Page last updated: 2024-09-03

l 648051 and pyrilamine

l 648051 has been researched along with pyrilamine in 2 studies

Compound Research Comparison

Studies
(l 648051)
Trials
(l 648051)
Recent Studies (post-2010)
(l 648051)
Studies
(pyrilamine)
Trials
(pyrilamine)
Recent Studies (post-2010) (pyrilamine)
24601,86026116

Protein Interaction Comparison

ProteinTaxonomyl 648051 (IC50)pyrilamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.13
Alpha-2A adrenergic receptorHomo sapiens (human)2.976
Cytochrome P450 2D6Homo sapiens (human)0.3
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.997
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.13
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.0015
Histamine H1 receptorRattus norvegicus (Norway rat)0.0126
Sodium-dependent serotonin transporterHomo sapiens (human)0.047
Histamine H1 receptorHomo sapiens (human)0.0166
5-hydroxytryptamine receptor 2BHomo sapiens (human)2.788
Sodium-dependent dopamine transporter Homo sapiens (human)0.879
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.1
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.558

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19902 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Björck, T; Dahlén, SE1
Charette, L; Denis, D; Jones, TR1

Other Studies

2 other study(ies) available for l 648051 and pyrilamine

ArticleYear
Evidence indicating that leukotrienes C4, D4 and E4 are major mediators of contraction induced by anti-IgE in human bronchi.
    Agents and actions, 1989, Volume: 26, Issue:1-2

    Topics: Acetylcholine; Antibodies, Anti-Idiotypic; Bronchi; Histamine; Humans; Immunoglobulin E; Keto Acids; Leukotriene E4; Leukotrienes; Metiamide; Muscle Contraction; Phenylbutyrates; Pyrilamine; SRS-A; Sulfones

1989
Leukotriene and anti-IgE induced contractions of human isolated trachea: studies with leukotriene receptor antagonists and a novel 5-lipoxygenase inhibitor.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:6

    Topics: Animals; Antibodies, Anti-Idiotypic; Arachidonate Lipoxygenases; Atropine; Benzofurans; Chromones; Goats; Humans; In Vitro Techniques; Indomethacin; Keto Acids; Lipoxygenase Inhibitors; Muscle Contraction; Phenylbutyrates; Pyrilamine; Receptors, Leukotriene; Receptors, Prostaglandin; SRS-A; Sulfones; Trachea

1988