Compounds > l 655240
Page last updated: 2024-09-03

l 655240 and l 663536

l 655240 has been researched along with l 663536 in 2 studies

Compound Research Comparison

Studies
(l 655240)		Trials
(l 655240)		Recent Studies (post-2010)
(l 655240)		Studies
(l 663536)		Trials
(l 663536)		Recent Studies (post-2010) (l 663536)
26044854138

Protein Interaction Comparison

ProteinTaxonomyl 655240 (IC50)l 663536 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.023
Prostaglandin E synthaseHomo sapiens (human)2.2274
Prostaglandin G/H synthase 1Ovis aries (sheep)8
Polyunsaturated fatty acid 5-lipoxygenaseHomo sapiens (human)0.57
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.023
Arachidonate 5-lipoxygenase-activating proteinHomo sapiens (human)0.025
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.023
Prostaglandin G/H synthase 2Homo sapiens (human)2.4
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.023
Leukotriene C4 synthaseHomo sapiens (human)3
Macrophage-expressed gene 1 proteinHomo sapiens (human)2.2
GABA theta subunitRattus norvegicus (Norway rat)0.023
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.023
Prostaglandin E synthase 2Homo sapiens (human)1.6

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aspiotis, R; Ethier, D; Friesen, RW; Gareau, Y; Grimm, EL; Guay, J; Guiral, S; Juteau, H; Mancini, JA; Méthot, N; Riendeau, D; Rubin, J1
Borgeat, P; Laviolette, M; Ménard, L; Naccache, PH; Pilote, S1

Other Studies

2 other study(ies) available for l 655240 and l 663536

ArticleYear
Inhibitors of the inducible microsomal prostaglandin E2 synthase (mPGES-1) derived from MK-886.
    Bioorganic & medicinal chemistry letters, 2005, Jul-15, Volume: 15, Issue:14

    Topics: Cell Line, Tumor; Cell Proliferation; Cyclooxygenase Inhibitors; Humans; Indoles; Intramolecular Oxidoreductases; Microsomes; Prostaglandin-E Synthases; Structure-Activity Relationship

2005
Inhibitory effects of MK-886 on arachidonic acid metabolism in human phagocytes.
    British journal of pharmacology, 1990, Volume: 100, Issue:1

    Topics: Actins; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Cell Survival; Chromatography, High Pressure Liquid; Colony-Stimulating Factors; Eosinophils; Humans; In Vitro Techniques; Indoles; Leukotriene Antagonists; Leukotrienes; Neutrophils; Phagocytes; Platelet Activating Factor; Superoxides

1990