Page last updated: 2024-09-03

kf 4317 and cocaine

kf 4317 has been researched along with cocaine in 1 studies

Compound Research Comparison

Studies
(kf 4317)
Trials
(kf 4317)
Recent Studies (post-2010)
(kf 4317)
Studies
(cocaine)
Trials
(cocaine)
Recent Studies (post-2010) (cocaine)
50032,4611,0969,400

Protein Interaction Comparison

ProteinTaxonomykf 4317 (IC50)cocaine (IC50)
Amyloid-beta precursor proteinHomo sapiens (human)0.338
Fatty acid-binding protein, heartHomo sapiens (human)0.367
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0855
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0855
DRattus norvegicus (Norway rat)5.7544
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)5.7544
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)5.7544
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.2861
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.4321
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0855
Sodium-dependent serotonin transporterHomo sapiens (human)0.5442
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.8885
Sodium-dependent dopamine transporter Homo sapiens (human)0.3796
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5.541
Sodium-dependent dopamine transporterMus musculus (house mouse)0.2
Sigma non-opioid intracellular receptor 1Homo sapiens (human)1.05
TransporterRattus norvegicus (Norway rat)3.2277

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19901 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Doggrell, SA; Hughes, EW1

Other Studies

1 other study(ies) available for kf 4317 and cocaine

ArticleYear
The effects of KF-4317, a novel combined alpha- and beta 1-adrenoreceptor antagonist, on the rat isolated right ventricle and aorta.
    Journal of autonomic pharmacology, 1986, Volume: 6, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Aorta; Benzeneacetamides; Cocaine; Drug Interactions; Electric Stimulation; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Phenylephrine; Propanolamines; Rats; Rats, Inbred Strains; Serotonin Antagonists; Tritium

1986