Page last updated: 2024-09-02

kt 5823 and isoproterenol

kt 5823 has been researched along with isoproterenol in 6 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(isoproterenol)
Trials
(isoproterenol)
Recent Studies (post-2010) (isoproterenol)
31705930,7808032,640

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)isoproterenol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.246
Beta-1 adrenergic receptorHomo sapiens (human)0.333
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)1.77
Beta-1 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-3 adrenergic receptorRattus norvegicus (Norway rat)0.2125
Beta-2 adrenergic receptorCanis lupus familiaris (dog)0.6667

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's2 (33.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dollinger, SJ; Wahler, GM1
Makhlouf, GM; Murthy, KS1
Chik, CL; Ho, AK; Karpinski, E; Li, B1
Joyner, RW; Kumar, R; Wagner, MB; Wang, Y1
Keung, W; Man, RY; Vanhoutte, PM1
Chen, YX; Fleischmann, B; Hescheler, J; Ji, G; Miao, L; Wang, M; Yin, WX; Yuan, Q1

Other Studies

6 other study(ies) available for kt 5823 and isoproterenol

ArticleYear
Nitric oxide donor SIN-1 inhibits mammalian cardiac calcium current through cGMP-dependent protein kinase.
    The American journal of physiology, 1995, Volume: 268, Issue:1 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Alkaloids; Aminoquinolines; Animals; Calcium; Carbazoles; Cyclic GMP-Dependent Protein Kinases; Electric Conductivity; Guanylate Cyclase; Guinea Pigs; Heart; Indoles; Isoproterenol; Molsidomine; Myocardium; Nitric Oxide; Protein Kinase Inhibitors

1995
Differential regulation of phospholipase A2 (PLA2)-dependent Ca2+ signaling in smooth muscle by cAMP- and cGMP-dependent protein kinases. Inhibitory phosphorylation of PLA2 by cyclic nucleotide-dependent protein kinases.
    The Journal of biological chemistry, 1998, Dec-18, Volume: 273, Issue:51

    Topics: Alkaloids; Animals; Arachidonic Acid; Calcium; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; In Vitro Techniques; Indoles; Intestines; Isoproterenol; Isoquinolines; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Nitroprusside; Phospholipases A; Phospholipases A2; Phosphorylation; Rabbits; Signal Transduction; Sulfonamides; Thionucleotides; Vasoactive Intestinal Peptide

1998
Regulation of the L-type Ca2+ channel current in rat pinealocytes: role of basal phosphorylation.
    Journal of neurochemistry, 1999, Volume: 72, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenergic beta-Agonists; Alkaloids; Animals; Antifungal Agents; Calcium Channels; Calcium Channels, L-Type; Carbazoles; Cyclic AMP; Cyclic GMP; Enzyme Inhibitors; Indoles; Isoproterenol; Isoquinolines; Male; Marine Toxins; Membrane Potentials; Nerve Tissue Proteins; Norepinephrine; Okadaic Acid; Oxazoles; Patch-Clamp Techniques; Phosphoric Monoester Hydrolases; Phosphorylation; Pineal Gland; Protein Kinase C; Pyrans; Rats; Rats, Sprague-Dawley; Spiro Compounds; Sulfonamides; Sympathomimetics

1999
cGMP-dependent protein kinase mediates stimulation of L-type calcium current by cGMP in rabbit atrial cells.
    Cardiovascular research, 2000, Volume: 48, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Alkaloids; Animals; Blotting, Western; Calcium Channels, L-Type; Carbazoles; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Enzyme Inhibitors; Heart Atria; Indoles; Isoproterenol; Myocardium; Nitric Oxide Donors; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Rabbits; Stimulation, Chemical; Time Factors

2000
Acute impairment of contractile responses by 17beta-estradiol is cAMP and protein kinase G dependent in vascular smooth muscle cells of the porcine coronary arteries.
    British journal of pharmacology, 2005, Volume: 144, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Adenylyl Cyclase Inhibitors; Animals; Carbazoles; Coronary Vessels; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Drug Interactions; Estradiol; Indoles; Isometric Contraction; Isoproterenol; Muscle, Smooth, Vascular; Swine; Thionucleotides; Time Factors

2005
Atrial natriuretic peptide regulates Ca channel in early developmental cardiomyocytes.
    PloS one, 2010, Jan-22, Volume: 5, Issue:1

    Topics: Action Potentials; Adrenergic beta-Antagonists; Animals; Atrial Natriuretic Factor; Base Sequence; Calcium Channels, L-Type; Carbazoles; Cells, Cultured; Colforsin; DNA Primers; Embryonic Stem Cells; Enzyme Inhibitors; Fluorescent Antibody Technique; Heart; Isoproterenol; Mice; Myocardium; NG-Nitroarginine Methyl Ester; Reverse Transcriptase Polymerase Chain Reaction

2010