kynurenic acid and piperidines

kynurenic acid has been researched along with piperidines in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's24 (61.54)18.2507
2000's11 (28.21)29.6817
2010's4 (10.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Nicklas, WJ; Zeevalk, GD1
Baron, BM; Chi, EM; Harrison, BL; Kehne, JH; McCloskey, TC; Palfreyman, MG; Whitten, JP1
Canton, H; Colpaert, F; Lehmann, J1
Bowen, DM; Cross, AJ; Francis, PT; Green, AR; Steele, JE1
Ferkany, JW; Kaplita, PV1
Ammendola, D; De Sarro, A; De Sarro, G; Nava, F1
Oblin, A; Schoemaker, H1
Carter, C; Fage, D; Voltz, C1
Ogita, K; Suzuki, T; Yoneda, Y1
Layer, RT; Olds, T; Popik, P; Skolnick, P1
Lu, L; Luo, J; McGonigle, P; Munir, M; Wang, YH; Wolfe, BB1
Doyle, KM; Shaw, GG1
Aulakh, CS; Mazzola-Pomietto, P; Murphy, DL1
Couratier, P; Dussartre, C; Hugon, J; Lesort, M; Terro, F1
Johnson, SW; Wu, YN1
Aizenman, E; Boeckman, FA1
Misawa, M; Suzuki, T; Tsuda, M2
Leibrock, J; Prücher, H; Rautenberg, W1
Camarasa, J; Camins, A; Escubedo, E; Gabriel, C; Pallàs, M; Sureda, FX1
Daggett, LP; Deal, C; Hess, SD; Johnson, EC; Lu, CC; Veliçelebi, G1
Abdrachmanova, G; Palecek, JI; Vlachová, V; Vyklick, L1
Bear, MF; Huganir, RL; Philpot, BD; Quinlan, EM1
Arvigo, D; Bonfanti, A; Pittaluga, A; Raiteri, M1
Bunney, BS; Shi, WX; Zhang, XX1
Gemignani, A; Paudice, P; Pittaluga, A; Raiteri, M1
Bakalkin, G; Esashi, A; Kisara, K; Nakagawasai, O; Niijima, F; Sakurada, C; Sakurada, T; Tadano, T; Tan-No, K; Terenius, L1
Boros, A; Dezso, P; Kolok, S; Nagy, J; Szombathelyi, Z1
Ogonowski, AA; Smith, JB1
Borza, I; Domány, G; Farkas, S; Galgóczy, K; Gere, A; Greiner, I; Horváth, C; Kolok, S1
Esashi, A; Furuta, S; Nakagawasai, O; Niijima, F; Sato, T; Satoh, S; Tadano, T; Tan-No, K; Yasuhara, H1
Gómez-Urquijo, S; Morera-Herreras, T; Ruiz-Ortega, JA; Ugedo, L1
Han, TZ; Li, YH; Meng, K1
Kloc, R; Luchowska, E; Owe-Larsson, B; Urbanska, EM; Wielosz, M1
Jean, A; Lebrun, B; Roux, J; Trouslard, J; Wanaverbecq, N1
Ahn, DK; Bae, YC; Bonfa, E; Park, MK; Woo, YW; Yang, GY1
Ahn, DK; Bae, YC; Kim, MJ; Lee, JH; Park, MK; Park, YY; Won, KA; Yang, GY1
Fukunaga, K; Moriguchi, S; Narahashi, T; Tanaka, T1
Fischer, MJ; Kageneck, C; Messlinger, K; Nixdorf-Bergweiler, BE1

Other Studies

39 other study(ies) available for kynurenic acid and piperidines

ArticleYear
Developmental differences in antagonism of NMDA toxicity by the polyamine site antagonist ifenprodil.
    Brain research. Developmental brain research, 1992, Feb-21, Volume: 65, Issue:2

    Topics: Amino Acids; Animals; Biogenic Polyamines; Chick Embryo; Dizocilpine Maleate; Kynurenic Acid; N-Methylaspartate; Pipecolic Acids; Piperidines; Receptors, Glutamate; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Receptors, Phencyclidine; Retina

1992
NMDA receptor complex antagonists have potential anxiolytic effects as measured with separation-induced ultrasonic vocalizations.
    European journal of pharmacology, 1991, Feb-14, Volume: 193, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Anxiety, Separation; Behavior, Animal; Buspirone; Diazepam; Dioxins; Dizocilpine Maleate; Dose-Response Relationship, Drug; Indoles; Kynurenic Acid; Maternal Deprivation; Mephenesin; Piperidines; Quinolizines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Serotonin Antagonists; Spiro Compounds; Valine; Vocalization, Animal

1991
Glutamate and glycine co-activate while polyamines merely modulate the NMDA receptor complex.
    Progress in neuro-psychopharmacology & biological psychiatry, 1991, Volume: 15, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Adrenergic alpha-Antagonists; Animals; Biguanides; Binding, Competitive; Biogenic Polyamines; Biotransformation; Brain; Dizocilpine Maleate; Glutamates; Glutamic Acid; Glycine; In Vitro Techniques; Kynurenic Acid; Piperidines; Rats; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine

1991
Spermidine enhancement of [3H]MK-801 binding to the NMDA receptor complex in human cortical membranes.
    European journal of pharmacology, 1990, Sep-18, Volume: 189, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Cerebral Cortex; Dizocilpine Maleate; Female; Humans; In Vitro Techniques; Kynurenic Acid; Male; Membranes; Piperidines; Radioligand Assay; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Spermidine

1990
Evidence for direct interactions between the NMDA and glycine recognition sites in brain.
    European journal of pharmacology, 1990, Mar-13, Volume: 188, Issue:2-3

    Topics: Amino Acids; Animals; Brain Chemistry; In Vitro Techniques; Kynurenic Acid; Male; Pipecolic Acids; Piperazines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Neurotransmitter; Serine

1990
Effects of some excitatory amino acid antagonists on imipenem-induced seizures in DBA/2 mice.
    Brain research, 1995, Feb-06, Volume: 671, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amino Acids; Animals; Anticonvulsants; Dizocilpine Maleate; Excitatory Amino Acids; Glutamine; Imipenem; Kynurenic Acid; Mice; Mice, Inbred DBA; Muscimol; Piperazines; Piperidines; Quinoxalines; Seizures

1995
Complex allosteric modulation of the binding of the NMDA receptor antagonist [3H]CGP39653.
    European journal of pharmacology, 1994, Jan-01, Volume: 266, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Allosteric Regulation; Animals; Biguanides; Binding Sites; Glycine; In Vitro Techniques; Kynurenic Acid; Male; Piperidines; Prosencephalon; Putrescine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine

1994
Synergism between the NMDA receptor antagonistic effects of ifenprodil and the glycine antagonist, 7-chlorokynurenate, in vivo.
    European journal of pharmacology, 1994, Apr-01, Volume: 255, Issue:1-3

    Topics: Animals; Chromatography, High Pressure Liquid; Drug Synergism; Glycine; Injections; Kynurenic Acid; Male; N-Methylaspartate; Neostriatum; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermidine; Spermine

1994
Differential profiles of binding of a radiolabeled agonist and antagonist at a glycine recognition domain on the N-methyl-D-aspartate receptor ionophore complex in rat brain.
    Journal of neurochemistry, 1994, Volume: 62, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Glycine; Kinetics; Kynurenic Acid; Male; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes; Tritium

1994
Antidepressant-like actions of the polyamine site NMDA antagonist, eliprodil (SL-82.0715).
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:3

    Topics: Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Animals; Antidepressive Agents; Behavior, Animal; Biogenic Polyamines; Brain Chemistry; Down-Regulation; Excitatory Amino Acid Antagonists; Glycine; Imipramine; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Motor Activity; Piperidines; Receptors, Glycine

1995
Pharmacological and immunological characterization of N-methyl-D-aspartate receptors in human NT2-N neurons.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Glutamic Acid; Humans; Immunoblotting; Kynurenic Acid; Neurons; Piperidines; Putrescine; Rats; Receptors, N-Methyl-D-Aspartate

1996
Investigation of the involvement of the N-methyl-D-aspartate receptor macrocomplex in the development of spermine-induced CNS excitation in vivo.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Animals; Brain; Cerebral Ventricles; Dizocilpine Maleate; Female; Kynurenic Acid; Mice; Neuroprotective Agents; Piperazines; Piperidines; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Seizures; Spermine; Tremor

1996
NMDA receptor antagonists block development of tolerance to m-CPP-induced increases in ACTH concentrations in rats.
    European journal of pharmacology, 1996, Jul-25, Volume: 308, Issue:3

    Topics: Adrenocorticotropic Hormone; Animals; Dimethyl Sulfoxide; Dizocilpine Maleate; Drug Tolerance; Kynurenic Acid; Male; Phencyclidine; Piperazines; Piperidines; Pyrrolidinones; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Serotonin Receptor Agonists

1996
NMDA antagonist blockade of AT8 tau immunoreactive changes in neuronal cultures.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Cell Survival; Cells, Cultured; Cerebral Cortex; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Female; Fetus; Fluorescent Antibody Technique; Kynurenic Acid; Microscopy, Confocal; Neurons; Piperidines; Pregnancy; Rats; Receptors, N-Methyl-D-Aspartate; tau Proteins

1996
Pharmacological characterization of inward current evoked by N-methyl-D-aspartate in dopamine neurons in the rat brain slice.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Animals; Dizocilpine Maleate; Excitatory Amino Acid Agonists; In Vitro Techniques; Kynurenic Acid; Magnesium; Male; Membrane Potentials; N-Methylaspartate; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Sodium; Spermine; Substantia Nigra; Ventral Tegmental Area

1996
Pharmacological properties of acquired excitotoxicity in Chinese hamster ovary cells transfected with N-methyl-D-aspartate receptor subunits.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Animals; Calcium; Cell Survival; CHO Cells; Cricetinae; Dizocilpine Maleate; Kynurenic Acid; L-Lactate Dehydrogenase; Luciferases; Pipecolic Acids; Piperidines; Receptors, N-Methyl-D-Aspartate; Transfection

1996
Role of the NMDA receptor complex in DMCM-induced seizure in mice.
    Neuroreport, 1997, Feb-10, Volume: 8, Issue:3

    Topics: Animals; Carbolines; Cerebral Ventricles; Convulsants; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Infusions, Intravenous; Injections, Intraventricular; Injections, Spinal; Kynurenic Acid; Male; Mice; Mice, Inbred Strains; Phencyclidine; Piperidines; Receptors, N-Methyl-D-Aspartate; Seizures; Spinal Cord

1997
Recovery of decreased seizure threshold for pentylenetetrazole during diazepam withdrawal by NMDA receptor antagonists.
    European journal of pharmacology, 1997, Apr-11, Volume: 324, Issue:1

    Topics: Animals; Anticonvulsants; Convulsants; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Drug Interactions; Excitatory Amino Acid Antagonists; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Subcutaneous; Kynurenic Acid; Male; Mice; Neuroprotective Agents; Pentylenetetrazole; Piperidines; Receptors, N-Methyl-D-Aspartate; Seizures; Substance Withdrawal Syndrome

1997
EMD 95885, a new eliprodil analogue with higher affinity for the N-methyl-D-aspartate (NMDA) receptor.
    Die Pharmazie, 1997, Volume: 52, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Binding, Competitive; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Kainic Acid; Kynurenic Acid; Male; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate

1997
Modulation of neuronal mitochondrial membrane potential by the NMDA receptor: role of arachidonic acid.
    Brain research, 1997, Nov-28, Volume: 777, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Anesthetics, Local; Animals; Arachidonic Acid; Biomarkers; Cells, Cultured; Cerebellum; Dibucaine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Flow Cytometry; Fluorescent Dyes; Glycine; Intracellular Membranes; Kynurenic Acid; Membrane Potentials; Mitochondria; N-Methylaspartate; Piperidines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Rhodamine 123; Rhodamines; Sulfonamides

1997
Functional characterization of human N-methyl-D-aspartate subtype 1A/2D receptors.
    Journal of neurochemistry, 1998, Volume: 70, Issue:3

    Topics: Animals; Calcium; Cells, Cultured; DNA, Complementary; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fetus; Glutamic Acid; Glycine; Humans; Kidney; Kynurenic Acid; Membrane Potentials; Molecular Sequence Data; N-Methylaspartate; Oocytes; Patch-Clamp Techniques; Pipecolic Acids; Piperidines; Receptors, N-Methyl-D-Aspartate; Recombinant Proteins; Sequence Homology, Amino Acid; Serine; Xenopus laevis

1998
Properties of NMDA receptors in rat spinal cord motoneurons.
    The European journal of neuroscience, 1999, Volume: 11, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Age Factors; Animals; Animals, Newborn; Electric Conductivity; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Glycine; Ion Channel Gating; Kainic Acid; Kynurenic Acid; Magnesium; Male; Motor Neurons; N-Methylaspartate; Organ Culture Techniques; Patch-Clamp Techniques; Piperidines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spinal Cord

1999
Rapid, experience-dependent expression of synaptic NMDA receptors in visual cortex in vivo.
    Nature neuroscience, 1999, Volume: 2, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Animals, Suckling; Bicuculline; Cycloheximide; Darkness; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; Gene Expression Regulation, Developmental; Glycine; Kynurenic Acid; Light; Male; Models, Neurological; Nerve Tissue Proteins; Neuronal Plasticity; Optic Nerve; Photic Stimulation; Piperidines; Protein Synthesis Inhibitors; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Sensory Deprivation; Synapses; Vision, Ocular; Visual Cortex; Zinc

1999
Aniracetam, 1-BCP and cyclothiazide differentially modulate the function of NMDA and AMPA receptors mediating enhancement of noradrenaline release in rat hippocampal slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Dioxoles; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Heterocyclic Compounds; Hippocampus; In Vitro Techniques; Kynurenic Acid; Male; N-Methylaspartate; Nootropic Agents; Norepinephrine; Piperidines; Pyrrolidinones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tritium

1999
Enhancement of NMDA-induced current by the putative NR2B selective antagonist ifenprodil.
    Synapse (New York, N.Y.), 2000, Volume: 37, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Kynurenic Acid; Male; Membrane Potentials; N-Methylaspartate; Organ Culture Techniques; Piperidines; Prefrontal Cortex; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spermine

2000
The HIV-1 coat protein gp120 and some of its fragments potently activate native cerebral NMDA receptors mediating neuropeptide release.
    The European journal of neuroscience, 2000, Volume: 12, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; Animals; Cerebral Cortex; Cholecystokinin; Dizocilpine Maleate; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; HIV Envelope Protein gp120; HIV-1; Indoles; Kynurenic Acid; Male; Maleimides; Neurons; Nitroarginine; Peptide Fragments; Pipecolic Acids; Piperazines; Piperidines; Potassium; Protein Structure, Tertiary; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Somatostatin; Synaptic Transmission; Synaptosomes; Zinc

2000
Intrathecally administered big dynorphin, a prodynorphin-derived peptide, produces nociceptive behavior through an N-methyl-D-aspartate receptor mechanism.
    Brain research, 2002, Oct-11, Volume: 952, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analgesics, Opioid; Animals; Behavior, Animal; Dizocilpine Maleate; Dynorphins; Endorphins; Enkephalins; Excitatory Amino Acid Antagonists; Injections, Spinal; Kynurenic Acid; Male; Mice; Morphine; Neurokinin A; Nociceptors; Peptide Fragments; Piperidines; Protein Precursors; Receptors, N-Methyl-D-Aspartate; Receptors, Tachykinin; Substance P

2002
Differential alterations in the expression of NMDA receptor subunits following chronic ethanol treatment in primary cultures of rat cortical and hippocampal neurones.
    Neurochemistry international, 2003, Volume: 42, Issue:1

    Topics: Animals; Animals, Newborn; Cells, Cultured; Cerebral Cortex; Culture Media, Serum-Free; Dizocilpine Maleate; Ethanol; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Hippocampus; Kynurenic Acid; N-Methylaspartate; Nerve Tissue Proteins; Neurons; Piperidines; Protein Subunits; Rats; Receptors, N-Methyl-D-Aspartate; RNA Splicing

2003
Behavioral effects of NMDA receptor agonists and antagonists in combination with nitric oxide-related compounds.
    European journal of pharmacology, 2003, Jun-20, Volume: 471, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Arginine; Conditioning, Operant; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Gallic Acid; Guanidines; Indazoles; Injections, Intraperitoneal; Kynurenic Acid; Molsidomine; N-Methylaspartate; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitroprusside; Phencyclidine; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

2003
Kynurenic acid amides as novel NR2B selective NMDA receptor antagonists.
    Bioorganic & medicinal chemistry letters, 2007, Jan-15, Volume: 17, Issue:2

    Topics: Amides; Analgesics; Animals; Binding Sites; Chromatography, High Pressure Liquid; Formaldehyde; Indicators and Reagents; Kynurenic Acid; Magnetic Resonance Spectroscopy; Mice; Pain Measurement; Piperidines; Receptors, N-Methyl-D-Aspartate; Spectrophotometry, Infrared; Structure-Activity Relationship

2007
Intrathecally administered D-cycloserine produces nociceptive behavior through the activation of N-methyl-D-aspartate receptor ion-channel complex acting on the glycine recognition site.
    Journal of pharmacological sciences, 2007, Volume: 104, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Agmatine; Animals; Cycloserine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Injections, Spinal; Ion Channels; Kynurenic Acid; Mice; Morphine; Neurokinin A; Nociceptors; Pain; Peptide Fragments; Piperidines; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Receptors, Tachykinin; Substance P

2007
Involvement of subthalamic nucleus in the stimulatory effect of Delta(9)-tetrahydrocannabinol on dopaminergic neurons.
    Neuroscience, 2008, Feb-06, Volume: 151, Issue:3

    Topics: Action Potentials; Analysis of Variance; Animals; Apomorphine; Dopamine; Dopamine Agonists; Dose-Response Relationship, Drug; Dronabinol; Excitatory Amino Acid Agonists; Ibotenic Acid; Kynurenic Acid; Male; Neurons; Piperidines; Psychotropic Drugs; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant; Substantia Nigra; Subthalamic Nucleus

2008
Tonic facilitation of glutamate release by glycine binding sites on presynaptic NR2B-containing NMDA autoreceptors in the rat visual cortex.
    Neuroscience letters, 2008, Feb-27, Volume: 432, Issue:3

    Topics: Animals; Animals, Newborn; Binding Sites; Dizocilpine Maleate; Drug Interactions; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; In Vitro Techniques; Kynurenic Acid; Patch-Clamp Techniques; Phenols; Piperidines; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Visual Cortex

2008
Memantine increases brain production of kynurenic acid via protein kinase A-dependent mechanism.
    Neuroscience letters, 2008, Apr-18, Volume: 435, Issue:2

    Topics: Analysis of Variance; Animals; Animals, Newborn; Brain; Carbazoles; Cells, Cultured; Chromatography, High Pressure Liquid; Cyclic AMP-Dependent Protein Kinases; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; In Vitro Techniques; Isoquinolines; Kynurenic Acid; Male; Memantine; Neurons; Piperidines; Pyrroles; Rats; Rats, Wistar

2008
Depolarization-induced release of endocannabinoids by murine dorsal motor nucleus of the vagus nerve neurons differentially regulates inhibitory and excitatory neurotransmission.
    Neuropharmacology, 2009, Volume: 56, Issue:8

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Arachidonic Acids; Benzoxazines; Brain Stem; Calcium Signaling; Cannabinoid Receptor Modulators; Capsaicin; Efferent Pathways; Endocannabinoids; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Inhibitory Postsynaptic Potentials; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Morpholines; Naphthalenes; Neurons; Piperidines; Pyrazoles; Pyridazines; Receptor, Cannabinoid, CB1; Receptors, Presynaptic; Rimonabant; Tetrodotoxin; Vagus Nerve

2009
Intracisternal administration of NR2 antagonists attenuates facial formalin-induced nociceptive behavior in rats.
    Journal of orofacial pain, 2010,Spring, Volume: 24, Issue:2

    Topics: Animals; Behavior, Animal; Cisterna Magna; Disease Models, Animal; Excitatory Amino Acid Antagonists; Facial Pain; Formaldehyde; Injections; Injections, Subcutaneous; Kynurenic Acid; Male; Memantine; Motor Activity; Nociceptors; Phenols; Piperazines; Piperidines; Pruritus; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Time Factors; Vibrissae

2010
Peripheral administration of NR2 antagonists attenuates orofacial formalin-induced nociceptive behavior in rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 2011, Jun-01, Volume: 35, Issue:4

    Topics: Animals; Behavior, Animal; Excitatory Amino Acid Antagonists; Facial Pain; Injections; Kynurenic Acid; Male; Memantine; Pain Measurement; Phenols; Piperidines; Postural Balance; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Vibrissae

2011
Novel nootropic drug sunifiram enhances hippocampal synaptic efficacy via glycine-binding site of N-methyl-D-aspartate receptor.
    Hippocampus, 2013, Volume: 23, Issue:10

    Topics: Animals; CA1 Region, Hippocampal; Dose-Response Relationship, Drug; Electrodes, Implanted; Excitatory Amino Acid Antagonists; Glycine; Kynurenic Acid; Long-Term Potentiation; Male; Mice; Mice, Inbred C57BL; Nootropic Agents; Piperazines; Piperidines; Polyamines; Protein Binding; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

2013
Release of CGRP from mouse brainstem slices indicates central inhibitory effect of triptans and kynurenate.
    The journal of headache and pain, 2014, Feb-08, Volume: 15

    Topics: Animals; Brain Stem; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Female; Kynurenic Acid; Male; Mice; Mice, Inbred C57BL; Neural Inhibition; Organ Culture Techniques; Piperidines; Rats, Sprague-Dawley; Tryptamines

2014