Page last updated: 2024-09-02

kt 5823 and suramin

kt 5823 has been researched along with suramin in 3 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(suramin)
Trials
(suramin)
Recent Studies (post-2010) (suramin)
3170593,02392431

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)suramin (IC50)
ATP-dependent 6-phosphofructokinaseTrypanosoma brucei brucei3
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)9.76
P2X purinoceptor 2Rattus norvegicus (Norway rat)4
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)1.7
DNA primaseMycobacterium tuberculosis CDC15518.2
RmtAAspergillus nidulans5.9
Reverse transcriptase/RNaseH Human immunodeficiency virus 19.4
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)1.15
NAD-dependent protein deacetylase sirtuin-1Homo sapiens (human)1.5667
Protein arginine N-methyltransferase 1Homo sapiens (human)5.33
NAD-dependent protein deacylase sirtuin-5, mitochondrialHomo sapiens (human)2.5

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
De Godoy, M; Li, F; Rattan, S1
Bianciotti, LG; di Nunzio, A; Hope, SI; Legaz, G; Morgazo, C; Perfume, G; Vatta, MS1
Harada, N; Kubo, N; Shen, J; Takeda-Nakazawa, H; Yamashita, T; Zenner, HP1

Other Studies

3 other study(ies) available for kt 5823 and suramin

ArticleYear
Role of adenylate and guanylate cyclases in beta1-, beta2-, and beta3-adrenoceptor-mediated relaxation of internal anal sphincter smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 308, Issue:3

    Topics: Adenine; Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Carbazoles; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; GTP-Binding Proteins; Guanylate Cyclase; Indoles; Male; Muscle Relaxation; Muscle, Smooth; Oxadiazoles; Procaterol; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Suramin; Xamoterol

2004
Involvement of nitric oxide pathways in short term modulation of tyrosine hydroxylase activity by endothelins 1 and 3 in the rat anterior hypothalamus.
    Biochemical and biophysical research communications, 2005, Sep-02, Volume: 334, Issue:3

    Topics: Animals; Carbazoles; Cyclic GMP; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Endothelin-3; Hypothalamus, Anterior; Indazoles; Indoles; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase Type I; Nitroprusside; Oligopeptides; Oxadiazoles; Piperidines; Quinoxalines; Rats; Suramin; Tyrosine 3-Monooxygenase

2005
Hyposmotic stimulation-induced nitric oxide production in outer hair cells of the guinea pig cochlea.
    Hearing research, 2007, Volume: 230, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium; Carbazoles; Cell Size; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Enzyme Inhibitors; Gadolinium; Guanylate Cyclase; Guinea Pigs; Hair Cells, Auditory, Outer; Hypotonic Solutions; Indoles; Kinetics; Membrane Potentials; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Organ of Corti; Osmotic Pressure; Phorbol Esters; Potassium; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; S-Nitroso-N-Acetylpenicillamine; Signal Transduction; Sodium Chloride; Suramin; TRPV Cation Channels

2007
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