Page last updated: 2024-09-02

kt 5823 and staurosporine

kt 5823 has been researched along with staurosporine in 11 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(staurosporine)
Trials
(staurosporine)
Recent Studies (post-2010) (staurosporine)
3170594160286
3170596,27258976

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)staurosporine (IC50)
Chain A, Glycogen Synthase Kinase-3 BetaHomo sapiens (human)0.015
Chain B, Glycogen Synthase Kinase-3 BetaHomo sapiens (human)0.015
Chain A, Glycogen Synthase Kinase-3 BetaHomo sapiens (human)0.015
Chain A, Tyrosine-protein kinase ZAP-70Homo sapiens (human)0.0558
Chain A, Tyrosine-protein kinase SYKHomo sapiens (human)0.012
Chain A, Proto-oncogene serine/threonine-protein kinase Pim-1Homo sapiens (human)0.01
Chain A, Proto-oncogene serine/threonine-protein kinase Pim-1Homo sapiens (human)0.01
Chain X, Proto-oncogene tyrosine-protein kinase FynHomo sapiens (human)0.0048
Chain A, Serine/threonine-protein kinase TAO2Rattus norvegicus (Norway rat)3
epidermal growth factor receptor isoform a precursorHomo sapiens (human)0.4467
Serine/threonine-protein kinase Sgk1Homo sapiens (human)0.01
Cell division cycle 7-related protein kinaseHomo sapiens (human)0.0549
Serine/threonine-protein kinase PLK4Homo sapiens (human)0.0083
Serine/threonine-protein kinase 25Homo sapiens (human)0.0029
Citron Rho-interacting kinaseHomo sapiens (human)0.749
Dual specificity mitogen-activated protein kinase kinase 7Homo sapiens (human)0.9255
Telomerase reverse transcriptaseHomo sapiens (human)6.9517
Serine/threonine-protein kinase Chk1Homo sapiens (human)0.1772
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)0.5561
Aurora kinase AHomo sapiens (human)0.0087
Cyclin-G-associated kinaseHomo sapiens (human)0.011
Serine/threonine-protein kinase DCLK1Homo sapiens (human)0.267
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)0.1265
Muscle, skeletal receptor tyrosine-protein kinaseHomo sapiens (human)0.1161
Mitogen-activated protein kinase 13Homo sapiens (human)0.4137
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)0.0072
Death-associated protein kinase 3Homo sapiens (human)0.0026
Mitogen-activated protein kinase kinase kinase 7Homo sapiens (human)0.0565
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)0.356
Dual specificity tyrosine-phosphorylation-regulated kinase 3Homo sapiens (human)0.0231
NUAK family SNF1-like kinase 1Homo sapiens (human)0.003
Cyclin-T1Homo sapiens (human)0.0118
Cyclin-T2Homo sapiens (human)0.0038
Tyrosine-protein kinase JAK2Homo sapiens (human)0.0016
Rho-associated protein kinase 2Homo sapiens (human)0.0045
Serine/threonine-protein kinase ULK1Homo sapiens (human)0.0096
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)0.1246
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)0.0011
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)0.0071
Serine/threonine-protein kinase 16Homo sapiens (human)0.2385
Cyclin-KHomo sapiens (human)0.0948
Serine/threonine-protein kinase PAK 3Homo sapiens (human)0.0003
Serine/threonine-protein kinase 17BHomo sapiens (human)0.0258
Serine/threonine-protein kinase 10Homo sapiens (human)0.008
Serine/threonine-protein kinase D3Homo sapiens (human)0.1446
Cyclin-dependent kinase 14Homo sapiens (human)0.1145
G2/mitotic-specific cyclin-B2Homo sapiens (human)0.0107
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)0.2829
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)0.0005
Serine/threonine-protein kinase LATS1Homo sapiens (human)0.013
Serine/threonine-protein kinase PAK 4Homo sapiens (human)0.0132
Serine/threonine-protein kinase Chk2Homo sapiens (human)0.0212
G1/S-specific cyclin-E2Homo sapiens (human)0.011
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.0812
Tyrosine-protein kinase ABL1Homo sapiens (human)0.1233
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)0.0063
Epidermal growth factor receptorHomo sapiens (human)0.083
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)0.1281
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)0.0713
High affinity nerve growth factor receptorHomo sapiens (human)0.2403
Protein kinase C gamma typeHomo sapiens (human)0.1167
Platelet-derived growth factor receptor betaMus musculus (house mouse)0.002
Protein kinase C alpha typeRattus norvegicus (Norway rat)0.2327
Protein kinase C beta typeHomo sapiens (human)0.0684
Prostaglandin G/H synthase 1Ovis aries (sheep)0.056
Insulin receptorHomo sapiens (human)0.0706
Tyrosine-protein kinase LckHomo sapiens (human)0.1784
Tyrosine-protein kinase FynHomo sapiens (human)0.0929
Retinoblastoma-associated protein Homo sapiens (human)0.066
Cyclin-dependent kinase 1Homo sapiens (human)0.0075
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)0.0039
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)0.1269
Tyrosine-protein kinase YesHomo sapiens (human)0.0029
Tyrosine-protein kinase LynHomo sapiens (human)0.0012
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)0.0021
Insulin-like growth factor 1 receptorHomo sapiens (human)0.5534
Hepatocyte growth factor receptorHomo sapiens (human)0.1917
Tyrosine-protein kinase HCKHomo sapiens (human)0.0025
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)0.0004
Protein kinase C delta typeRattus norvegicus (Norway rat)0.274
Protein kinase C epsilon typeRattus norvegicus (Norway rat)0.274
Protein kinase C zeta typeRattus norvegicus (Norway rat)0.274
Platelet-derived growth factor receptor betaHomo sapiens (human)0.3707
Tyrosine-protein kinase FgrHomo sapiens (human)0.0009
Cytochrome P450 2D6Homo sapiens (human)0.0002
Mast/stem cell growth factor receptor KitHomo sapiens (human)0.0412
Breakpoint cluster region proteinHomo sapiens (human)0.0945
Calcium/calmodulin-dependent protein kinase type II subunit alphaRattus norvegicus (Norway rat)0.059
Serine/threonine-protein kinase pim-1Homo sapiens (human)0.0216
Fibroblast growth factor receptor 1Homo sapiens (human)0.0699
Cyclin-dependent kinase 1 Mus musculus (house mouse)0.008
Cyclin-dependent kinase 4Homo sapiens (human)0.0429
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.3642
Acyl-CoA desaturase 1Mus musculus (house mouse)3.4
Insulin receptor-related proteinHomo sapiens (human)0.0113
G2/mitotic-specific cyclin-B1Homo sapiens (human)0.0088
Dipeptidyl peptidase 4Rattus norvegicus (Norway rat)0.003
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)4
Serine/threonine-protein kinase B-rafHomo sapiens (human)0.0107
Insulin receptorMus musculus (house mouse)0.2
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)0.0004
Platelet-derived growth factor receptor alphaHomo sapiens (human)0.0007
Tyrosine-protein kinase FerHomo sapiens (human)0.0008
Protein kinase C alpha typeHomo sapiens (human)0.0655
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)0.0115
Vascular endothelial growth factor receptor 1 Homo sapiens (human)0.0149
Cytochrome P450 11B2, mitochondrialHomo sapiens (human)0.011
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)0.1
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)0.0025
Casein kinase II subunit alpha'Homo sapiens (human)2.0215
Cyclin-A2Homo sapiens (human)0.009
Cannabinoid receptor 1Rattus norvegicus (Norway rat)0.01
Serine/threonine-protein kinase MAKHomo sapiens (human)0.0257
Ephrin type-A receptor 1Homo sapiens (human)0.0947
Fibroblast growth factor receptor 2Homo sapiens (human)0.0504
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)0.0106
Fibroblast growth factor receptor 4Homo sapiens (human)0.17
Fibroblast growth factor receptor 3Homo sapiens (human)0.0554
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)0.0137
Cyclin-OHomo sapiens (human)0.0015
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)0.0148
Ribosomal protein S6 kinase beta-1Homo sapiens (human)0.0007
Tyrosine-protein kinase JAK1Homo sapiens (human)0.004
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.028
G1/S-specific cyclin-D1Homo sapiens (human)0.0355
Protein kinase C eta typeHomo sapiens (human)0.1165
Cyclin-CHomo sapiens (human)0.0105
G1/S-specific cyclin-E1Homo sapiens (human)0.0108
Cyclin-dependent kinase 2Homo sapiens (human)0.0073
Beta-adrenergic receptor kinase 1Homo sapiens (human)1.1595
Platelet-derived growth factor receptor alpha Mus musculus (house mouse)0.002
Mitogen-activated protein kinase 3 Homo sapiens (human)4.6724
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)0.0004
cAMP-dependent protein kinase catalytic subunit alpha Rattus norvegicus (Norway rat)0.055
Mitogen-activated protein kinase 1Homo sapiens (human)2.6853
Ephrin type-A receptor 2Homo sapiens (human)0.1257
Ephrin type-A receptor 3Homo sapiens (human)0.0347
Ephrin type-A receptor 8Homo sapiens (human)0.1061
Ephrin type-B receptor 2Homo sapiens (human)0.1191
Leukocyte tyrosine kinase receptorHomo sapiens (human)0.0173
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)0.0137
G1/S-specific cyclin-D3Homo sapiens (human)0.055
Tyrosine-protein kinase receptor UFOHomo sapiens (human)0.0131
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)0.1848
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)0.4119
G protein-coupled receptor kinase 4Homo sapiens (human)0.0914
Kinesin-1 heavy chainHomo sapiens (human)0.0015
G protein-coupled receptor kinase 5Homo sapiens (human)0.0489
Hexokinase-4Homo sapiens (human)0.0006
Beta-adrenergic receptor kinase 2Homo sapiens (human)0.856
Vascular endothelial growth factor receptor 3Homo sapiens (human)0.0146
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.1791
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)0.026
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)0.0014
Bone morphogenetic protein receptor type-1AHomo sapiens (human)4.288
Activin receptor type-1BHomo sapiens (human)9.118
TGF-beta receptor type-1Homo sapiens (human)2.2823
Serine/threonine-protein kinase receptor R3Homo sapiens (human)0.85
Tyrosine-protein kinase CSKHomo sapiens (human)0.2071
Protein kinase C iota typeHomo sapiens (human)0.1739
Megakaryocyte-associated tyrosine-protein kinaseHomo sapiens (human)0.442
Tyrosine-protein kinase TecHomo sapiens (human)0.0338
Tyrosine-protein kinase TXKHomo sapiens (human)0.0203
Tyrosine-protein kinase ABL2Homo sapiens (human)0.0505
Tyrosine-protein kinase FRKHomo sapiens (human)0.0108
G protein-coupled receptor kinase 6Homo sapiens (human)0.0473
Tyrosine-protein kinase ZAP-70Homo sapiens (human)0.0175
Tyrosine-protein kinase SYKHomo sapiens (human)0.0057
Mitogen-activated protein kinase 8Homo sapiens (human)1.1067
Mitogen-activated protein kinase 9Homo sapiens (human)2.0555
Dual specificity mitogen-activated protein kinase kinase 4Homo sapiens (human)0.863
Phosphorylase b kinase regulatory subunit alpha, liver isoformHomo sapiens (human)0.0005
Phosphorylase b kinase regulatory subunit alpha, skeletal muscle isoformHomo sapiens (human)0.0005
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)0.0099
Casein kinase I isoform alphaHomo sapiens (human)3.412
Casein kinase I isoform deltaHomo sapiens (human)1.4
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)9
MAP kinase-activated protein kinase 2Homo sapiens (human)0.735
Cyclin-dependent kinase 8Homo sapiens (human)0.0105
Casein kinase I isoform epsilonHomo sapiens (human)1.4
Dual specificity protein kinase CLK1Homo sapiens (human)0.0108
Dual specificity protein kinase CLK2Homo sapiens (human)0.6508
Dual specificity protein kinase CLK3Homo sapiens (human)0.92
Glycogen synthase kinase-3 alphaHomo sapiens (human)0.0103
Glycogen synthase kinase-3 betaHomo sapiens (human)0.0435
D(1A) dopamine receptorSus scrofa (pig)0.001
Cyclin-dependent kinase 7Homo sapiens (human)0.2793
Cyclin-dependent kinase 9Homo sapiens (human)0.0474
Tyrosine-protein kinase BlkHomo sapiens (human)0.0011
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)0.0377
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)0.0002
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)0.0046
cAMP-dependent protein kinase catalytic subunit PRKXHomo sapiens (human)0.0014
Cyclin-HHomo sapiens (human)0.2793
CDK-activating kinase assembly factor MAT1Homo sapiens (human)0.1216
Serine/threonine-protein kinase Nek2Homo sapiens (human)1.7683
Serine/threonine-protein kinase Nek4Homo sapiens (human)0.0851
Tyrosine-protein kinase JAK3Homo sapiens (human)0.0084
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)0.0036
Serine/threonine-protein kinase PLK1Homo sapiens (human)0.4397
Death-associated protein kinase 1Homo sapiens (human)0.0101
LIM domain kinase 1Homo sapiens (human)0.0026
LIM domain kinase 2Homo sapiens (human)0.0956
Mitogen-activated protein kinase 12Homo sapiens (human)0.4512
Mitogen-activated protein kinase 10Homo sapiens (human)0.0731
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)1.1354
Ephrin type-B receptor 3Homo sapiens (human)1.2855
Ephrin type-A receptor 5Homo sapiens (human)0.0159
Ephrin type-B receptor 4Homo sapiens (human)0.1869
Ephrin type-B receptor 1Homo sapiens (human)0.0694
Ephrin type-A receptor 4Homo sapiens (human)0.0105
Serine/threonine-protein kinase SIK1Homo sapiens (human)0.0009
Calcium-dependent protein kinase 1Plasmodium falciparum K10.24
Protein kinase C gamma typeRattus norvegicus (Norway rat)0.2168
Casein kinase II subunit betaHomo sapiens (human)3.4
Casein kinase II subunit alphaHomo sapiens (human)3.4723
Protein kinase C beta typeRattus norvegicus (Norway rat)0.2029
SRSF protein kinase 2Homo sapiens (human)0.206
Casein kinase I isoform gamma-2Homo sapiens (human)1.9467
Cyclin-A1Homo sapiens (human)0.0013
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)0.0044
MO15-related protein kinase Pfmrk Plasmodium falciparum (malaria parasite P. falciparum)4
Cyclin-dependent kinase 3Homo sapiens (human)0.0118
Cyclin-dependent kinase 6Homo sapiens (human)0.0395
Cyclin-dependent-like kinase 5 Homo sapiens (human)0.0141
Cyclin-dependent kinase 16Homo sapiens (human)0.0206
Cyclin-dependent kinase 17Homo sapiens (human)0.0135
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.048
Protein kinase C epsilon typeHomo sapiens (human)0.0767
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)0.2314
Angiopoietin-1 receptorHomo sapiens (human)0.0823
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)0.1952
Protein kinase C theta typeHomo sapiens (human)0.1168
Activin receptor type-1Homo sapiens (human)1.1354
Macrophage-stimulating protein receptorHomo sapiens (human)0.2195
Focal adhesion kinase 1Homo sapiens (human)0.078
Protein kinase C zeta typeHomo sapiens (human)0.1722
Protein kinase C delta typeHomo sapiens (human)0.1283
Tyrosine-protein kinase BTKHomo sapiens (human)0.0288
Aldehyde oxidaseHomo sapiens (human)0.0023
Tyrosine-protein kinase receptor TYRO3Homo sapiens (human)0.0177
Cyclin-dependent kinase 18Homo sapiens (human)0.0587
Activated CDC42 kinase 1Homo sapiens (human)0.0299
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)0.9655
Tyrosine-protein kinase ITK/TSKHomo sapiens (human)0.0068
Myotonin-protein kinaseHomo sapiens (human)0.1735
Mitogen-activated protein kinase kinase kinase 12Homo sapiens (human)0.0992
Tyrosine-protein kinase MerHomo sapiens (human)0.0331
Serine/threonine-protein kinase 4Homo sapiens (human)0.0013
Serine/threonine-protein kinase PAK 1Homo sapiens (human)0.0004
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)0.0252
Mitogen-activated protein kinase 7Homo sapiens (human)4.0032
Serine/threonine-protein kinase PAK 2Homo sapiens (human)0.0021
Serine/threonine-protein kinase 3Homo sapiens (human)0.0034
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)0.438
cGMP-dependent protein kinase 2Homo sapiens (human)0.0161
Rho-associated protein kinase 1Homo sapiens (human)0.0038
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)0.0012
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)0.0018
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)0.0026
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)0.0024
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)0.0095
Bone morphogenetic protein receptor type-2Homo sapiens (human)1.94
Protein-tyrosine kinase 6Homo sapiens (human)0.484
cGMP-dependent protein kinase 1 Homo sapiens (human)0.0027
Cyclin-dependent kinase 13Homo sapiens (human)0.057
Calcium/calmodulin-dependent protein kinase type 1Homo sapiens (human)0.0032
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)0.0003
Protein-tyrosine kinase 2-betaHomo sapiens (human)0.0095
Maternal embryonic leucine zipper kinaseHomo sapiens (human)0.0006
Lysine--tRNA ligaseHomo sapiens (human)0.0049
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)0.0141
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrialHomo sapiens (human)0.0005
Serine/threonine-protein kinase D1Homo sapiens (human)0.1448
Serine/threonine-protein kinase 38Homo sapiens (human)0.0037
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)0.183
Ribosomal protein S6 kinase alpha-2Homo sapiens (human)0.0002
Ephrin type-A receptor 7Homo sapiens (human)0.0477
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)0.0004
Dual specificity testis-specific protein kinase 1Homo sapiens (human)0.1995
Myosin light chain kinase, smooth muscleHomo sapiens (human)0.0448
TGF-beta-activated kinase 1 and MAP3K7-binding protein 1Homo sapiens (human)0.037
Mitogen-activated protein kinase 11Homo sapiens (human)1
Serine/threonine-protein kinase STK11Homo sapiens (human)0.0598
Rhodopsin kinase GRK1Homo sapiens (human)0.068
Coiled-coil domain-containing protein 6Homo sapiens (human)0.0022
NT-3 growth factor receptorHomo sapiens (human)0.0002
Serine/threonine-protein kinase N1Homo sapiens (human)0.0025
Serine/threonine-protein kinase N2Homo sapiens (human)0.0055
Mitogen-activated protein kinase 14Homo sapiens (human)0.5052
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)0.1475
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)0.016
BDNF/NT-3 growth factors receptorHomo sapiens (human)0.0004
MAP kinase-activated protein kinase 3Homo sapiens (human)2.775
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformHomo sapiens (human)0.0017
Discoidin domain-containing receptor 2Homo sapiens (human)0.0008
Thioredoxin reductase 1, cytoplasmicHomo sapiens (human)0.0432
Rho-associated protein kinase 2Bos taurus (cattle)0.0417
Myosin light chain kinase 3Homo sapiens (human)0.1585
Serine/threonine-protein kinase SBK1Homo sapiens (human)0.1464
Mitogen-activated protein kinase kinase kinase 19Homo sapiens (human)0.0087
Leucine-rich repeat serine/threonine-protein kinase 2Homo sapiens (human)0.0077
Mitogen-activated protein kinase kinase kinase 21Homo sapiens (human)1.1175
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)0.0032
Sigma non-opioid intracellular receptor 1Cavia porcellus (domestic guinea pig)0.0067
Testis-specific serine/threonine-protein kinase 1Mus musculus (house mouse)0.0003
Dual specificity tyrosine-phosphorylation-regulated kinase 1ARattus norvegicus (Norway rat)0.012
Protein kinase C eta typeRattus norvegicus (Norway rat)0.274
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)0.0005
Calcium/calmodulin-dependent protein kinase type 1BHomo sapiens (human)0.0044
Serine/threonine-protein kinase Nek5Homo sapiens (human)0.0864
Serine/threonine-protein kinase N3Homo sapiens (human)0.0105
Serine/threonine-protein kinase ULK3Homo sapiens (human)0.0027
Kinase suppressor of Ras 2Homo sapiens (human)5.4
Dual serine/threonine and tyrosine protein kinaseHomo sapiens (human)0.0552
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)0.0416
Serine/threonine-protein kinase MARK2Homo sapiens (human)0.0001
Serine/threonine-protein kinase TAO1Homo sapiens (human)0.0008
Serine/threonine-protein kinase Nek8Homo sapiens (human)0.0263
Serine/threonine-protein kinase tousled-like 2Homo sapiens (human)0.0035
Serine/threonine-protein kinase 32CHomo sapiens (human)0.232
Serine/threonine-protein kinase pim-3Homo sapiens (human)0.0001
Myosin light chain kinase family member 4Homo sapiens (human)0.0537
Homeodomain-interacting protein kinase 1Homo sapiens (human)2.639
Calcium/calmodulin-dependent protein kinase type 1DHomo sapiens (human)0.0003
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)0.0001
Kinase suppressor of Ras 1Homo sapiens (human)6.265
Cyclin-dependent kinase-like 3Homo sapiens (human)1.1
MAP kinase-activated protein kinase 5Homo sapiens (human)0.212
Serine/threonine-protein kinase BRSK2Homo sapiens (human)0.0028
Serine/threonine-protein kinase NIM1Homo sapiens (human)0.1102
Serine/threonine-protein kinase ULK2Homo sapiens (human)0.0032
Misshapen-like kinase 1Homo sapiens (human)0.0004
Serine/threonine-protein kinase DCLK2Homo sapiens (human)0.089
Calcium/calmodulin-dependent protein kinase kinase 1Homo sapiens (human)0.0359
Casein kinase I isoform alpha-likeHomo sapiens (human)1.84
Cyclin-YHomo sapiens (human)0.0518
Homeodomain-interacting protein kinase 4Homo sapiens (human)0.226
Myosin-IIIaHomo sapiens (human)0.0425
Serine/threonine-protein kinase Nek11Homo sapiens (human)0.521
Protein odd-skipped-related 1Homo sapiens (human)0.0402
Mitogen-activated protein kinase 15Homo sapiens (human)0.0081
Serine/threonine-protein kinase Nek9Homo sapiens (human)0.101
Serine/threonine-protein kinase BRSK1Homo sapiens (human)0.0007
Serine/threonine-protein kinase haspinHomo sapiens (human)0.0422
Rhodopsin kinase GRK7Homo sapiens (human)0.0053
G2/mitotic-specific cyclin-B3Homo sapiens (human)0.0107
Myosin-IIIbHomo sapiens (human)0.0058
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)0.18
Phosphorylase b kinase regulatory subunit betaHomo sapiens (human)0.0005
Serine/threonine-protein kinase Sgk3Homo sapiens (human)0.073
Aurora kinase BHomo sapiens (human)0.007
Lymphokine-activated killer T-cell-originated protein kinaseHomo sapiens (human)0.0691
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)0.0001
Calcium/calmodulin-dependent protein kinase type 1GHomo sapiens (human)0.0047
Testis-specific serine/threonine-protein kinase 2Homo sapiens (human)0.0038
Testis-specific serine/threonine-protein kinase 3Homo sapiens (human)0.0051
Serine/threonine-protein kinase Nek1Homo sapiens (human)0.0122
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)0.0107
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)0.0246
SRSF protein kinase 1Homo sapiens (human)0.0337
Mitogen-activated protein kinase kinase kinase 14Homo sapiens (human)2.3
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)0.215
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)0.0092
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)0.0531
Testis-specific serine/threonine-protein kinase 6Homo sapiens (human)0.1525
Serine/threonine-protein kinase 33Homo sapiens (human)0.0374
Serine/threonine-protein kinase D2Homo sapiens (human)0.0014
NUAK family SNF1-like kinase 2Homo sapiens (human)0.0018
Serine/threonine-protein kinase SIK2Homo sapiens (human)0.3669
Myosin light chain kinase 2, skeletal/cardiac muscleHomo sapiens (human)0.0147
STE20-like serine/threonine-protein kinase Homo sapiens (human)0.0142
Serine/threonine-protein kinase TAO3Homo sapiens (human)0.0017
Homeodomain-interacting protein kinase 2Homo sapiens (human)0.3655
Tyrosine-protein kinase SrmsHomo sapiens (human)6.5
Homeodomain-interacting protein kinase 3Homo sapiens (human)0.456
Serine/threonine-protein kinase PLK3Homo sapiens (human)0.203
Inactive tyrosine-protein kinase PEAK1Homo sapiens (human)0.0025
Dual specificity protein kinase CLK4Homo sapiens (human)0.0723
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)0.0221
Serine/threonine-protein kinase Sgk2Homo sapiens (human)0.0159
Casein kinase I isoform gamma-1Homo sapiens (human)5.3367
NADPH oxidase 4Homo sapiens (human)0.0708
Serine/threonine-protein kinase PAK 6Homo sapiens (human)0.0327
SNF-related serine/threonine-protein kinaseHomo sapiens (human)0.0059
Serine/threonine-protein kinase LATS2Homo sapiens (human)0.0062
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)0.0122
Serine/threonine-protein kinase 32BHomo sapiens (human)0.0375
Cyclin-dependent kinase 12Homo sapiens (human)0.053
Serine/threonine-protein kinase PLK2Homo sapiens (human)0.546
Serine/threonine-protein kinase MARK1Homo sapiens (human)0.0003
Serine/threonine-protein kinase pim-2Homo sapiens (human)0.0813
Serine/threonine-protein kinase PAK 5Homo sapiens (human)0.0039
Serine/threonine-protein kinase 26Homo sapiens (human)0.0124
Serine/threonine-protein kinase NLKHomo sapiens (human)0.0666
Ribosomal protein S6 kinase beta-2Homo sapiens (human)0.0015
Protein DBF4 homolog AHomo sapiens (human)0.0549
Serine/threonine-protein kinase 17AHomo sapiens (human)0.0386
STE20/SPS1-related proline-alanine-rich protein kinaseHomo sapiens (human)0.0158
Ephrin type-A receptor 6Homo sapiens (human)0.0161
Serine/threonine-protein kinase TBK1Homo sapiens (human)0.003
Death-associated protein kinase 2Homo sapiens (human)0.0064
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)0.0001
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)0.0103
Serine/threonine-protein kinase tousled-like 1Homo sapiens (human)0.0295
Serine/threonine-protein kinase TAO2Homo sapiens (human)0.0076
ALK tyrosine kinase receptorHomo sapiens (human)0.0044
SRSF protein kinase 3Homo sapiens (human)1.77
Serine/threonine-protein kinase ICKHomo sapiens (human)0.0443
Aurora kinase CHomo sapiens (human)0.0022
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)0.0024
Protein kinase C theta typeRattus norvegicus (Norway rat)0.274
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)0.3701
Serine/threonine-protein kinase 38-likeHomo sapiens (human)0.0012
Serine/threonine-protein kinase SIK3Homo sapiens (human)0.1541
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)0.0335
Serine/threonine-protein kinase WNK2Homo sapiens (human)1.455
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)0.0017
5'-AMP-activated protein kinase subunit beta-1Homo sapiens (human)1.1354
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)0.0002
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)0.0027
Serine/threonine-protein kinase 24Homo sapiens (human)0.0065
Casein kinase I isoform gamma-3Homo sapiens (human)2.675
Chain A, Ribosomal protein S6 kinase alpha-1Homo sapiens (human)0.0003
Chain X, Tyrosine-protein kinase LynHomo sapiens (human)0.0013

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (63.64)18.2507
2000's4 (36.36)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Birdsall, NJ; Lazareno, S; Popham, A1
Hayashi, T; Kato, H; Koshino, Y; Kutsumi, Y; Miyabo, S; Nakai, T1
Bradbury, EM; Crissman, HA; Gadbois, DM; Tobey, RA1
Garcia, NH; Garvin, JL1
Ayusawa, D; Fujii, M; Ide, T; Kaul, SC; Mitsui, Y; Ogata, T; Oishi, M; Tahara, H; Wadhwa, R1
Sansom, SC; Stockand, JD1
Blau, N; Leimbacher, W; Scherer-Oppliger, T; Thöny, B1
Knox, FG; Liang, M1
Ardenghi, P; Barros, DM; Izquierdo, I; Izquierdo, LA; Medinam, JH; Mello e Souza, T; Rodrigues, C; Sant'Anna, MK; Vianna, M1
Andreka, P; Bishopric, NH; Evans, WH; Haywood, GA; Martin, PE; Turner, MS; Webster, KA; You, L1
Liu, L; Xu, J1

Other Studies

11 other study(ies) available for kt 5823 and staurosporine

ArticleYear
Allosteric interactions of staurosporine and other indolocarbazoles with N-[methyl-(3)H]scopolamine and acetylcholine at muscarinic receptor subtypes: identification of a second allosteric site.
    Molecular pharmacology, 2000, Volume: 58, Issue:1

    Topics: Acetylcholine; Allosteric Regulation; Allosteric Site; Animals; Carbazoles; CHO Cells; Cricetinae; Enzyme Inhibitors; Indole Alkaloids; Indoles; N-Methylscopolamine; Pyrroles; Radioligand Assay; Receptors, Muscarinic; Staurosporine

2000
Glucocorticoids increase Ca2+ influx through dihydropyridine-sensitive channels linked to activation of protein kinase C in vascular smooth muscle cells.
    Biochemical and biophysical research communications, 1992, Oct-30, Volume: 188, Issue:2

    Topics: Alkaloids; Animals; Aorta; Calcium; Calcium Channels; Carbazoles; Cell Line; Cell Membrane; Cytosol; Dexamethasone; Indoles; Isradipine; Kinetics; Muscle, Smooth, Vascular; Protein Kinase C; Pyrroles; Rats; Staurosporine

1992
Multiple kinase arrest points in the G1 phase of nontransformed mammalian cells are absent in transformed cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1992, Sep-15, Volume: 89, Issue:18

    Topics: Alkaloids; Carbazoles; Cell Cycle; Cell Transformation, Neoplastic; Cells, Cultured; Humans; In Vitro Techniques; Indole Alkaloids; Indoles; Interphase; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Staurosporine

1992
ANF and angiotensin II interact via kinases in the proximal straight tubule.
    The American journal of physiology, 1995, Volume: 268, Issue:4 Pt 2

    Topics: 1-Methyl-3-isobutylxanthine; Absorption; Alkaloids; Angiotensin II; Animals; Atrial Natriuretic Factor; Carbazoles; Cyclic AMP; Drug Interactions; Indoles; Kidney Tubules, Proximal; Male; Phosphotransferases; Rats; Rats, Sprague-Dawley; Staurosporine

1995
Inhibitors of cGMP-dependent protein kinase block senescence induced by inactivation of T antigen in SV40-transformed immortal human fibroblasts.
    Oncogene, 1995, Aug-17, Volume: 11, Issue:4

    Topics: Alkaloids; Antigens, Polyomavirus Transforming; Biomarkers; Carbazoles; Cell Line, Transformed; Cell Nucleus; Cell Transformation, Neoplastic; Cellular Senescence; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP-Dependent Protein Kinases; Cycloheximide; Fibroblasts; Heat-Shock Proteins; HSP70 Heat-Shock Proteins; Humans; Immunohistochemistry; Indoles; Isoquinolines; Mitochondrial Proteins; Myosin-Light-Chain Kinase; Protein Kinase C; Signal Transduction; Simian virus 40; Staurosporine; Sulfonamides

1995
Mechanism of activation by cGMP-dependent protein kinase of large Ca(2+)-activated K+ channels in mesangial cells.
    The American journal of physiology, 1996, Volume: 271, Issue:5 Pt 1

    Topics: Adenosine Triphosphate; Alkaloids; Calcium; Carbazoles; Cells, Cultured; Cyclic GMP-Dependent Protein Kinases; Dibutyryl Cyclic GMP; Enzyme Activation; Enzyme Inhibitors; Glomerular Mesangium; Humans; Indoles; Kinetics; Membrane Potentials; Okadaic Acid; Patch-Clamp Techniques; Potassium Channels; Protein Kinase Inhibitors; Pyrroles; Staurosporine

1996
Serine 19 of human 6-pyruvoyltetrahydropterin synthase is phosphorylated by cGMP protein kinase II.
    The Journal of biological chemistry, 1999, Oct-29, Volume: 274, Issue:44

    Topics: Alkaloids; Amino Acid Metabolism, Inborn Errors; Amino Acid Sequence; Animals; Carbazoles; Consensus Sequence; COS Cells; Cyclic GMP-Dependent Protein Kinase Type II; Cyclic GMP-Dependent Protein Kinases; Fibroblasts; Humans; Indoles; Mice; Mice, Knockout; Molecular Sequence Data; Mutation; Phosphorus-Oxygen Lyases; Phosphorylation; Protein Serine-Threonine Kinases; Recombinant Proteins; Serine; Skin; Staurosporine

1999
Nitric oxide activates PKCalpha and inhibits Na+-K+-ATPase in opossum kidney cells.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Alkaloids; Animals; Arachidonic Acids; Carbazoles; Cell Line; Enzyme Activation; Enzyme Inhibitors; Estrenes; Indoles; Isoenzymes; Kidney; Kidney Tubules, Proximal; Kinetics; Naphthalenes; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Opossums; Protein Kinase C; Protein Kinase C-alpha; Pyrrolidinones; Sodium-Potassium-Exchanging ATPase; Staurosporine; Tetradecanoylphorbol Acetate

1999
Short- and long-term memory are differentially affected by metabolic inhibitors given into hippocampus and entorhinal cortex.
    Neurobiology of learning and memory, 2000, Volume: 73, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Aminoquinolines; Animals; Avoidance Learning; Carbazoles; Entorhinal Cortex; Enzyme Inhibitors; Flavonoids; Guanylate Cyclase; Hippocampus; Indoles; Inhibition, Psychological; Male; Memory; Memory, Short-Term; Phenols; Protein Kinase Inhibitors; Pyrroles; Rats; Rats, Wistar; Sodium Chloride; Staurosporine

2000
Reversible connexin 43 dephosphorylation during hypoxia and reoxygenation is linked to cellular ATP levels.
    Circulation research, 2004, Oct-01, Volume: 95, Issue:7

    Topics: Adenosine Triphosphate; Alkaloids; Aminoimidazole Carboxamide; Animals; Antimycin A; Benzophenanthridines; Brefeldin A; Carbazoles; Cell Hypoxia; Cells, Cultured; Connexin 43; Cycloheximide; Deoxyglucose; Flavonoids; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Myocardial Contraction; Myocytes, Cardiac; Okadaic Acid; Ouabain; Phenanthridines; Phosphorylation; Potassium Cyanide; Protein Processing, Post-Translational; Pyridines; Pyrroles; Rats; Recombinant Fusion Proteins; Ribonucleotides; Staurosporine; Tacrolimus; Tetradecanoylphorbol Acetate

2004
The role of calcium desensitization in vascular hyporeactivity and its regulation after hemorrhagic shock in the rat.
    Shock (Augusta, Ga.), 2005, Volume: 23, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Blood Vessels; Calcium; Carbazoles; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Indoles; Insulin; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Oxazoles; Perfusion; Protein Kinase Inhibitors; Rats; Rats, Wistar; Shock, Hemorrhagic; Staurosporine; Tetradecanoylphorbol Acetate

2005