Page last updated: 2024-09-02

kt 5823 and omega-n-methylarginine

kt 5823 has been researched along with omega-n-methylarginine in 14 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(omega-n-methylarginine)
Trials
(omega-n-methylarginine)
Recent Studies (post-2010) (omega-n-methylarginine)
3170594,411344336

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)omega-n-methylarginine (IC50)
Neutrophil elastaseHomo sapiens (human)0.3
Proteinase-activated receptor 1Homo sapiens (human)0.0018
Nitric oxide synthase, endothelialBos taurus (cattle)7
Nitric oxide synthase, endothelialHomo sapiens (human)2.9489
Nitric oxide synthase, brainHomo sapiens (human)3.3983
Nitric oxide synthase, brain Rattus norvegicus (Norway rat)7.5
Nitric oxide synthase, inducibleMus musculus (house mouse)2.3
Nitric oxide synthase, inducibleHomo sapiens (human)2.9252
Collagenase 3Homo sapiens (human)0.3
Nitric oxide synthase, brainMus musculus (house mouse)4.3

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (28.57)18.2507
2000's10 (71.43)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kanagawa, A; Morita, T; Shimada, Y; Ueki, H1
Granger, HJ; Huang, Q; Wu, HM; Yuan, Y1
Huang, Q; Yuan, Y1
Lew, WY; Yasuda, S1
Chang, YS; Frangos, JA; Lakshminarayanan, S; Tarbell, JM; Yaccino, JA1
Johns, RA; Li, D; Shirakami, G; Zhan, X1
Antonetti, DA; Gardner, TW; Lakshminarayanan, S; Tarbell, JM1
Caldarera, CM; Clô, C; Facchini, A; Fattori, M; Flamigni, F; Giordano, E; Pignatti, C; Stefanelli, C; Tantini, B1
Gardner, TW; Lakshminarayanan, S; Tarbell, JM1
Barlow, RS; Carrier, GO; Catravas, JD; Dimitropoulou, C; El-Mowafy, AM; Han, G; Maunz, M; Snead, C; White, RE; Yu, X; Zhu, S1
Cunha, FQ; Ferreira, SH; Sachs, D1
Díaz-Troya, S; Najib, S; Sánchez-Margalet, V1
Brito, GA; Cunha, FQ; Ferreira, SH; Lotufo, CM; Ribeiro, RA; Sachs, D; Vale, ML1
Azuma, H; Hirata, Y; Imamura, M; Sakurada, M; Shichiri, M1

Other Studies

14 other study(ies) available for kt 5823 and omega-n-methylarginine

ArticleYear
Stimulation of nitric oxide-cyclic GMP pathway by L-arginine increases the release of hepatic lipase from cultured rat hepatocytes.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:10

    Topics: Alkaloids; Animals; Arginine; Carbazoles; Cyclic GMP; Enzyme Inhibitors; Indoles; Lipase; Liver; Methylene Blue; Nitric Oxide; omega-N-Methylarginine; Protein Kinase Inhibitors; Rats

1996
VEGF induces NO-dependent hyperpermeability in coronary venules.
    The American journal of physiology, 1996, Volume: 271, Issue:6 Pt 2

    Topics: Alkaloids; Animals; Capillary Permeability; Carbazoles; Coronary Vessels; Cyclic GMP-Dependent Protein Kinases; Endothelial Growth Factors; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indoles; Lymphokines; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Swine; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Venules

1996
Interaction of PKC and NOS in signal transduction of microvascular hyperpermeability.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Alkaloids; Animals; Calcium; Capillary Permeability; Carbazoles; Coronary Circulation; Cyclic GMP-Dependent Protein Kinases; Cytosol; Enzyme Inhibitors; Histamine; In Vitro Techniques; Indoles; Ionomycin; Kinetics; Microcirculation; Models, Cardiovascular; Nitric Oxide Synthase; omega-N-Methylarginine; Protein Kinase C; Signal Transduction; Swine; Tetradecanoylphorbol Acetate; Venules

1997
Lipopolysaccharide depresses cardiac contractility and beta-adrenergic contractile response by decreasing myofilament response to Ca2+ in cardiac myocytes.
    Circulation research, 1997, Volume: 81, Issue:6

    Topics: Actin Cytoskeleton; Alkaloids; Animals; Calcium; Carbazoles; Indoles; Lipopolysaccharides; Myocardial Contraction; Nitric Oxide; omega-N-Methylarginine; Rabbits; Receptors, Adrenergic, beta

1997
Shear-induced increase in hydraulic conductivity in endothelial cells is mediated by a nitric oxide-dependent mechanism.
    Arteriosclerosis, thrombosis, and vascular biology, 2000, Volume: 20, Issue:1

    Topics: Alkaloids; Aminoquinolines; Animals; Carbazoles; Cattle; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; omega-N-Methylarginine; Penicillamine; Protein Kinase Inhibitors; Protein Kinases; Stress, Mechanical

2000
Regulation of ciliary beat frequency by the nitric oxide-cyclic guanosine monophosphate signaling pathway in rat airway epithelial cells.
    American journal of respiratory cell and molecular biology, 2000, Volume: 23, Issue:2

    Topics: Alkaloids; Animals; Arginine; Carbazoles; Cells, Cultured; Cilia; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epithelial Cells; Glutathione; Indoles; Nitric Oxide; Nitric Oxide Donors; Nitroso Compounds; omega-N-Methylarginine; Oxadiazoles; Purinones; Quinoxalines; Rats; S-Nitrosoglutathione; Signal Transduction; Trachea

2000
Effect of VEGF on retinal microvascular endothelial hydraulic conductivity: the role of NO.
    Investigative ophthalmology & visual science, 2000, Volume: 41, Issue:13

    Topics: Alkaloids; Aminoquinolines; Animals; Biological Transport; Body Water; Carbazoles; Cattle; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Endothelial Growth Factors; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Lymphokines; Nitrates; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitrites; omega-N-Methylarginine; Permeability; Retinal Vessels; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2000
Polyamines, NO and cGMP mediate stimulation of DNA synthesis by tumor necrosis factor and lipopolysaccharide in chick embryo cardiomyocytes.
    Cardiovascular research, 2001, Feb-01, Volume: 49, Issue:2

    Topics: Alkaloids; Aminoquinolines; Animals; Carbazoles; Cells, Cultured; Chick Embryo; Cyclic GMP; DNA; Eflornithine; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Lipopolysaccharides; Methylene Blue; Myocardium; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Ornithine Decarboxylase; Ornithine Decarboxylase Inhibitors; Polyamines; Protein Kinase Inhibitors; Stimulation, Chemical; Tumor Necrosis Factor-alpha

2001
Effect of shear stress on the hydraulic conductivity of cultured bovine retinal microvascular endothelial cell monolayers.
    Current eye research, 2000, Volume: 21, Issue:6

    Topics: Alkaloids; Aminoquinolines; Animals; Biological Transport; Blood-Retinal Barrier; Body Water; Carbazoles; Cattle; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Nitric Oxide; omega-N-Methylarginine; Retinal Vessels; Stress, Mechanical; Water

2000
Endothelium-independent effect of estrogen on Ca(2+)-activated K(+) channels in human coronary artery smooth muscle cells.
    Cardiovascular research, 2002, Feb-15, Volume: 53, Issue:3

    Topics: Alkaloids; Analysis of Variance; Carbazoles; Coronary Vessels; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Estradiol; Humans; Indoles; Microscopy, Fluorescence; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Patch-Clamp Techniques; Peptides; Potassium Channels, Calcium-Activated; Potassium Channels, Voltage-Gated

2002
Peripheral analgesic blockade of hypernociception: activation of arginine/NO/cGMP/protein kinase G/ATP-sensitive K+ channel pathway.
    Proceedings of the National Academy of Sciences of the United States of America, 2004, Mar-09, Volume: 101, Issue:10

    Topics: Adenosine Triphosphate; Analgesics; Animals; Arginine; Carbazoles; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dinoprostone; Indoles; Male; Nitric Oxide; Nociceptors; omega-N-Methylarginine; Oxadiazoles; Potassium Channels; Quinoxalines; Rats; Rats, Wistar; Signal Transduction

2004
eNOS, nNOS, cGMP and protein kinase G mediate the inhibitory effect of pancreastatin, a chromogranin A-derived peptide, on growth and proliferation of hepatoma cells.
    Regulatory peptides, 2005, Feb-15, Volume: 125, Issue:1-3

    Topics: Aminoquinolines; Animals; Arginine; Calcium; Carbazoles; Carcinoma, Hepatocellular; Cell Enlargement; Cell Proliferation; Chromogranin A; Chromogranins; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; DNA; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Isoenzymes; Leucine; Liver; MAP Kinase Signaling System; Nerve Tissue Proteins; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type III; omega-N-Methylarginine; Ornithine; Pancreatic Hormones; Peptides; Phospholipase C beta; Protein Isoforms; Rats; Receptors, Atrial Natriuretic Factor; Spermidine; Thymidine; Time Factors; Type C Phospholipases

2005
Peripheral antinociceptive effect of pertussis toxin: activation of the arginine/NO/cGMP/PKG/ ATP-sensitive K channel pathway.
    The European journal of neuroscience, 2006, Volume: 24, Issue:4

    Topics: Adenosine Triphosphate; Analgesia; Analgesics; Animals; Arginine; Bucladesine; Carbazoles; Cells, Cultured; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dinoprostone; Enzyme Inhibitors; Ganglia, Spinal; Glyburide; Indoles; KATP Channels; Male; Neurons; Nitric Oxide; omega-N-Methylarginine; Oxadiazoles; Pain; Pain Measurement; Pertussis Toxin; Potassium Channels, Inwardly Rectifying; Quinoxalines; Rats; Rats, Wistar; Signal Transduction; Tolbutamide

2006
Nitric oxide upregulates dimethylarginine dimethylaminohydrolase-2 via cyclic GMP induction in endothelial cells.
    Hypertension (Dallas, Tex. : 1979), 2008, Volume: 52, Issue:5

    Topics: Amidohydrolases; Animals; Arginine; Carbazoles; Cells, Cultured; Cyclic GMP; Endothelium, Vascular; Male; Natriuretic Peptide, C-Type; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Nitro Compounds; omega-N-Methylarginine; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; RNA, Messenger; S-Nitroso-N-Acetylpenicillamine; Up-Regulation

2008