Page last updated: 2024-09-03

l 663581 and zolpidem

l 663581 has been researched along with zolpidem in 4 studies

Compound Research Comparison

Studies
(l 663581)
Trials
(l 663581)
Recent Studies (post-2010)
(l 663581)
Studies
(zolpidem)
Trials
(zolpidem)
Recent Studies (post-2010) (zolpidem)
12001,825368683

Protein Interaction Comparison

ProteinTaxonomyl 663581 (IC50)zolpidem (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.048
Translocator proteinRattus norvegicus (Norway rat)4.7
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.048
GABA theta subunitRattus norvegicus (Norway rat)0.048
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.048

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cook, JM; Dayer, CA; He, X; Huang, Q; Liu, R; Ma, C; McKernan, R; Wenger, GR; Yu, S1
Jackson, A1
Dawson, G; Draper, F; Jackson, A; Roe, S; Stanhope, KJ1
Hadingham, KL; Palmer, KJ; Thompson, SA; Wafford, KA; Whiting, PJ1

Other Studies

4 other study(ies) available for l 663581 and zolpidem

ArticleYear
Pharmacophore/receptor models for GABA(A)/BzR subtypes (alpha1beta3gamma2, alpha5beta3gamma2, and alpha6beta3gamma2) via a comprehensive ligand-mapping approach.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Animals; Benzodiazepines; Carbolines; Cell Line; Columbidae; Conditioning, Operant; Crystallography, X-Ray; Humans; Indoles; Ligands; Male; Models, Molecular; Pyrimidines; Quinolones; Radioligand Assay; Receptors, GABA-A; Saimiri; Stereoisomerism; Structure-Activity Relationship

2000
State-dependent effects of atypical benzodiazepine-receptor agonists.
    Psychopharmacology, 1995, Volume: 119, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Benzodiazepines; Benzodiazepinones; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Pyridines; Rats; Rats, Wistar; Zolpidem

1995
Effect of the benzodiazepine receptor agonist, zolpidem, on palatable fluid consumption in the rat.
    Psychopharmacology, 1993, Volume: 111, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepines; Benzodiazepinones; Dose-Response Relationship, Drug; Drinking Behavior; Environment; GABA-A Receptor Agonists; Glucose; Hypnotics and Sedatives; Male; Motivation; Pyridines; Rats; Zolpidem

1993
Expression and pharmacology of human GABAA receptors containing gamma 3 subunits.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Base Sequence; Benzodiazepines; Benzodiazepinones; Carbolines; Flumazenil; Flunitrazepam; GABA Modulators; Humans; Molecular Sequence Data; Pyrazoles; Pyridazines; Pyridines; Receptors, GABA-A; Recombinant Proteins; Sequence Homology, Amino Acid; Triazolam; Xenopus; Zolpidem

1995