Page last updated: 2024-09-02

kt 5823 and zaprinast

kt 5823 has been researched along with zaprinast in 8 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(zaprinast)
Trials
(zaprinast)
Recent Studies (post-2010) (zaprinast)
317059576287

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)zaprinast (IC50)
cGMP-specific 3',5'-cyclic phosphodiesteraseHomo sapiens (human)1.9442
cGMP-specific 3',5'-cyclic phosphodiesteraseCanis lupus familiaris (dog)0.76
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A Bos taurus (cattle)2.6
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1AHomo sapiens (human)3.55
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1BBos taurus (cattle)2.6
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1BHomo sapiens (human)3.55
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1CHomo sapiens (human)3.55
cGMP-specific 3',5'-cyclic phosphodiesteraseBos taurus (cattle)0.4
G-protein coupled receptor 35Homo sapiens (human)0.8294

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (37.50)18.2507
2000's4 (50.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anwyl, R; Rowan, MJ; Wang, Y; Wu, J1
Chik, CL; Hashimoto, K; Ho, AK1
Gong, G; Scholz, PM; Straznicka, M; Weiss, HR; Yan, L1
Johns, RA; Li, D; Shirakami, G; Zhan, X1
Baba, A; Enomoto, R; Lee, E; Matsuda, T; Mori, K; Takuma, K1
Chai, Y; Lin, YF; Mao, X1
Chai, Y; Lin, YF1
Cai, CY; Cai, ZX; Guo, HS; Li, P; Qu, CL; Zhang, SY1

Other Studies

8 other study(ies) available for kt 5823 and zaprinast

ArticleYear
Evidence for involvement of the cGMP-protein kinase G signaling system in the induction of long-term depression, but not long-term potentiation, in the dentate gyrus in vitro.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, May-15, Volume: 18, Issue:10

    Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Alkaloids; Animals; Benzoates; Carbazoles; Cyclic GMP; Dentate Gyrus; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; GTP-Binding Proteins; Guanylate Cyclase; Indoles; Long-Term Potentiation; Neurons; Oxadiazoles; Phosphodiesterase Inhibitors; Protein Kinases; Purinones; Quinoxalines; Rats; Receptors, Metabotropic Glutamate; Signal Transduction

1998
3',5'-cyclic guanosine monophosphate activates mitogen-activated protein kinase in rat pinealocytes.
    Journal of neurochemistry, 1999, Volume: 73, Issue:2

    Topics: Alkaloids; Animals; Atrial Natriuretic Factor; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cells, Cultured; Cyclic GMP; Dibutyryl Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Indoles; Isoquinolines; Male; Naphthalenes; Natriuretic Peptide, C-Type; Neurosecretory Systems; Nitroprusside; Phosphodiesterase Inhibitors; Phosphorylation; Pineal Gland; Protein Kinase C; Purinones; Rats; Rats, Sprague-Dawley; Sulfhydryl Reagents; Sulfonamides; Thionucleotides

1999
Cyclic GMP protein kinase mediates negative metabolic and functional effects of cyclic GMP in control and hypertrophied rabbit cardiac myocytes.
    Journal of cardiovascular pharmacology, 1999, Volume: 34, Issue:2

    Topics: Alkaloids; Animals; Carbazoles; Cardiomegaly; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Indoles; Myocardium; Oxygen Consumption; Purinones; Rabbits

1999
Regulation of ciliary beat frequency by the nitric oxide-cyclic guanosine monophosphate signaling pathway in rat airway epithelial cells.
    American journal of respiratory cell and molecular biology, 2000, Volume: 23, Issue:2

    Topics: Alkaloids; Animals; Arginine; Carbazoles; Cells, Cultured; Cilia; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epithelial Cells; Glutathione; Indoles; Nitric Oxide; Nitric Oxide Donors; Nitroso Compounds; omega-N-Methylarginine; Oxadiazoles; Purinones; Quinoxalines; Rats; S-Nitrosoglutathione; Signal Transduction; Trachea

2000
Ibudilast attenuates astrocyte apoptosis via cyclic GMP signalling pathway in an in vitro reperfusion model.
    British journal of pharmacology, 2001, Volume: 133, Issue:6

    Topics: Alkaloids; Animals; Animals, Newborn; Apoptosis; Astrocytes; Carbazoles; Cell Survival; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Cytochrome c Group; Dipyridamole; DNA; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hydrogen Peroxide; Indoles; Mitochondria; Pentoxifylline; Peptide Hydrolases; Phosphodiesterase Inhibitors; Purinones; Pyridines; Rats; Rats, Wistar; Reperfusion Injury; Signal Transduction; Theophylline; Vinca Alkaloids

2001
Dual regulation of the ATP-sensitive potassium channel by caffeine.
    American journal of physiology. Cell physiology, 2007, Volume: 292, Issue:6

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine Triphosphate; Animals; Caffeine; Carbazoles; Cell Line; Dose-Response Relationship, Drug; Gene Expression Regulation; Humans; Indoles; Insulin; Insulin Secretion; Ion Channel Gating; Islets of Langerhans; Isoquinolines; Muscle, Smooth; Pancreas; Potassium Channels; Protein Isoforms; Purinones; Rats; Sulfonamides

2007
Dual regulation of the ATP-sensitive potassium channel by activation of cGMP-dependent protein kinase.
    Pflugers Archiv : European journal of physiology, 2008, Volume: 456, Issue:5

    Topics: Adenosine Triphosphate; Animals; Carbazoles; Cell Line; Cyclic GMP-Dependent Protein Kinases; Enzyme Inhibitors; Humans; KATP Channels; Neurons; Nitric Oxide; Nitric Oxide Donors; Nitroso Compounds; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Purinones; Recombinant Fusion Proteins; Signal Transduction

2008
Effect of dendroaspis natriuretic peptide (DNP) on L-type calcium channel current and its pathway.
    Regulatory peptides, 2010, Sep-24, Volume: 164, Issue:2-3

    Topics: Aminoquinolines; Animals; Calcium Channels, L-Type; Carbazoles; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Elapid Venoms; Electrophysiology; Enzyme Inhibitors; Guanylate Cyclase; Guinea Pigs; Intercellular Signaling Peptides and Proteins; Myocytes, Smooth Muscle; Peptides; Purinones; Pyloric Antrum; Radioimmunoassay

2010