Page last updated: 2024-09-03

l 703606 and capsaicin

l 703606 has been researched along with capsaicin in 12 studies

Compound Research Comparison

Studies
(l 703606)
Trials
(l 703606)
Recent Studies (post-2010)
(l 703606)
Studies
(capsaicin)
Trials
(capsaicin)
Recent Studies (post-2010) (capsaicin)
7401211,2386613,410

Protein Interaction Comparison

ProteinTaxonomyl 703606 (IC50)capsaicin (IC50)
Transient receptor potential cation channel subfamily V member 1Rattus norvegicus (Norway rat)0.019
Lysine-specific histone demethylase 1AHomo sapiens (human)0.6
Bile salt export pumpHomo sapiens (human)10
Cytochrome P450 1A2Homo sapiens (human)3
Prostaglandin G/H synthase 1Homo sapiens (human)2.6755
Transient receptor potential cation channel subfamily V member 1Homo sapiens (human)0.008

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (16.67)18.2507
2000's8 (66.67)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bunnett, NW; Grady, EF; Martínez, V; Marvizón, JC; Mayer, EA1
Mustafa, S; Oriowo, MA1
Gear, RW; Levine, JD; Tambeli, CH; Young, A1
Horie, S; Minowa, S; Murayama, T; Someya, A; Tsuchiya, S1
Nies, M; Ro, JY; Zhang, Y1
Bell, EB; Beresford, LJ; Miyan, JA; Shepherd, AJ1
Fujiwara, N; Maeda, T; Seo, K; Someya, G; Takeuchi, K1
Kawana, S; Yamaoka, J1
Feng, NH; Lee, HH; Ma, MC; Shiang, JC1
Sachs, JR; Wang, DH; Xie, C1
Hamity, MV; Hammond, DL; White, SR1
Chen, PX; Guo, HM; Huang, JH; Luo, YL; Zhang, YL; Zhou, WL; Zhu, YX1

Other Studies

12 other study(ies) available for l 703606 and capsaicin

ArticleYear
Neurokinin 1 receptor internalization in spinal cord slices induced by dorsal root stimulation is mediated by NMDA receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Nov-01, Volume: 17, Issue:21

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Capsaicin; Electric Stimulation; Endocytosis; Evoked Potentials; Ganglia, Spinal; Hyperalgesia; Long-Term Potentiation; Male; Microscopy, Confocal; Microscopy, Fluorescence; Models, Neurological; N-Methylaspartate; Neurokinin-1 Receptor Antagonists; Quinuclidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Substance P

1997
Inhibitory effect of capsaicin on cholinergic transmission in ovine airways: evidence for non-cholinergic contractions.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Acetylcholine; Animals; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptides, Cyclic; Quinuclidines; Receptors, Drug; Receptors, Neurokinin-2; Serotonin; Sheep; Substance P; Synaptic Transmission; Trachea

1999
Contribution of spinal glutamatergic mechanisms in heterosegmental antinociception induced by noxious stimulation.
    Pain, 2003, Volume: 106, Issue:1-2

    Topics: Animals; Benzoates; Capsaicin; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Isoquinolines; Male; Nociceptors; Pyridines; Quinoxalines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Cord; Stimulation, Chemical; Substance P

2003
Role of neuropeptide receptor systems in vanilloid VR1 receptor-mediated gastric acid secretion in rat brain.
    European journal of pharmacology, 2004, Feb-23, Volume: 486, Issue:3

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Excitatory Amino Acid Antagonists; Gastric Acid; Hypothalamus; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Quinuclidines; Rats; Rats, Wistar; Receptor Cross-Talk; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Glutamate; Receptors, Neurokinin-2; Time Factors; TRPV Cation Channels

2004
Substance P does not play a critical role in neurogenic inflammation in the rat masseter muscle.
    Brain research, 2005, Jun-14, Volume: 1047, Issue:1

    Topics: Analgesics; Animals; Capsaicin; Disease Models, Animal; Edema; Inflammation Mediators; Male; Masseter Muscle; Mustard Plant; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Plant Extracts; Plant Oils; Pyrrolidonecarboxylic Acid; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P

2005
Mobilisation of specific T cells from lymph nodes in contact sensitivity requires substance P.
    Journal of neuroimmunology, 2005, Volume: 164, Issue:1-2

    Topics: Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cell Movement; Dermatitis, Contact; Dinitrochlorobenzene; Dose-Response Relationship, Drug; Drug Interactions; Immunohistochemistry; Lymph Nodes; Mice; Nerve Fibers; Quinuclidines; Skin; Substance P; Sympathectomy, Chemical; T-Lymphocytes

2005
Postnatal development of excitation propagation in the trigeminal subnucleus caudalis evoked by afferent stimulation in mice.
    Neuroscience research, 2005, Volume: 52, Issue:3

    Topics: Afferent Pathways; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Capsaicin; Diagnostic Imaging; Dizocilpine Maleate; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Neurokinin-1 Receptor Antagonists; Quinuclidines; Silver Staining; Time Factors; Trigeminal Caudal Nucleus

2005
A transient unresponsive state of self-scratching behaviour is induced in mice by skin-scratching stimulation.
    Experimental dermatology, 2007, Volume: 16, Issue:9

    Topics: Analgesics, Non-Narcotic; Animals; Behavior, Animal; Calcitonin Gene-Related Peptide; Capsaicin; Disease Models, Animal; Male; Mice; Mice, Inbred ICR; Peptide Fragments; Physical Stimulation; Pruritus; Quinuclidines; Self Stimulation; Signal Transduction; Skin Physiological Phenomena; Substance P

2007
Transient receptor potential vanilloid type 1 channels act as mechanoreceptors and cause substance P release and sensory activation in rat kidneys.
    American journal of physiology. Renal physiology, 2008, Volume: 294, Issue:2

    Topics: Action Potentials; Animals; Blood Pressure; Capsaicin; Cell Membrane; Cytosol; Diterpenes; Electrophysiology; Female; Kidney; Kidney Pelvis; Mechanoreceptors; Models, Biological; Neurokinin-1 Receptor Antagonists; Perfusion; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Sensory System Agents; Substance P; TRPV Cation Channels; Ubiquitin Thiolesterase

2008
Interdependent regulation of afferent renal nerve activity and renal function: role of transient receptor potential vanilloid type 1, neurokinin 1, and calcitonin gene-related peptide receptors.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 325, Issue:3

    Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Ganglia, Spinal; Isoindoles; Kidney Pelvis; Male; Neurokinin-1 Receptor Antagonists; Neurons, Afferent; Peptide Fragments; Quinuclidines; Rats; Rats, Wistar; Receptors, Calcitonin Gene-Related Peptide; Receptors, Neurokinin-1; Substance P; TRPV Cation Channels

2008
Effects of neurokinin-1 receptor agonism and antagonism in the rostral ventromedial medulla of rats with acute or persistent inflammatory nociception.
    Neuroscience, 2010, Feb-03, Volume: 165, Issue:3

    Topics: Animals; Capsaicin; Central Nervous System Agents; Freund's Adjuvant; Hot Temperature; Male; Medulla Oblongata; Mustard Plant; Neurokinin-1 Receptor Antagonists; Pain; Pain Measurement; Pain Threshold; Physical Stimulation; Piperidines; Plant Oils; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Time Factors

2010
Cellular mechanism underlying formaldehyde-stimulated Cl- secretion in rat airway epithelium.
    PloS one, 2013, Volume: 8, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Anions; Biological Transport; Capsaicin; Cells, Cultured; Chlorides; Colforsin; Epinephrine; Epithelial Cells; Formaldehyde; Imines; Male; Nerve Endings; ortho-Aminobenzoates; Quinuclidines; Rats; Respiratory Mucosa; Substance P; Trachea; TRPV Cation Channels

2013