l-697661 and r-82913
l-697661 has been researched along with r-82913 in 8 studies
Research
Studies (8)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Balani, SK; Ciccarone, TM; Condra, JH; Emini, EA; Goldman, ME; Greenlee, WJ; Kauffman, LR; MacTough, SC; Rooney, CS; Williams, TM | 1 |
Bell, FW; Cantrell, AS; Högberg, M; Jaskunas, SR; Johansson, NG; Jordan, CL; Kinnick, MD; Lind, P; Morin, JM; Noréen, R | 1 |
Cantrell, AS; Engelhardt, P; Högberg, M; Jaskunas, SR; Johansson, NG; Jordan, CL; Kangasmetsä, J; Kinnick, MD; Lind, P; Morin, JM; Muesing, MA; Noreén, R; Oberg, B; Pranc, P; Sahlberg, C; Ternansky, RJ; Vasileff, RT; Vrang, L; West, SJ; Zhang, H | 1 |
Condra, JH; Emini, EA; Gotlib, L; Graham, DJ; Lineberger, DW; Long, WJ; Sardana, VV; Schlabach, AJ; Wolfgang, JA | 1 |
Byrnes, VW; Condra, JH; Emini, EA; Sardana, VV; Schleif, WA | 1 |
Bäckbro, K; Noréen, R; Oberg, B; Unge, T; Vrang, L; Zhang, H | 1 |
Evans, DB; Fan, N; Rank, KB; Sharma, SK; Tarpley, WG; Thomas, RC | 1 |
Chen, IS; Dueweke, TJ; Poppe, SM; Pushkarskaya, T; Stevenson, M; Swaney, SM; Tarpley, WG; Zhao, JQ | 1 |
Reviews
1 review(s) available for l-697661 and r-82913
Article | Year |
---|---|
The genetic and functional basis of HIV-1 resistance to nonnucleoside reverse transcriptase inhibitors.
Topics: Antiviral Agents; Benzodiazepines; Benzoxazoles; Clinical Trials as Topic; Drug Resistance, Microbial; Genetic Variation; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Imidazoles; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1994 |
Other Studies
7 other study(ies) available for l-697661 and r-82913
Article | Year |
---|---|
5-chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase.
Topics: Animals; Antiviral Agents; Base Sequence; Biological Availability; HIV; HIV Reverse Transcriptase; HIV-1; Indoles; Macaca mulatta; Molecular Sequence Data; Molecular Structure; Reverse Transcriptase Inhibitors; Sulfoxides | 1993 |
Phenethylthiazolethiourea (PETT) compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure-activity relationship studies of PETT analogs.
Topics: Animals; Antiviral Agents; Cell Line; HIV-1; Humans; Isothiocyanates; Rats; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles; Thiourea | 1995 |
Phenethylthiazolylthiourea (PETT) compounds as a new class of HIV-1 reverse transcriptase inhibitors. 2. Synthesis and further structure-activity relationship studies of PETT analogs.
Topics: Animals; Anti-HIV Agents; Cells, Cultured; HIV Reverse Transcriptase; Intercalating Agents; Structure-Activity Relationship; Thiazoles; Thiourea | 1996 |
Functional analysis of HIV-1 reverse transcriptase amino acids involved in resistance to multiple nonnucleoside inhibitors.
Topics: Amino Acid Sequence; Antiviral Agents; Azepines; Benzodiazepines; Benzoxazoles; Drug Resistance, Microbial; HIV Reverse Transcriptase; HIV-1; Imidazoles; Kinetics; Mutagenesis, Site-Directed; Nevirapine; Pyridines; Pyridones; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Structure-Activity Relationship | 1992 |
Enzymatic properties and sensitivity to inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase with Glu-138-->Arg and Tyr-188-->His mutations.
Topics: Amino Acids; Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Binding, Competitive; Deoxyguanine Nucleotides; Dideoxynucleotides; Foscarnet; HIV Reverse Transcriptase; Humans; Imidazoles; Kinetics; Molecular Sequence Data; Mutation; Nevirapine; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Sensitivity and Specificity | 1994 |
Simultaneous mutations at Tyr-181 and Tyr-188 in HIV-1 reverse transcriptase prevents inhibition of RNA-dependent DNA polymerase activity by the bisheteroarylpiperazine (BHAP) U-90152s.
Topics: Amino Acid Sequence; Antiviral Agents; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; HIV Reverse Transcriptase; HIV-1; HIV-2; Imidazoles; Indoles; Kinetics; Molecular Sequence Data; Mutagenesis, Site-Directed; Nevirapine; Piperazines; Point Mutation; Pyridines; Pyridones; Recombinant Fusion Proteins; Recombinant Proteins; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Tyrosine | 1995 |
A mutation in reverse transcriptase of bis(heteroaryl)piperazine-resistant human immunodeficiency virus type 1 that confers increased sensitivity to other nonnucleoside inhibitors.
Topics: Antiviral Agents; Base Sequence; Benzodiazepines; Benzoxazoles; Cloning, Molecular; Delavirdine; Drug Resistance; HIV Reverse Transcriptase; Imidazoles; Indoles; Molecular Sequence Data; Mutation; Nevirapine; Oligodeoxyribonucleotides; Piperazines; Pyridines; Pyridones; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase | 1993 |