l 365031 has been researched along with devazepide in 4 studies
| Studies (l 365031) | Trials (l 365031) | Recent Studies (post-2010) (l 365031) | Studies (devazepide) | Trials (devazepide) | Recent Studies (post-2010) (devazepide) |
|---|---|---|---|---|---|
| 7 | 0 | 0 | 780 | 5 | 42 |
| Protein | Taxonomy | l 365031 (IC50) | devazepide (IC50) |
|---|---|---|---|
| Bile salt export pump | Homo sapiens (human) | 10 | |
| Cholecystokinin receptor type A | Rattus norvegicus (Norway rat) | 0.0009 | |
| Gastrin/cholecystokinin type B receptor | Rattus norvegicus (Norway rat) | 0.0008 | |
| Cholecystokinin receptor type A | Homo sapiens (human) | 0.0002 | |
| Gastrin/cholecystokinin type B receptor | Homo sapiens (human) | 0.245 | |
| Cholecystokinin receptor type A | Cavia porcellus (domestic guinea pig) | 0.27 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 2 (50.00) | 18.7374 |
| 1990's | 2 (50.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Anderson, PS; Bock, MG; Chang, RS; DiPardo, RM; Evans, BE; Freidinger, RM; Lundell, GF; Rittle, KE; Veber, DF; Whitter, WL | 1 |
| Hopfinger, AJ; Tokarski, JS | 1 |
| Campbell, NJ; Hill, DR; Shaw, TM; Woodruff, GN | 1 |
| Dourish, CT; Hendrie, CA; Neill, JC; Shepherd, JK | 1 |
4 other study(ies) available for l 365031 and devazepide
| Article | Year |
|---|---|
Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists.
Topics: Administration, Oral; Animals; Benzodiazepines; Chemical Phenomena; Chemistry; Cholecystokinin; Drug Design; Mice; Receptors, Cholecystokinin; Receptors, GABA-A; Structure-Activity Relationship | 1988 |
Three-dimensional molecular shape analysis-quantitative structure-activity relationship of a series of cholecystokinin-A receptor antagonists.
Topics: Animals; Benzodiazepines; Chemical Phenomena; Chemistry, Physical; Crystallization; Crystallography, X-Ray; Guinea Pigs; Lipid Metabolism; Molecular Conformation; Molecular Structure; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Structure-Activity Relationship; Thermodynamics | 1994 |
Autoradiographic localization and biochemical characterization of peripheral type CCK receptors in rat CNS using highly selective nonpeptide CCK antagonists.
Topics: Animals; Autoradiography; Benzodiazepinones; Brain Chemistry; Devazepide; Guinea Pigs; Male; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Sincalide | 1987 |
The effects of CCKA and CCKB antagonists on activity in the black/white exploration model of anxiety in mice.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Exploratory Behavior; Male; Mice; Mice, Inbred DBA; Phenylurea Compounds; Receptors, Cholecystokinin | 1993 |