ksg 504 has been researched along with sincalide in 6 studies
| Studies (ksg 504) | Trials (ksg 504) | Recent Studies (post-2010) (ksg 504) | Studies (sincalide) | Trials (sincalide) | Recent Studies (post-2010) (sincalide) |
|---|---|---|---|---|---|
| 13 | 0 | 0 | 4,015 | 72 | 533 |
| Protein | Taxonomy | ksg 504 (IC50) | sincalide (IC50) |
|---|---|---|---|
| Cholecystokinin receptor type A | Rattus norvegicus (Norway rat) | 0.0006 | |
| Cholecystokinin receptor type A | Homo sapiens (human) | 0.0006 | |
| Gastrin/cholecystokinin type B receptor | Homo sapiens (human) | 0.001 | |
| Gastrin/cholecystokinin type B receptor | Mus musculus (house mouse) | 0.0008 | |
| Cholecystokinin receptor type A | Cavia porcellus (domestic guinea pig) | 0.0004 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 6 (100.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Akahane, M; Iizuka, K; Kitazawa, M; Kobayashi, M; Kurashina, Y; Yamazaki, Y | 1 |
| Kihara, Y; Otsuki, M | 1 |
| Ajisawa, Y; Akahane, M; Takeda, H; Tsubaki, A; Yamazaki, Y | 1 |
| Ajisawa, Y; Akahane, M; Kobayashi, M; Shinagawa, K; Sugiura, M; Yamazaki, Y | 1 |
| Ajisawa, Y; Akahane, M; Kobayashi, M; Shinagawa, K; Takeda, H; Yamazaki, Y | 1 |
| Ajisawa, Y; Akahane, M; Kobayashi, M; Takeda, H; Yamazaki, Y | 1 |
6 other study(ies) available for ksg 504 and sincalide
| Article | Year |
|---|---|
Pharmacological profile of KSG-504, a new cholecystokinin-A-receptor antagonist.
Topics: Amylases; Animals; Dogs; Female; Gallbladder; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Naphthalenes; Pancreas; Pentanoic Acids; Rabbits; Radioligand Assay; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Species Specificity | 1993 |
Different inhibitory effects of the newly developed CCK receptor antagonists FK480 and KSG-504 on pancreatic exocrine and endocrine secretion in the isolated perfused rat pancreas.
Topics: Animals; Benzodiazepinones; In Vitro Techniques; Indoles; Insulin; Insulin Secretion; Male; Naphthalenes; Pancreas; Pentanoic Acids; Perfusion; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1995 |
[Behavioral studies of KSG-504, a new CCK-A receptor antagonist].
Topics: Animals; Behavior, Animal; Dogs; Drug Synergism; Female; Male; Mice; Mice, Inbred ICR; Motor Activity; Naphthalenes; Pentanoic Acids; Rabbits; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Thiopental | 1996 |
[Effects of KSG-504, a new CCK-A receptor antagonist, on gallbladder and gastrointestinal functions].
Topics: Animals; Dose-Response Relationship, Drug; Duodenum; Gallbladder; Gallbladder Emptying; Gastric Acid; Gastric Emptying; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Naphthalenes; Pentanoic Acids; Rabbits; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide | 1996 |
Cholecystokinin-A specific antagonism of KSG-504 to cholecystokinin receptor binding and pancreatic secretion in mammals.
Topics: Amylases; Animals; Binding, Competitive; Dose-Response Relationship, Drug; Hormone Antagonists; Male; Naphthalenes; Pancreas; Pentanoic Acids; Radioligand Assay; Rats; Rats, Wistar; Sincalide | 1995 |
Effects of KSG-504, a new cholecystokinin-A-receptor antagonist, on pancreatic exocrine and endocrine secretions in rats.
Topics: Animals; Dose-Response Relationship, Drug; Hormone Antagonists; Male; Naphthalenes; Pancreas; Pentanoic Acids; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide | 1996 |