Page last updated: 2024-09-05

l 163191 and fedratinib

l 163191 has been researched along with fedratinib in 1 studies

Compound Research Comparison

Studies
(l 163191)
Trials
(l 163191)
Recent Studies (post-2010)
(l 163191)
Studies
(fedratinib)
Trials
(fedratinib)
Recent Studies (post-2010) (fedratinib)
3501712016111

Protein Interaction Comparison

ProteinTaxonomyl 163191 (IC50)fedratinib (IC50)
Cyclin-G-associated kinaseHomo sapiens (human)0.001
Tyrosine-protein kinase JAK2Homo sapiens (human)0.0035
Bromodomain-containing protein 4Homo sapiens (human)0.29
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)0.0325
Tyrosine-protein kinase JAK1Homo sapiens (human)0.053
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)0.078
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)0.02
Tyrosine-protein kinase JAK3Homo sapiens (human)0.3917
AP2-associated protein kinase 1Homo sapiens (human)0.032
Bromodomain testis-specific proteinHomo sapiens (human)0.34

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1

Other Studies

1 other study(ies) available for l 163191 and fedratinib

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013