Page last updated: 2024-09-03

kf 17837s and n(6)-cyclohexyladenosine

kf 17837s has been researched along with n(6)-cyclohexyladenosine in 6 studies

Compound Research Comparison

Studies
(kf 17837s)
Trials
(kf 17837s)
Recent Studies (post-2010)
(kf 17837s)
Studies
(n(6)-cyclohexyladenosine)
Trials
(n(6)-cyclohexyladenosine)
Recent Studies (post-2010) (n(6)-cyclohexyladenosine)
3900555033

Protein Interaction Comparison

ProteinTaxonomykf 17837s (IC50)n(6)-cyclohexyladenosine (IC50)
Adenosine receptor A1Rattus norvegicus (Norway rat)0.0024
Adenosine receptor A3Rattus norvegicus (Norway rat)0.0024
Adenosine receptor A2bRattus norvegicus (Norway rat)0.588
Adenosine receptor A2aRattus norvegicus (Norway rat)0.588
Adenosine receptor A1Gallus gallus (chicken)0.0025

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arslan, G; Dionisotti, S; Fredholm, BB; Kull, B; Ongini, E; Zocchi, C1
Hayaishi, O; Matsumura, H; Satoh, S; Suzuki, F1
Constantino, MD; Cunha, RA; Fredholm, BB; Johansson, B; Sebastião, AM1
Karasawa, A; Nagashima, K1
Frobenius, W; Geis, U; Hipp, J; Müller, CE; Pawłowski, M; Sandoval-Ramírez, J; Schobert, U; Suzuki, F1
Kondo, Y; Morishima, T; Tsuge, M; Wada, T; Yashiro, M; Yasui, K1

Other Studies

6 other study(ies) available for kf 17837s and n(6)-cyclohexyladenosine

ArticleYear
Characterization of human A2A adenosine receptors with the antagonist radioligand [3H]-SCH 58261.
    British journal of pharmacology, 1997, Volume: 121, Issue:3

    Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Cyclic AMP; Humans; Purinergic P1 Receptor Antagonists; Pyrimidines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Species Specificity; Transfection; Triazoles

1997
Promotion of sleep mediated by the A2a-adenosine receptor and possible involvement of this receptor in the sleep induced by prostaglandin D2 in rats.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, Jun-11, Volume: 93, Issue:12

    Topics: Adenosine; Animals; Male; Phenethylamines; Prosencephalon; Prostaglandin D2; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Sleep; Xanthines

1996
Evidence for high-affinity binding sites for the adenosine A2A receptor agonist [3H] CGS 21680 in the rat hippocampus and cerebral cortex that are different from striatal A2A receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:3

    Topics: 2-Chloroadenosine; Adenosine; Animals; Binding, Competitive; Cerebral Cortex; Corpus Striatum; Dose-Response Relationship, Drug; Hippocampus; Male; Phenethylamines; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Xanthines

1996
Modulation of erythropoietin production by selective adenosine agonists and antagonists in normal and anemic rats.
    Life sciences, 1996, Volume: 59, Issue:9

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Analysis of Variance; Anemia; Animals; Erythropoietin; Hematocrit; Hypoxia; Kinetics; Male; Nephrectomy; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Time Factors; Xanthines

1996
Synthesis and structure-activity relationships of 3,7-dimethyl-1-propargylxanthine derivatives, A2A-selective adenosine receptor antagonists.
    Journal of medicinal chemistry, 1997, Dec-19, Volume: 40, Issue:26

    Topics: Adenosine; Animals; Binding, Competitive; Brain; Caffeine; Molecular Structure; Phenethylamines; Protein Binding; Purinergic P1 Receptor Antagonists; Rats; Receptors, Purinergic P1; Structure-Activity Relationship; Theobromine; Xanthines

1997
Theophylline inhibits the differentiation of human monocyte into dendritic cell potentially via adenosine receptor antagonism.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2009, Volume: 39, Issue:12

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine Deaminase; Adenosine-5'-(N-ethylcarboxamide); Adult; Apoptosis; Caspase 3; CD11c Antigen; Cell Differentiation; Dendritic Cells; Granulocyte-Macrophage Colony-Stimulating Factor; HLA-DR Antigens; Humans; Interleukin-4; Male; Monocytes; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A1; Receptors, Purinergic P1; Recombinant Proteins; RNA, Small Interfering; Rolipram; Theophylline; Xanthines

2009