ketoprofen has been researched along with piroxicam in 86 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (15.12) | 18.7374 |
1990's | 22 (25.58) | 18.2507 |
2000's | 25 (29.07) | 29.6817 |
2010's | 23 (26.74) | 24.3611 |
2020's | 3 (3.49) | 2.80 |
Authors | Studies |
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Andricopulo, AD; Moda, TL; Montanari, CA | 1 |
Apiwattanakul, N; Chairoungdua, A; Endou, H; Kanai, Y; Nakajima, N; Sekine, T; Sophasan, S | 1 |
Cihlar, T; Ho, ES; Mulato, AS | 1 |
Faller, B; Wohnsland, F | 1 |
Cha, SH; Endou, H; Hosoyamada, M; Khamdang, S; Kimura, H; Narikawa, S; Sekine, T; Takeda, M | 1 |
Beroza, P; Cai, D; Damodaran, K; Gomez, RF; Hsu, N; Keck, JG; Laborde, E; Lum, RT; Macke, TJ; Martin, G; Schow, SR; Simon, RJ; Villar, HO; Wick, MM | 1 |
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL | 1 |
Carrupt, PA; Martel, S; Ottaviani, G | 2 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Akamatsu, M; Fujikawa, M; Nakao, K; Shimizu, R | 1 |
Baert, B; Beetens, J; Bodé, S; De Spiegeleer, B; Deconinck, E; Lambert, J; Slegers, G; Slodicka, M; Stoppie, P; Van Gele, M; Vander Heyden, Y | 1 |
Artursson, P; Bergström, CA; Draheim, R; Holmén, AG; Wassvik, CM | 1 |
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W | 1 |
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S | 1 |
Conradi, R; Lee, PH; Shanmugasundaram, V | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Campillo, NE; Guerra, A; Páez, JA | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Avdeef, A; Tam, KY | 1 |
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ | 1 |
Gozalbes, R; Pineda-Lucena, A | 1 |
Ekins, S; Williams, AJ; Xu, JJ | 1 |
Buttar, D; Colclough, N; Gerhardt, S; MacFaul, PA; Maskos, K; Phillips, SD; Plowright, A; Steinbacher, S; Steuber, H; Tam, K; Whittamore, P | 1 |
Akamatsu, M | 1 |
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K | 1 |
Barber, S; Dew, TP; Farrell, TL; Poquet, L; Williamson, G | 1 |
Kumar, M; Sinha, VR; Thareja, S | 1 |
Chen, L; Fei, J; Mei, Y; Ren, S; Yan, SF; Zeng, J; Zhang, JZ | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL | 1 |
de Pouvourville, G | 1 |
Cerretani, D; Fiaschi, AI; Giorgi, G; Micheli, L | 2 |
Aligia, C; Kelloff, G; Kulkarni, N; Reddy, BS; Tokumo, K | 1 |
Louisot, P; Mathieu, P; Richard, M; Vignon, E | 1 |
Collier, S; Ghosh, P | 1 |
Abdel-Moneam, NM; Mostafa, MH; Sheweita, SA | 1 |
Battellino, LJ; Dorronsoro de Cattoni, ST; Ragagnin, C | 1 |
Ejstrup, L; Knudsen, JV; Petersen, L | 1 |
Paulus, HE; Schlegel, SI | 1 |
Simon, L | 1 |
Sallmann, AR | 2 |
Tariq, M | 1 |
Doury, P; Roux, H | 1 |
Bassi, GP; Borghi, C; Camarri, E; Cocco, F; Francucci, BM; Giannini, R; Giordano, N; Marcolongo, R; Mordini, M; Neri, D | 1 |
Burnham, WR; O'Brien, JD | 1 |
Ward, JR | 1 |
Evangelista, S; Giolitti, A; Grimaldi, G; Maggi, CA; Meli, A; Santicioli, P | 1 |
Court, H; Volans, GN | 1 |
Hatano, M; Hoya, I; Ishihara, M; Miura, K; Miyata, K; Okusawa, S; Yamada, T; Yoshida, A | 1 |
Dreiser, RL; Riebenfeld, D | 1 |
Chanaud, B; Chancerelle, Y; De Sousa, M; Florentin, I; Giroud, JP; Kergonou, JF; Masson, I; Mathieu, J; Strazlko, S | 1 |
Bressolle, F; Combe, B; Edno, L; Galtier, M | 1 |
Dainaka, J; Hashii, H; Inoue, K; Kimura, K; Motonaga, A; Nishimura, T; Ueda, F; Yamate, K | 1 |
Aguejouf, O; Doutremepuich, C; Doutremepuich, F; Imbault, P; Oualane, FA | 1 |
Franchimont, P; Reginster, JY | 1 |
Bradley, JD; Brater, DC; Greene, PK; Tracy, TS; Worster, T | 1 |
Baeyens, W; Donato, MG; Sandra, P; van den Bossche, W | 1 |
Dobson, A; Henry, D; Turner, C | 1 |
Becker, L; Eberlein-König, B; Przybilla, B | 1 |
Fox, SM; Johnston, SA | 1 |
Carmody, JJ; Day, RO; Sheather-Reid, RB; Vial, JH; Walker, JS | 1 |
Catalioto, RM; Criscuoli, M; Cucchi, P; Lecci, A; Maggi, CA; Meini, S | 1 |
Amidon, GL; Hilgendorf, C; Langguth, P; Lipka, E; Regårdh, CG; Spahn-Langguth, H | 1 |
Pontes, RM; Prado, WA | 1 |
Cowan, A; Raffa, RB; Tallarida, RJ | 1 |
Djordjevic, J; Michniak, B; Uhrich, KE | 1 |
Inoue, M; Naito, H; Okumura, T; Suzuki, Y | 1 |
Altikat, S; Ciftci, M; Coban, A; Ozdemir, H | 1 |
Arslan, G; Bozdogan, N; Donmez, A; Ozer, C; Sener, M; Yilmaz, I; Yilmazer, C | 1 |
Ciftci, M; Irfan Kufrevioglu, O; Senturk, M | 1 |
Au, AL; Chan, SW; Kwan, YW; Lee, SM; Leung, GP; Li, RW; Seto, SW; Tse, CM | 1 |
Beydemir, S; Ekinci, D | 1 |
Amerov, DB; Kazennov, VV; Shishkin, MN; Tsar'kov, DB | 1 |
Aguilar, C; Borrull, F; Botello, I; Calull, M | 1 |
Ardic, S; Arziman, I; Bayir, A; Cevik, E; Cinar, O; Salman, N; Youngquist, ST | 1 |
Büget, M; Güresti, E; Koltka, K; Özyalçın, S; Sentürk, M; Sivrikoz, N | 1 |
Bendtsen, L; Derry, S; Moore, RA; Wiffen, PJ | 1 |
Aldington, D; Bell, RF; Derry, S; Gaskell, H; Kalso, EA; Moore, RA; Phillips, T; Wiffen, PJ | 1 |
Kocak, AO | 1 |
Akbas, I; Cakir, Z; Kocak, AO; Kocak, MB | 1 |
Gromova, OA; Putilina, MV; Rudakov, KV; Stakhovskaia, LV; Torshin, IY | 1 |
Elshaer, SL; Shaaban, MI; Shaldam, MA | 1 |
7 review(s) available for ketoprofen and piroxicam
Article | Year |
---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Non-steroidal and analgesic therapy in the elderly.
Topics: Acetaminophen; Aged; Analgesics; Analgesics, Opioid; Anti-Inflammatory Agents; Apazone; Aspirin; Central Nervous System Diseases; Chemical and Drug Induced Liver Injury; Diclofenac; Drug Hypersensitivity; Gastrointestinal Diseases; Hematologic Diseases; Humans; Ibuprofen; Indomethacin; Ketoprofen; Kidney Diseases; Kinetics; Naproxen; Phenylbutazone; Piroxicam; Salicylates; Thiazines | 1986 |
Update on ibuprofen for rheumatoid arthritis.
Topics: Anti-Inflammatory Agents; Arthritis, Rheumatoid; Aspirin; Clinical Trials as Topic; Drug Tolerance; Fenoprofen; Humans; Ibuprofen; Indomethacin; Ketoprofen; Naproxen; Piroxicam; Sulindac; Thiazines; Tolmetin | 1984 |
Piroxicam-beta-cyclodextrin in the treatment of acute pain of rheumatic disease.
Topics: Acute Disease; Adult; beta-Cyclodextrins; Controlled Clinical Trials as Topic; Cyclodextrins; Diclofenac; Dipyrone; Drug Combinations; Etodolac; Humans; Ketoprofen; Middle Aged; Pain; Piroxicam; Rheumatic Diseases | 1993 |
Use of carprofen for the treatment of pain and inflammation in dogs.
Topics: Acetaminophen; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Carbazoles; Clonixin; Cyclooxygenase Inhibitors; Dog Diseases; Dogs; Ibuprofen; Indomethacin; Ketoprofen; Meclofenamic Acid; Meloxicam; Naproxen; Osteoarthritis; Pain; Phenylbutazone; Piroxicam; Thiazines; Thiazoles | 1997 |
Ibuprofen for acute treatment of episodic tension-type headache in adults.
Topics: Acetaminophen; Administration, Oral; Adult; Analgesics, Non-Narcotic; Cyclooxygenase Inhibitors; Diclofenac; Humans; Ibuprofen; Ketoprofen; Naproxen; Numbers Needed To Treat; Pain Measurement; Piroxicam; Randomized Controlled Trials as Topic; Tension-Type Headache; Time Factors | 2015 |
Topical analgesics for acute and chronic pain in adults - an overview of Cochrane Reviews.
Topics: Acute Pain; Adult; Analgesics; Arthritis, Rheumatoid; Capsaicin; Chronic Pain; Diclofenac; Humans; Ketoprofen; Musculoskeletal Pain; Neuralgia; Numbers Needed To Treat; Osteoarthritis; Piroxicam; Publication Bias; Review Literature as Topic | 2017 |
12 trial(s) available for ketoprofen and piroxicam
Article | Year |
---|---|
A randomised double-blind multicentre trial comparing tenoxicam and ketoprofen in osteoarthritis.
Topics: Adult; Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Double-Blind Method; Female; Humans; Ketoprofen; Male; Middle Aged; Multicenter Studies as Topic; Osteoarthritis; Pain Measurement; Piroxicam; Randomized Controlled Trials as Topic | 1989 |
Isoxicam vs ketoprofen in ankylosing spondylitis.
Topics: Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Double-Blind Method; Female; Humans; Ketoprofen; Male; Middle Aged; Pain Measurement; Phenylpropionates; Piroxicam; Random Allocation; Sleep; Spondylitis, Ankylosing | 1986 |
Double-blind preference and compliance multicentre study in osteoarthritis: once-a-day treatment.
Topics: Adult; Aged; Aspirin; Clinical Trials as Topic; Diclofenac; Double-Blind Method; Drug Administration Schedule; Humans; Indomethacin; Indoprofen; Ketoprofen; Middle Aged; Naproxen; Osteoarthritis; Pain; Patient Compliance; Piroxicam; Thiazines | 1985 |
Update on ibuprofen for rheumatoid arthritis.
Topics: Anti-Inflammatory Agents; Arthritis, Rheumatoid; Aspirin; Clinical Trials as Topic; Drug Tolerance; Fenoprofen; Humans; Ibuprofen; Indomethacin; Ketoprofen; Naproxen; Piroxicam; Sulindac; Thiazines; Tolmetin | 1984 |
Nimesulide in the treatment of osteoarthritis. Double-blind studies in comparison with piroxicam, ketoprofen and placebo.
Topics: Adult; Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Double-Blind Method; Female; Humans; Ketoprofen; Male; Middle Aged; Osteoarthritis; Piroxicam; Sulfonamides | 1993 |
Methotrexate disposition following concomitant administration of ketoprofen, piroxicam and flurbiprofen in patients with rheumatoid arthritis.
Topics: Administration, Oral; Adult; Aged; Arthritis, Rheumatoid; Drug Interactions; Drug Therapy, Combination; Female; Fluorescence Polarization Immunoassay; Flurbiprofen; Humans; Ketoprofen; Male; Metabolic Clearance Rate; Methotrexate; Middle Aged; Piroxicam | 1994 |
Nonsteroidal antiinflammatory drugs in rheumatoid arthritis and osteoarthritis: support for the concept of "responders" and "nonresponders".
Topics: Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Rheumatoid; Blood Sedimentation; Cross-Over Studies; Double-Blind Method; Female; Humans; Ketoprofen; Lymphocyte Count; Male; Middle Aged; Osteoarthritis; Piroxicam; Receptors, Interleukin-2; Thromboxane B2; Tumor Necrosis Factor-alpha | 1997 |
Efficacy of lornoxicam for acute postoperative pain relief after septoplasty: a comparison with diclofenac, ketoprofen, and dipyrone.
Topics: Adult; Aged; Analgesics, Opioid; Anti-Inflammatory Agents, Non-Steroidal; Diclofenac; Dipyrone; Double-Blind Method; Female; Humans; Ketoprofen; Male; Meperidine; Middle Aged; Nasal Septum; Pain Measurement; Pain, Postoperative; Piroxicam; Postoperative Nausea and Vomiting; Prospective Studies; Statistics, Nonparametric; Time Factors; Treatment Outcome | 2008 |
Comparing the efficacy of intravenous tenoxicam, lornoxicam, and dexketoprofen trometamol for the treatment of renal colic.
Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Double-Blind Method; Emergency Service, Hospital; Humans; Injections, Intravenous; Ketoprofen; Male; Pain Management; Pain Measurement; Piroxicam; Prospective Studies; Renal Colic; Treatment Outcome; Tromethamine | 2012 |
Perioperative dexketoprofen or lornoxicam administration for pain management after major orthopedic surgery: a randomized, controlled study.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Arthroplasty, Replacement, Hip; Double-Blind Method; Female; Humans; Infusions, Intravenous; Ketoprofen; Male; Middle Aged; Pain Measurement; Pain, Postoperative; Perioperative Care; Piroxicam; Prospective Studies; Treatment Outcome; Tromethamine | 2014 |
Intradermal mesotherapy versus systemic therapy in the treatment of musculoskeletal pain: A prospective randomized study.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Emergency Service, Hospital; Female; Follow-Up Studies; Humans; Injections, Intravenous; Ketoprofen; Male; Mesotherapy; Middle Aged; Musculoskeletal Pain; Piroxicam; Prospective Studies; Treatment Outcome; Tromethamine; Young Adult | 2019 |
Comparison of intradermal mesotherapy with systemic therapy in the treatment of low back pain: A prospective randomized study.
Topics: Adult; Anesthetics, Local; Anti-Inflammatory Agents, Non-Steroidal; Colchicine; Emergency Service, Hospital; Female; Humans; Intervertebral Disc Displacement; Ketoprofen; Lidocaine; Low Back Pain; Male; Mesotherapy; Middle Aged; Piroxicam; Prospective Studies; Visual Analog Scale | 2020 |
68 other study(ies) available for ketoprofen and piroxicam
Article | Year |
---|---|
Hologram QSAR model for the prediction of human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2007 |
Transport properties of nonsteroidal anti-inflammatory drugs by organic anion transporter 1 expressed in Xenopus laevis oocytes.
Topics: Animals; Anion Transport Proteins; Anti-Inflammatory Agents, Non-Steroidal; Biological Transport; Carrier Proteins; Oocytes; Xenopus laevis | 1999 |
Nonsteroidal anti-inflammatory drugs efficiently reduce the transport and cytotoxicity of adefovir mediated by the human renal organic anion transporter 1.
Topics: Adenine; Anion Transport Proteins; Anti-Inflammatory Agents, Non-Steroidal; Antiviral Agents; Biological Transport; Carrier Proteins; Humans; Kidney; Organophosphonates; Structure-Activity Relationship | 2000 |
High-throughput permeability pH profile and high-throughput alkane/water log P with artificial membranes.
Topics: Alkanes; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Membranes, Artificial; Octanols; Permeability; Pharmaceutical Preparations; Solubility; Water | 2001 |
Characterization of methotrexate transport and its drug interactions with human organic anion transporters.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biological Transport; Cells, Cultured; Humans; Indomethacin; Kinetics; Liver-Specific Organic Anion Transporter 1; Methotrexate; Mice; Mice, Transgenic; Nerve Tissue Proteins; Organic Anion Transporters, Sodium-Independent; Phenylbutazone; Potassium Channels; Potassium Channels, Tandem Pore Domain; Probenecid | 2002 |
Novel cyclooxygenase-1 inhibitors discovered using affinity fingerprints.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Combinatorial Chemistry Techniques; Cyclooxygenase 1; Cyclooxygenase Inhibitors; Drug Design; Drug Evaluation, Preclinical; Ibuprofen; Inhibitory Concentration 50; Isoenzymes; Models, Molecular; Models, Theoretical; Molecular Structure; Prospective Studies; Prostaglandin-Endoperoxide Synthases; Quantitative Structure-Activity Relationship | 2004 |
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration | 2004 |
Parallel artificial membrane permeability assay: a new membrane for the fast prediction of passive human skin permeability.
Topics: 1-Octanol; Diffusion; Dimethylpolysiloxanes; Humans; In Vitro Techniques; Membranes, Artificial; Myristates; Permeability; Skin; Skin Absorption; Water | 2006 |
In silico and in vitro filters for the fast estimation of skin permeation and distribution of new chemical entities.
Topics: Humans; Membranes, Artificial; Models, Biological; Models, Molecular; Octanols; Permeability; Pharmaceutical Preparations; Skin Absorption; Water | 2007 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
QSAR study on permeability of hydrophobic compounds with artificial membranes.
Topics: Biological Transport; Caco-2 Cells; Drug Evaluation, Preclinical; Humans; Hydrophobic and Hydrophilic Interactions; Membranes, Artificial; Permeability; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship | 2007 |
Transdermal penetration behaviour of drugs: CART-clustering, QSPR and selection of model compounds.
Topics: Anti-Inflammatory Agents; Cell Membrane Permeability; Cluster Analysis; Drug Evaluation, Preclinical; Humans; Models, Biological; Predictive Value of Tests; Quantitative Structure-Activity Relationship; Regression Analysis; Skin; Skin Absorption | 2007 |
Molecular characteristics for solid-state limited solubility.
Topics: Chemical Phenomena; Chemistry, Physical; Molecular Structure; Multivariate Analysis; Pharmaceutical Preparations; Regression Analysis; Solubility | 2008 |
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship | 2008 |
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution | 2009 |
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship | 2009 |
Development of an in silico model for human skin permeation based on a Franz cell skin permeability assay.
Topics: 1-Methyl-3-isobutylxanthine; Cell Line; Cell Membrane Permeability; Humans; Models, Biological; Quantitative Structure-Activity Relationship; Skin Absorption | 2010 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical | 2010 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
How well can the Caco-2/Madin-Darby canine kidney models predict effective human jejunal permeability?
Topics: Animals; Disease Models, Animal; Dogs; Humans; Jejunal Diseases; Kidney Diseases; Models, Biological; Permeability; Porosity; Regression Analysis | 2010 |
Developing structure-activity relationships for the prediction of hepatotoxicity.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes | 2010 |
QSAR-based solubility model for drug-like compounds.
Topics: Databases, Factual; Models, Molecular; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Solubility; Water | 2010 |
A predictive ligand-based Bayesian model for human drug-induced liver injury.
Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands | 2010 |
A combined spectroscopic and crystallographic approach to probing drug-human serum albumin interactions.
Topics: Binding Sites; Crystallography, X-Ray; Drug Interactions; Humans; Pharmaceutical Preparations; Protein Binding; Protein Structure, Tertiary; Serum Albumin; Spectrometry, Fluorescence | 2010 |
Importance of physicochemical properties for the design of new pesticides.
Topics: Anabasine; Animals; Biological Availability; Cell Membrane Permeability; Chemical Phenomena; Drug Design; Humans; Imidazoles; Insecticides; Neonicotinoids; Nitro Compounds; Pesticides; Quantitative Structure-Activity Relationship; Receptors, Nicotinic | 2011 |
QSAR-based permeability model for drug-like compounds.
Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2011 |
Predicting phenolic acid absorption in Caco-2 cells: a theoretical permeability model and mechanistic study.
Topics: Artificial Intelligence; Caco-2 Cells; Cell Membrane Permeability; Cinnamates; Enterocytes; Humans; Hydrophobic and Hydrophilic Interactions; Intestinal Absorption; Kinetics; Models, Biological; Molecular Conformation; Osmolar Concentration; Phenols | 2012 |
Self-organizing molecular field analysis of NSAIDs: assessment of pharmacokinetic and physicochemical properties using 3D-QSPkR approach.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Chemical Phenomena; Computational Biology; Least-Squares Analysis; Models, Molecular; Molecular Conformation; Quantitative Structure-Activity Relationship | 2012 |
Discovery and characterization of novel, potent, and selective cytochrome P450 2J2 inhibitors.
Topics: Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2J2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Drug Discovery; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Microsomes, Liver; Models, Molecular; Molecular Dynamics Simulation; Substrate Specificity | 2013 |
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat | 2016 |
The economic consequences of NSAID-induced gastropathy: the French context.
Topics: Ambulatory Care; Anti-Inflammatory Agents, Non-Steroidal; Cost of Illness; Diclofenac; Duodenal Ulcer; Economics, Hospital; Etodolac; France; Gastrointestinal Diseases; Humans; Ketoprofen; Naproxen; National Health Programs; Piroxicam; Rheumatic Diseases; Sulindac | 1992 |
Effect of non-steroidal anti-inflammatory drugs on glutathione levels in various organs of rat.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Brain; Cell Death; Eye; Gastric Mucosa; Glutathione; Heart; Ketoprofen; Liver; Male; Muscles; Naproxen; Piroxicam; Rats; Rats, Wistar; Stomach | 1992 |
Inhibition of colon carcinogenesis by prostaglandin synthesis inhibitors and related compounds.
Topics: Animals; Azoxymethane; Colonic Neoplasms; Glycyrrhetinic Acid; Ibuprofen; Ketoprofen; Male; Piroxicam; Random Allocation; Rats; Rats, Inbred F344 | 1992 |
In vitro effect of nonsteroidal antiinflammatory drugs on proteoglycanase and collagenase activity in human osteoarthritic cartilage.
Topics: Acetaminophen; Aged; Anti-Inflammatory Agents, Non-Steroidal; Cartilage, Articular; Diclofenac; Endopeptidases; Female; Humans; Indomethacin; Ketoprofen; Male; Metalloendopeptidases; Microbial Collagenase; Middle Aged; Osteoarthritis, Hip; Piroxicam; Salicylates; Salicylic Acid | 1991 |
Comparison of the effects of non-steroidal anti-inflammatory drugs (NSAIDs) on proteoglycan synthesis by articular cartilage explant and chondrocyte monolayer cultures.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cartilage, Articular; Cells, Cultured; Culture Techniques; Diclofenac; Indomethacin; Ketoprofen; Piroxicam; Propionates; Proteoglycans; Rabbits; Time Factors | 1991 |
Influence of some anti-inflammatory drugs on the activity of aryl hydrocarbon hydroxylase and the cytochrome P450 content.
Topics: Acetaminophen; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aryl Hydrocarbon Hydroxylases; Cytochrome P-450 Enzyme System; Injections, Intraperitoneal; Ketoprofen; Male; Mice; Microsomes, Liver; Phenylbutazone; Piroxicam; Pyrazoles | 1990 |
Impairment of human antipyrine metabolism by piroxicam.
Topics: Administration, Oral; Adolescent; Adult; Antipyrine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Humans; Ketoprofen; Male; Naproxen; Piroxicam; Saliva; Time Factors | 1990 |
Low back pain.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Back Pain; Diclofenac; Humans; Ketoprofen; Piroxicam | 1987 |
The history of diclofenac.
Topics: Chemical Phenomena; Chemistry; Diclofenac; Humans; Hydrogen-Ion Concentration; Ibuprofen; Indenes; Indomethacin; Ketoprofen; Naproxen; Phenylbutazone; Piroxicam; Prostaglandin-Endoperoxide Synthases; Structure-Activity Relationship; Thiazines | 1986 |
Effect of some new prostaglandin synthetase inhibitors on the endotoxin induced mortality and biochemical changes in experimental animals.
Topics: Acetates; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase Inhibitors; Endotoxins; Ketoprofen; Male; Mice; Piroxicam; Rats; Rats, Inbred Strains; Shock, Septic; Thiazoles | 1988 |
The history of diclofenac.
Topics: Diclofenac; History, 20th Century; Ibuprofen; Ketoprofen; Models, Molecular; Naproxen; Phenylbutazone; Piroxicam; Solubility; Structure-Activity Relationship; Thiazines | 1985 |
Bleeding from peptic ulcers and use of non-steroidal anti-inflammatory drugs in the Romford area.
Topics: Aged; Anti-Inflammatory Agents; Drug Utilization; England; Humans; Ketoprofen; Peptic Ulcer Hemorrhage; Piroxicam; Stomach Ulcer; Thiazines | 1985 |
Evidence for the involvement of arachidonic acid metabolites in spontaneous and drug-induced contractions of rat urinary bladder.
Topics: Adenosine Diphosphate; Animals; Anti-Inflammatory Agents; Arachidonic Acid; Arachidonic Acids; Aspirin; Diet; Fatty Acids, Essential; Hexamethonium Compounds; Indomethacin; Ketoprofen; Male; Muscle Contraction; Physostigmine; Piroxicam; Rats; Rats, Inbred Strains; Tetrodotoxin; Thiazines; Urinary Bladder | 1984 |
Poisoning after overdose with non-steroidal anti-inflammatory drugs.
Topics: Adolescent; Adult; Aged; Anti-Inflammatory Agents; Child; Child, Preschool; Diflunisal; Female; Fenoprofen; Feprazone; Humans; Ibuprofen; Indomethacin; Ketoprofen; London; Male; Mefenamic Acid; Naproxen; Oxyphenbutazone; Phenylbutazone; Piroxicam; Thiazines; Tolmetin | 1984 |
[Studies on isolated rat hepatocytes (6)].
Topics: Actihaemyl; Animals; Anti-Inflammatory Agents; Cefoperazone; Cell Survival; Cells, Cultured; Glutathione; Ketoprofen; Liver; Oxygen Consumption; Pipemidic Acid; Piperidines; Piroxicam; Pyridazines; Rats; Rats, Inbred Strains; Rifampin; Thiazines | 1984 |
Restoration of postburn impaired lymphocyte responsiveness by nonsteroidal anti-inflammatory drugs is independent of prostaglandin E2 inhibition.
Topics: Administration, Oral; Amino Acid Oxidoreductases; Animals; Anti-Inflammatory Agents, Non-Steroidal; Burns; Dinoprostone; Indomethacin; Ketoprofen; Lymphocyte Activation; Male; Niflumic Acid; Nitric Oxide Synthase; Piroxicam; Rats; Rats, Wistar; Salicylates | 1994 |
A reproducible and rapid HPLC assay for quantitation of piroxicam in plasma.
Topics: Calibration; Chromatography, High Pressure Liquid; Humans; Hydrogen-Ion Concentration; Ketoprofen; Linear Models; Piroxicam; Reproducibility of Results; Spectrophotometry, Ultraviolet | 1995 |
Effect of etodolac on prostaglandin E2 biosynthesis, active oxygen generation and bradykinin formation.
Topics: Animals; Aspirin; Bradykinin; Bromelains; Cartilage, Articular; Cell Line; Concanavalin A; Depression, Chemical; Diclofenac; Dinoprostone; Dogs; Etodolac; Gastric Mucosa; Guinea Pigs; Indomethacin; Interleukin-1; Ketoprofen; Kidney; Naproxen; Oxygen; Pain; Piroxicam; Rabbits; Rats | 1994 |
Effect of the low molecular weight heparin/non steroidal anti-inflammatory drugs association on an experimental thrombosis induced by laser.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Drug Therapy, Combination; Indomethacin; Injections, Subcutaneous; Ketoprofen; Lasers; Male; Nadroparin; Piroxicam; Platelet Aggregation; Rats; Rats, Wistar; Thrombolytic Therapy; Thrombosis | 1995 |
The determination of non-steroidal antiinflammatory drugs in pharmaceuticals by capillary zone electrophoresis and micellar electrokinetic capillary chromatography.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Buffers; Calibration; Chemistry, Pharmaceutical; Chromatography; Diclofenac; Dosage Forms; Electrophoresis; Ibuprofen; Indomethacin; Ketoprofen; Micelles; Piroxicam; Reference Standards; Regression Analysis; Reproducibility of Results | 1994 |
Non-steroidal anti-inflammatory drugs (NSAIDs) affect the glutathione (GSH) levels in the brain.
Topics: Animals; Brain Chemistry; Cerebellum; Cerebral Cortex; Glutathione; Ketoprofen; Male; Naproxen; Piroxicam; Rats; Rats, Wistar | 1993 |
Variability in the risk of major gastrointestinal complications from nonaspirin nonsteroidal anti-inflammatory drugs.
Topics: Administration, Oral; Administration, Rectal; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Alcohol Drinking; Aspirin; Case-Control Studies; Dose-Response Relationship, Drug; Female; Gastrointestinal Diseases; Humans; Incidence; Ketoprofen; Male; Middle Aged; Naproxen; Peptic Ulcer; Piroxicam; Prospective Studies; Risk Factors; Sex Factors; Time Factors | 1993 |
Phototoxicity of non-steroidal anti-inflammatory drugs: in vitro studies with visible light.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Carbazoles; Dermatitis, Phototoxic; Diclofenac; Erythrocytes; Hemolysis; Humans; Ibuprofen; In Vitro Techniques; Ketoprofen; Light; Naproxen; Phenylbutazone; Photosensitizing Agents; Piroxicam; Propionates | 1996 |
Inflammation modifies the role of cyclooxygenases in the contractile responses of the rat detrusor smooth muscle to kinin agonists.
Topics: Animals; Bradykinin; Cystitis; Dinoprostone; In Vitro Techniques; Ketoprofen; Male; Muscle Contraction; Nitrobenzenes; Piroxicam; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Receptors, Bradykinin; Sulfonamides; Urinary Bladder | 1998 |
Caco-2 versus Caco-2/HT29-MTX co-cultured cell lines: permeabilities via diffusion, inside- and outside-directed carrier-mediated transport.
Topics: Antipyrine; Atenolol; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Caco-2 Cells; Carrier Proteins; Cell Membrane Permeability; Cellular Senescence; Coculture Techniques; Furosemide; HT29 Cells; Humans; Intestinal Absorption; Intestinal Mucosa; Ketoprofen; Mannitol; Metoprolol; Microscopy, Electron; Piroxicam; Reproducibility of Results; Terbutaline | 2000 |
Presurgical ketoprofen, but not morphine, dipyrone, diclofenac or tenoxicam, preempts post-incisional mechanical allodynia in rats.
Topics: Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Diclofenac; Dipyrone; Ketoprofen; Male; Mechanoreceptors; Morphine; Pain Threshold; Pain, Postoperative; Physical Stimulation; Piroxicam; Postoperative Care; Preoperative Care; Rats; Rats, Wistar | 2002 |
Antinociceptive synergy, additivity, and subadditivity with combinations of oral glucosamine plus nonopioid analgesics in mice.
Topics: Acetaminophen; Administration, Oral; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Diclofenac; Disease Models, Animal; Drug Therapy, Combination; Glucosamine; Ibuprofen; Indomethacin; Ketoprofen; Mice; Pain; Piroxicam | 2003 |
Amphiphilic star-like macromolecules as novel carriers for topical delivery of nonsteroidal anti-inflammatory drugs.
Topics: Administration, Topical; Animals; Anti-Inflammatory Agents, Non-Steroidal; Chemistry, Pharmaceutical; Drug Carriers; Drug Delivery Systems; Female; Indomethacin; Ketoprofen; Macromolecular Substances; Male; Mice; Permeability; Piroxicam; Skin Absorption | 2003 |
Ultrasonic vocalization response elicited in adjuvant-induced arthritic rats as a useful method for evaluating analgesic drugs.
Topics: Analgesics; Animals; Arthritis, Experimental; Drug Evaluation, Preclinical; Ketoprofen; Lactones; Male; Piroxicam; Rats; Rats, Inbred Lew; Social Behavior; Sulfones; Ultrasonics; Vocalization, Animal | 2006 |
In vitro effects of some drugs on catalase purified from human skin.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Catalase; Diclofenac; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; In Vitro Techniques; Inhibitory Concentration 50; Ketoprofen; Piroxicam; Skin; Sulfamethoxazole | 2006 |
Effects of some analgesic anaesthetic drugs on human erythrocyte glutathione reductase: an in vitro study.
Topics: Analgesics; Anesthetics; Chromatography, Gel; Diclofenac; Dose-Response Relationship, Drug; Erythrocytes; Etomidate; Glutathione Reductase; Humans; Inhibitory Concentration 50; Ketoprofen; Kinetics; Morphine; Piroxicam; Propofol | 2009 |
Inhibitory effect of nonsteroidal anti-inflammatory drugs on adenosine transport in vascular smooth muscle cells.
Topics: Adenosine; Anti-Inflammatory Agents, Non-Steroidal; Aorta; Cell Proliferation; Cells, Cultured; Coloring Agents; Dose-Response Relationship, Drug; Etodolac; Humans; Indomethacin; Inhibitory Concentration 50; Ketoprofen; Kinetics; Mefenamic Acid; Muscle, Smooth, Vascular; Piroxicam; Sulindac; Temperature; Tetrazolium Salts; Thiazoles; Thioinosine | 2009 |
Effect of some analgesics on paraoxonase-1 purified from human serum.
Topics: Analgesics; Aryldialkylphosphatase; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Enzyme Inhibitors; Humans; Ketoprofen; Molecular Structure; Piroxicam; Serum | 2009 |
[Postoperative analgesia].
Topics: Acetaminophen; Adult; Aged; Analgesia; Analgesics, Non-Narcotic; Analgesics, Opioid; Anti-Inflammatory Agents, Non-Steroidal; Aorta, Abdominal; Blood Vessel Prosthesis; Drug Therapy, Combination; Female; Humans; Ketoprofen; Male; Middle Aged; Pain, Postoperative; Piroxicam; Tramadol | 2010 |
Electrokinetic supercharging focusing in capillary zone electrophoresis of weakly ionizable analytes in environmental and biological samples.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Diclofenac; Electrophoresis, Capillary; Fenoprofen; Humans; Hydrogen-Ion Concentration; Isoelectric Focusing; Ketoprofen; Methanol; Naproxen; Piroxicam; Reproducibility of Results; Rivers; Sensitivity and Specificity; Sodium Chloride; Time Factors; Water Pollutants, Chemical | 2010 |
[The chemoreactomic analysis of the central mechanisms of action of non-steroidal anti-inflammatory drugs].
Topics: Anti-Inflammatory Agents, Non-Steroidal; Diclofenac; Humans; Ketoprofen; Opiate Alkaloids; Pain; Piroxicam | 2020 |
Ketoprofen, piroxicam and indomethacin-suppressed quorum sensing and virulence factors in Acinetobacter baumannii.
Topics: Acinetobacter baumannii; Anti-Bacterial Agents; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Biofilms; Chromobacterium; Hydrogen; Indomethacin; Ketoprofen; Molecular Docking Simulation; Piroxicam; Quorum Sensing; Virulence Factors | 2022 |