Page last updated: 2024-09-02

kt 5823 and cocaine

kt 5823 has been researched along with cocaine in 2 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
31705932,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aunis, D; Jouvert, P; Langley, K; Lazaris, A; Revel, MO; Zwiller, J1
Cho, HW; Choe, ES; Kim, J; Lee, DK; Oh, JH; Ryu, IS; Seo, SY; Shim, YB; Yang, JH1

Other Studies

2 other study(ies) available for kt 5823 and cocaine

ArticleYear
Activation of the cGMP pathway in dopaminergic structures reduces cocaine-induced EGR-1 expression and locomotor activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Nov-24, Volume: 24, Issue:47

    Topics: Animals; Brain; Carbazoles; Central Nervous System Stimulants; Cocaine; Cyclic GMP; Cyclic GMP-Dependent Protein Kinase Type I; Cyclic GMP-Dependent Protein Kinases; DNA-Binding Proteins; Dopamine; Early Growth Response Protein 1; Enzyme Activation; Immediate-Early Proteins; Indoles; Injections, Intraventricular; Male; Motor Activity; Natriuretic Peptide, C-Type; Nerve Tissue Proteins; Rats; Rats, Wistar; RNA, Messenger; Signal Transduction; Synaptosomes; Transcription Factors

2004
Dopamine D4 receptors linked to protein kinase G are required for changes in dopamine release followed by locomotor activity after repeated cocaine administration.
    Experimental brain research, 2015, Volume: 233, Issue:5

    Topics: Analysis of Variance; Animals; Benzamides; Carbazoles; Cocaine; Cyclic GMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Male; Motor Activity; Nitric Oxide Synthase Type I; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D4; RNA, Messenger; Tyrosine 3-Monooxygenase

2015