Page last updated: 2024-09-02

kt 5823 and pd 98059

kt 5823 has been researched along with pd 98059 in 11 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(pd 98059)
Trials
(pd 98059)
Recent Studies (post-2010) (pd 98059)
3170594,93931,001

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)pd 98059 (IC50)
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)2.8
Luciferin 4-monooxygenasePhotinus pyralis (common eastern firefly)6.3
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)2.8
Prostaglandin G/H synthase 1Homo sapiens (human)1
Mitogen-activated protein kinase 1Homo sapiens (human)2.8
Dual specificity mitogen-activated protein kinase kinase 2 Rattus norvegicus (Norway rat)4.2
Dual specificity mitogen-activated protein kinase kinase 1 Rattus norvegicus (Norway rat)4.2
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)2.4

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (18.18)18.2507
2000's9 (81.82)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chik, CL; Hashimoto, K; Ho, AK1
Alexander, JS; Battarbee, H; Gute, D; Krsmanovic, A; Okayama, N; Park, JH1
Ardenghi, P; Barros, DM; Izquierdo, I; Izquierdo, LA; Medinam, JH; Mello e Souza, T; Rodrigues, C; Sant'Anna, MK; Vianna, M1
Chaby, R; Girard, R; Pedron, T1
Alexander, JS; Grisham, MB; Jordan, P; Laroux, FS; Oshima, T; Pavlick, KP; Verma, SK; Williams, L1
Forough, R; Granger, HJ; Meininger, CJ; Steinle, JJ; Wu, G; Wu, MH1
Andreka, P; Bishopric, NH; Evans, WH; Haywood, GA; Martin, PE; Turner, MS; Webster, KA; You, L1
Chakrabarti, MK; Chowdhury, P; Pal, A; Saha, S1
Rabkin, SW; Tsang, MY1
Beyer, C; Etgen, AM; Garcia-Juárez, M; Gómez-Camarillo, MA; Gómora-Arrati, P; González-Flores, O; Lima-Hernández, FJ1
Anand-Srivastava, MB; Arejian, M; Li, Y1

Other Studies

11 other study(ies) available for kt 5823 and pd 98059

ArticleYear
3',5'-cyclic guanosine monophosphate activates mitogen-activated protein kinase in rat pinealocytes.
    Journal of neurochemistry, 1999, Volume: 73, Issue:2

    Topics: Alkaloids; Animals; Atrial Natriuretic Factor; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cells, Cultured; Cyclic GMP; Dibutyryl Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Indoles; Isoquinolines; Male; Naphthalenes; Natriuretic Peptide, C-Type; Neurosecretory Systems; Nitroprusside; Phosphodiesterase Inhibitors; Phosphorylation; Pineal Gland; Protein Kinase C; Purinones; Rats; Rats, Sprague-Dawley; Sulfhydryl Reagents; Sulfonamides; Thionucleotides

1999
Hypoxia/aglycemia increases endothelial permeability: role of second messengers and cytoskeleton.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Alkaloids; beta Catenin; Cadherins; Calcium; Calcium Channel Blockers; Calcium Signaling; Carbazoles; Cell Hypoxia; Cell Membrane Permeability; Cell Survival; Cells, Cultured; Cyclic GMP-Dependent Protein Kinases; Cytoskeletal Proteins; Cytoskeleton; Dermis; Endothelium; Enzyme Inhibitors; Flavonoids; Gallic Acid; Glucose; Humans; Indoles; Intercellular Junctions; Isoenzymes; Membrane Proteins; Microspheres; Mitogen-Activated Protein Kinases; Occludin; Oxygen; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Second Messenger Systems; Thioglycolates; Trans-Activators

1999
Short- and long-term memory are differentially affected by metabolic inhibitors given into hippocampus and entorhinal cortex.
    Neurobiology of learning and memory, 2000, Volume: 73, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Aminoquinolines; Animals; Avoidance Learning; Carbazoles; Entorhinal Cortex; Enzyme Inhibitors; Flavonoids; Guanylate Cyclase; Hippocampus; Indoles; Inhibition, Psychological; Male; Memory; Memory, Short-Term; Phenols; Protein Kinase Inhibitors; Pyrroles; Rats; Rats, Wistar; Sodium Chloride; Staurosporine

2000
Protein phosphorylation pathways involved during lipopolysaccharide-induced expression of CD14 in mouse bone marrow granulocytes.
    FEMS immunology and medical microbiology, 2000, Volume: 28, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Bone Marrow Cells; Carbazoles; Cells, Cultured; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Female; Flavonoids; Flow Cytometry; Granulocytes; Immunoblotting; Indole Alkaloids; Indoles; Lipopolysaccharide Receptors; Lipopolysaccharides; Mice; Mice, Inbred C3H; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Protein-Tyrosine Kinases

2000
Regulation and distribution of MAdCAM-1 in endothelial cells in vitro.
    American journal of physiology. Cell physiology, 2001, Volume: 281, Issue:4

    Topics: Alkaloids; Animals; Benzophenanthridines; Benzopyrans; Carbazoles; Cell Adhesion Molecules; Cell Line, Transformed; Cysteine Proteinase Inhibitors; Endothelium; Enzyme Inhibitors; Flavonoids; Fluorescent Antibody Technique; Gene Expression; Genistein; Imidazoles; Immunoglobulins; In Vitro Techniques; Indoles; Inflammatory Bowel Diseases; Intestinal Mucosa; Isoquinolines; Leupeptins; MAP Kinase Signaling System; Mice; Mucoproteins; NF-kappa B; Phenanthridines; Pyridines; RNA, Messenger; Tumor Necrosis Factor-alpha

2001
Eph B4 receptor signaling mediates endothelial cell migration and proliferation via the phosphatidylinositol 3-kinase pathway.
    The Journal of biological chemistry, 2002, Nov-15, Volume: 277, Issue:46

    Topics: Alkaloids; Azepines; Blotting, Western; Calcium; Carbazoles; Cell Division; Cell Movement; Cells, Cultured; Chromones; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Flavonoids; Humans; Indoles; MAP Kinase Signaling System; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; Microcirculation; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Neovascularization, Pathologic; Nitric Oxide; Nitrites; Phosphatidylinositol 3-Kinases; Phosphorylation; Precipitin Tests; Receptor, EphB4; Signal Transduction; Time Factors

2002
Reversible connexin 43 dephosphorylation during hypoxia and reoxygenation is linked to cellular ATP levels.
    Circulation research, 2004, Oct-01, Volume: 95, Issue:7

    Topics: Adenosine Triphosphate; Alkaloids; Aminoimidazole Carboxamide; Animals; Antimycin A; Benzophenanthridines; Brefeldin A; Carbazoles; Cell Hypoxia; Cells, Cultured; Connexin 43; Cycloheximide; Deoxyglucose; Flavonoids; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Myocardial Contraction; Myocytes, Cardiac; Okadaic Acid; Ouabain; Phenanthridines; Phosphorylation; Potassium Cyanide; Protein Processing, Post-Translational; Pyridines; Pyrroles; Rats; Recombinant Fusion Proteins; Ribonucleotides; Staurosporine; Tacrolimus; Tetradecanoylphorbol Acetate

2004
Downregulation of human colon carcinoma cell (COLO-205) proliferation through PKG-MAP kinase mediated signaling cascade by E. coli heat stable enterotoxin (STa), a potent anti-angiogenic and anti-metastatic molecule.
    Journal of applied toxicology : JAT, 2008, Volume: 28, Issue:4

    Topics: Aminoquinolines; Angiogenesis Inhibitors; Bacterial Toxins; Blotting, Western; Carbazoles; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Cyclic GMP-Dependent Protein Kinases; Enterotoxins; Escherichia coli Proteins; Flavonoids; Guanylate Cyclase; Humans; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Neoplasm Metastasis; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-myc; Time Factors; Vascular Cell Adhesion Molecule-1; Vascular Endothelial Growth Factor A

2008
The action of nitric oxide to enhance cell survival in chick cardiomyocytes is mediated through a cGMP and ERK1/2 pathway while p38 mitogen-activated protein kinase-dependent pathways do not alter cell death.
    Experimental physiology, 2008, Volume: 93, Issue:7

    Topics: Animals; Carbazoles; Cell Death; Cell Survival; Cells, Cultured; Chick Embryo; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Imidazoles; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocytes, Cardiac; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Pyridines; Signal Transduction

2008
Nitric oxide and ERK/MAPK mediation of estrous behavior induced by GnRH, PGE2 and db-cAMP in rats.
    Physiology & behavior, 2009, Mar-23, Volume: 96, Issue:4-5

    Topics: Analysis of Variance; Animals; Carbazoles; Cyclic AMP; Dinoprostone; Enzyme Inhibitors; Estrous Cycle; Extracellular Signal-Regulated MAP Kinases; Female; Flavonoids; Gonadotropin-Releasing Hormone; Guanylate Cyclase; Injections, Intraventricular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Rats; Rats, Sprague-Dawley; Second Messenger Systems; Sexual Behavior, Animal; Signal Transduction; Statistics, Nonparametric

2009
Nitric oxide attenuates the expression of natriuretic peptide receptor C and associated adenylyl cyclase signaling in aortic vascular smooth muscle cells: role of MAPK.
    American journal of physiology. Heart and circulatory physiology, 2009, Volume: 296, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Aorta; Carbazoles; Cells, Cultured; Down-Regulation; Enzyme Inhibitors; Flavonoids; Free Radical Scavengers; GTP-Binding Protein alpha Subunits, Gi-Go; MAP Kinase Signaling System; Metalloporphyrins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Phosphorylation; Protein Kinase Inhibitors; Quinoxalines; Rats; Receptors, Atrial Natriuretic Factor; S-Nitroso-N-Acetylpenicillamine

2009