Page last updated: 2024-09-02

kt 5823 and carbachol

kt 5823 has been researched along with carbachol in 4 studies

Compound Research Comparison

Studies
(kt 5823)
Trials
(kt 5823)
Recent Studies (post-2010)
(kt 5823)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
31705913,91881968

Protein Interaction Comparison

ProteinTaxonomykt 5823 (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ding, JM; Faiman, LE; Gillette, MU; Liu, C1
Herring, N; Paterson, DJ1
Iida, H; Inoue, N; Ishida, H; Ishikawa, Y; Yuan, Z1
Fukui, H; Horio, S; Izumi, N; Kawakami, N; Miyoshi, K; Wakayama, Y1

Other Studies

4 other study(ies) available for kt 5823 and carbachol

ArticleYear
Coupling of muscarinic cholinergic receptors and cGMP in nocturnal regulation of the suprachiasmatic circadian clock.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jan-15, Volume: 17, Issue:2

    Topics: Acetylcholine; Afferent Pathways; Alkaloids; Aminoquinolines; Animals; Atropine; Carbachol; Carbazoles; Cholinergic Agents; Cholinergic Fibers; Circadian Rhythm; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Enzyme Inhibitors; Guanylate Cyclase; Indoles; Muscarinic Antagonists; Nerve Tissue Proteins; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Signal Transduction; Suprachiasmatic Nucleus; Time Factors

1997
Nitric oxide-cGMP pathway facilitates acetylcholine release and bradycardia during vagal nerve stimulation in the guinea-pig in vitro.
    The Journal of physiology, 2001, Sep-01, Volume: 535, Issue:Pt 2

    Topics: Acetylcholine; Alkaloids; Animals; Bradycardia; Calcium Channel Blockers; Calcium Channels; Carbachol; Carbazoles; Cardiotonic Agents; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Electric Stimulation; Enzyme Inhibitors; Female; Guanylate Cyclase; Guinea Pigs; Heart Rate; In Vitro Techniques; Indoles; Isoquinolines; Milrinone; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; omega-Conotoxin GVIA; Oxadiazoles; Phosphorylation; Presynaptic Terminals; Quinoxalines; Sinoatrial Node; Sulfonamides; Synaptic Transmission; Tritium; Vagus Nerve

2001
Effect of SNI-2011 on amylase secretion from parotid tissue in rats and in neuronal nitric oxide synthase knockout mice.
    European journal of pharmacology, 2003, Mar-19, Volume: 464, Issue:2-3

    Topics: Alkaloids; Amylases; Animals; Azepines; Benzoates; Benzylamines; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Carbazoles; Chelating Agents; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Gallic Acid; Genotype; Guanylate Cyclase; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Mice, Knockout; Molsidomine; Muscarinic Agonists; Myosin-Light-Chain Kinase; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxadiazoles; Parotid Gland; Penicillamine; Phosphodiesterase Inhibitors; Pilocarpine; Protein Kinase Inhibitors; Pyrroles; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Wistar; Sulfonamides; Thiophenes; Type C Phospholipases

2003
Histamine H1 receptor down-regulation mediated by M3 muscarinic acetylcholine receptor subtype.
    Journal of pharmacological sciences, 2004, Volume: 95, Issue:4

    Topics: Animals; Atropine; Carbachol; Carbazoles; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Down-Regulation; Histamine H1 Antagonists; Indoles; Inositol Phosphates; Muscarinic Antagonists; Phosphorylation; Protein Kinase C; Pyrilamine; Radioligand Assay; Receptor, Muscarinic M3; Receptors, Histamine H1; Signal Transduction; Time Factors

2004