capsazepine

l 703606 has been researched along with capsazepine in 4 studies

Compound Research Comparison

Studies
(l 703606)
Trials
(l 703606)
Recent Studies (post-2010)
(l 703606)
Studies
(capsazepine)
Trials
(capsazepine)
Recent Studies (post-2010) (capsazepine)
740127813273

Protein Interaction Comparison

ProteinTaxonomyl 703606 (IC50)capsazepine (IC50)
Transient receptor potential cation channel subfamily V member 1Rattus norvegicus (Norway rat)0.4293
Transient receptor potential cation channel subfamily V member 1Homo sapiens (human)0.2587
Transient receptor potential cation channel subfamily V member 4Rattus norvegicus (Norway rat)0.6333
Transient receptor potential cation channel subfamily V member 2Rattus norvegicus (Norway rat)0.6333

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Mustafa, S; Oriowo, MA1
Feng, NH; Lee, HH; Ma, MC; Shiang, JC1
Sachs, JR; Wang, DH; Xie, C1
Chen, PX; Guo, HM; Huang, JH; Luo, YL; Zhang, YL; Zhou, WL; Zhu, YX1

Other Studies

4 other study(ies) available for l 703606 and capsazepine

ArticleYear
Inhibitory effect of capsaicin on cholinergic transmission in ovine airways: evidence for non-cholinergic contractions.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Acetylcholine; Animals; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptides, Cyclic; Quinuclidines; Receptors, Drug; Receptors, Neurokinin-2; Serotonin; Sheep; Substance P; Synaptic Transmission; Trachea

1999
Transient receptor potential vanilloid type 1 channels act as mechanoreceptors and cause substance P release and sensory activation in rat kidneys.
    American journal of physiology. Renal physiology, 2008, Volume: 294, Issue:2

    Topics: Action Potentials; Animals; Blood Pressure; Capsaicin; Cell Membrane; Cytosol; Diterpenes; Electrophysiology; Female; Kidney; Kidney Pelvis; Mechanoreceptors; Models, Biological; Neurokinin-1 Receptor Antagonists; Perfusion; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Sensory System Agents; Substance P; TRPV Cation Channels; Ubiquitin Thiolesterase

2008
Interdependent regulation of afferent renal nerve activity and renal function: role of transient receptor potential vanilloid type 1, neurokinin 1, and calcitonin gene-related peptide receptors.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 325, Issue:3

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Ganglia, Spinal; Isoindoles; Kidney Pelvis; Male; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Peptide Fragments; Quinuclidines; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Substance P; TRPV Cation Channels

2008
Cellular mechanism underlying formaldehyde-stimulated Cl- secretion in rat airway epithelium.
    PloS one, 2013, Volume: 8, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anions; Biological Transport; Capsaicin; Cells, Cultured; Chlorides; Colforsin; Epinephrine; Epithelial Cells; Formaldehyde; Imines; Male; Nerve Endings; ortho-Aminobenzoates; Quinuclidines; Rats; Respiratory Mucosa; Substance P; Trachea; TRPV Cation Channels

2013