Page last updated: 2024-09-02

kt 5823 and pyrilamine

kt 5823 has been researched along with pyrilamine in 1 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(pyrilamine)
Trials
(pyrilamine)
Recent Studies (post-2010) (pyrilamine)
3170591,86026116

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)pyrilamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.13
Alpha-2A adrenergic receptorHomo sapiens (human)2.976
Cytochrome P450 2D6Homo sapiens (human)0.3
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.997
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.13
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.0015
Histamine H1 receptorRattus norvegicus (Norway rat)0.0126
Sodium-dependent serotonin transporterHomo sapiens (human)0.047
Histamine H1 receptorHomo sapiens (human)0.0166
5-hydroxytryptamine receptor 2BHomo sapiens (human)2.788
Sodium-dependent dopamine transporter Homo sapiens (human)0.879
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.1
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.558

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fukui, H; Horio, S; Izumi, N; Kawakami, N; Miyoshi, K; Wakayama, Y1

Other Studies

1 other study(ies) available for kt 5823 and pyrilamine

ArticleYear
Histamine H1 receptor down-regulation mediated by M3 muscarinic acetylcholine receptor subtype.
    Journal of pharmacological sciences, 2004, Volume: 95, Issue:4

    Topics: Animals; Atropine; Carbachol; Carbazoles; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Down-Regulation; Histamine H1 Antagonists; Indoles; Inositol Phosphates; Muscarinic Antagonists; Phosphorylation; Protein Kinase C; Pyrilamine; Radioligand Assay; Receptor, Muscarinic M3; Receptors, Histamine H1; Signal Transduction; Time Factors

2004