Page last updated: 2024-09-03

l 694247 and ritanserin

l 694247 has been researched along with ritanserin in 3 studies

Compound Research Comparison

Studies
(l 694247)
Trials
(l 694247)
Recent Studies (post-2010)
(l 694247)
Studies
(ritanserin)
Trials
(ritanserin)
Recent Studies (post-2010) (ritanserin)
32087357571

Protein Interaction Comparison

ProteinTaxonomyl 694247 (IC50)ritanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.001
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.047
Diacylglycerol kinase alphaHomo sapiens (human)9
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.047
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.047
D(2) dopamine receptorRattus norvegicus (Norway rat)0.012

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Böing, C; Bühlen, M; Fink, K; Göthert, M1
Bult, H; Geerts, IS; Herman, AG; Matthys, KE1
Calama, E; Martín, ML; Morán, A; Ortíz de Urbina, AV; San Román, L1

Other Studies

3 other study(ies) available for l 694247 and ritanserin

ArticleYear
Evidence for presynaptic location of inhibitory 5-HT1D beta-like autoreceptors in the guinea-pig brain cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: Animals; Autoreceptors; Binding, Competitive; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Ketanserin; Male; Methiothepin; Oxadiazoles; Oxymetazoline; Potassium; Radioligand Assay; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Synaptosomes; Tritium; Tryptamines

1996
Involvement of 5-HT1B receptors in collar-induced hypersensitivity to 5-hydroxytryptamine of the rabbit carotid artery.
    British journal of pharmacology, 1999, Volume: 127, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Braces; Carotid Arteries; Dose-Response Relationship, Drug; Hypersensitivity; In Vitro Techniques; Ketanserin; Male; Methysergide; Oxadiazoles; Piperazines; Potassium Chloride; Rabbits; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sumatriptan; Tryptamines; Vasoconstriction

1999
Effect of 5-hydroxytryptamine on neurogenic vasoconstriction in the isolated, autoperfused hindquarters of the rat.
    Clinical and experimental pharmacology & physiology, 2005, Volume: 32, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Biguanides; Biphenyl Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Hindlimb; In Vitro Techniques; Infusions, Intravenous; Male; Methiothepin; Oxadiazoles; Perfusion; Piperazines; Pressure; Quinoxalines; Rats; Rats, Wistar; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT3 Receptor Agonists; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Tryptamines; Vasoconstriction

2005