l 703606 has been researched along with capsaicin in 12 studies
Studies (l 703606) | Trials (l 703606) | Recent Studies (post-2010) (l 703606) | Studies (capsaicin) | Trials (capsaicin) | Recent Studies (post-2010) (capsaicin) |
---|---|---|---|---|---|
74 | 0 | 12 | 11,238 | 661 | 3,410 |
Protein | Taxonomy | l 703606 (IC50) | capsaicin (IC50) |
---|---|---|---|
Transient receptor potential cation channel subfamily V member 1 | Rattus norvegicus (Norway rat) | 0.019 | |
Lysine-specific histone demethylase 1A | Homo sapiens (human) | 0.6 | |
Bile salt export pump | Homo sapiens (human) | 10 | |
Cytochrome P450 1A2 | Homo sapiens (human) | 3 | |
Prostaglandin G/H synthase 1 | Homo sapiens (human) | 2.6755 | |
Transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | 0.008 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (16.67) | 18.2507 |
2000's | 8 (66.67) | 29.6817 |
2010's | 2 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bunnett, NW; Grady, EF; Martínez, V; Marvizón, JC; Mayer, EA | 1 |
Mustafa, S; Oriowo, MA | 1 |
Gear, RW; Levine, JD; Tambeli, CH; Young, A | 1 |
Horie, S; Minowa, S; Murayama, T; Someya, A; Tsuchiya, S | 1 |
Nies, M; Ro, JY; Zhang, Y | 1 |
Bell, EB; Beresford, LJ; Miyan, JA; Shepherd, AJ | 1 |
Fujiwara, N; Maeda, T; Seo, K; Someya, G; Takeuchi, K | 1 |
Kawana, S; Yamaoka, J | 1 |
Feng, NH; Lee, HH; Ma, MC; Shiang, JC | 1 |
Sachs, JR; Wang, DH; Xie, C | 1 |
Hamity, MV; Hammond, DL; White, SR | 1 |
Chen, PX; Guo, HM; Huang, JH; Luo, YL; Zhang, YL; Zhou, WL; Zhu, YX | 1 |
12 other study(ies) available for l 703606 and capsaicin
Article | Year |
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Neurokinin 1 receptor internalization in spinal cord slices induced by dorsal root stimulation is mediated by NMDA receptors.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Capsaicin; Electric Stimulation; Endocytosis; Evoked Potentials; Ganglia, Spinal; Hyperalgesia; Long-Term Potentiation; Male; Microscopy, Confocal; Microscopy, Fluorescence; Models, Neurological; N-Methylaspartate; Neurokinin-1 Receptor Antagonists; Quinuclidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Substance P | 1997 |
Inhibitory effect of capsaicin on cholinergic transmission in ovine airways: evidence for non-cholinergic contractions.
Topics: Acetylcholine; Animals; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptides, Cyclic; Quinuclidines; Receptors, Drug; Receptors, Neurokinin-2; Serotonin; Sheep; Substance P; Synaptic Transmission; Trachea | 1999 |
Contribution of spinal glutamatergic mechanisms in heterosegmental antinociception induced by noxious stimulation.
Topics: Animals; Benzoates; Capsaicin; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Isoquinolines; Male; Nociceptors; Pyridines; Quinoxalines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Stimulation, Chemical; Substance P | 2003 |
Role of neuropeptide receptor systems in vanilloid VR1 receptor-mediated gastric acid secretion in rat brain.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Excitatory Amino Acid Antagonists; Gastric Acid; Hypothalamus; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Quinuclidines; Rats; Rats, Wistar; Receptor Cross-Talk; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Glutamate; Receptors, Neurokinin-2; Time Factors; TRPV Cation Channels | 2004 |
Substance P does not play a critical role in neurogenic inflammation in the rat masseter muscle.
Topics: Analgesics; Animals; Capsaicin; Disease Models, Animal; Edema; Inflammation Mediators; Male; Masseter Muscle; Mustard Plant; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Plant Extracts; Plant Oils; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P | 2005 |
Mobilisation of specific T cells from lymph nodes in contact sensitivity requires substance P.
Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cell Movement; Dermatitis, Contact; Dinitrochlorobenzene; Dose-Response Relationship, Drug; Drug Interactions; Immunohistochemistry; Lymph Nodes; Mice; Nerve Fibers; Quinuclidines; Skin; Substance P; Sympathectomy, Chemical; T-Lymphocytes | 2005 |
Postnatal development of excitation propagation in the trigeminal subnucleus caudalis evoked by afferent stimulation in mice.
Topics: Afferent Pathways; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Capsaicin; Diagnostic Imaging; Dizocilpine Maleate; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neurokinin-1 Receptor Antagonists; Quinuclidines; Silver Staining; Time Factors; Trigeminal Caudal Nucleus | 2005 |
A transient unresponsive state of self-scratching behaviour is induced in mice by skin-scratching stimulation.
Topics: Analgesics, Non-Narcotic; Animals; Behavior, Animal; Calcitonin Gene-Related Peptide; Capsaicin; Disease Models, Animal; Male; Mice; Mice, Inbred ICR; Peptide Fragments; Physical Stimulation; Pruritus; Quinuclidines; Self Stimulation; Signal Transduction; Skin Physiological Phenomena; Substance P | 2007 |
Transient receptor potential vanilloid type 1 channels act as mechanoreceptors and cause substance P release and sensory activation in rat kidneys.
Topics: Action Potentials; Animals; Blood Pressure; Capsaicin; Cell Membrane; Cytosol; Diterpenes; Electrophysiology; Female; Kidney; Kidney Pelvis; Mechanoreceptors; Models, Biological; Neurokinin-1 Receptor Antagonists; Perfusion; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Sensory System Agents; Substance P; TRPV Cation Channels; Ubiquitin Thiolesterase | 2008 |
Interdependent regulation of afferent renal nerve activity and renal function: role of transient receptor potential vanilloid type 1, neurokinin 1, and calcitonin gene-related peptide receptors.
Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Ganglia, Spinal; Isoindoles; Kidney Pelvis; Male; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Peptide Fragments; Quinuclidines; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Substance P; TRPV Cation Channels | 2008 |
Effects of neurokinin-1 receptor agonism and antagonism in the rostral ventromedial medulla of rats with acute or persistent inflammatory nociception.
Topics: Animals; Capsaicin; Central Nervous System Agents; Freund's Adjuvant; Hot Temperature; Male; Medulla Oblongata; Mustard Plant; Neurokinin-1 Receptor Antagonists; Pain; Pain Measurement; Pain Threshold; Physical Stimulation; Piperidines; Plant Oils; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Time Factors | 2010 |
Cellular mechanism underlying formaldehyde-stimulated Cl- secretion in rat airway epithelium.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anions; Biological Transport; Capsaicin; Cells, Cultured; Chlorides; Colforsin; Epinephrine; Epithelial Cells; Formaldehyde; Imines; Male; Nerve Endings; ortho-Aminobenzoates; Quinuclidines; Rats; Respiratory Mucosa; Substance P; Trachea; TRPV Cation Channels | 2013 |