ketoconazole and pentamidine

ketoconazole has been researched along with pentamidine in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19904 (16.00)18.7374
1990's8 (32.00)18.2507
2000's2 (8.00)29.6817
2010's10 (40.00)24.3611
2020's1 (4.00)2.80

Authors

AuthorsStudies
Bernardino, AMR; Boechat, N; Dos Santos, MS; Faria, JV; Miguita, AGC; Vegi, PF1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Carvalho, L; Castanys, S; Gamarro, F; Manzano, JI; Pérez-Victoria, JM1
Amaral, VF; Bernardino, AM; Canto-Cavalheiro, MM; de Carvalho, FT; de Léo, RM; dos Santos, MS; Leon, LL; Oliveira, ML1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Bowlin, TL; Ding, X; Kwasny, SM; Nguyen, ST; Opperman, TJ; Peet, NP; Williams, JD1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Chaffanjon, P; Delbeke, E; Lafeuillade, A; Quilichini, R1
Aggarwal, P; Gupta, U; Saluja, S; Singh, S; Wali, JP1
St-Germain, G1
Berman, JD; Gallalee, JV1
Berman, JD; Lee, LS1
Berman, JD1
Berman, JD; Langreth, SG; Lee, LS; Riordan, GP1
Buffet, P; Caumes, E; Gentilini, M1
Chandra, J; Patwari, AK1
Gaspari, AA; Pabico, RC; Sickel, JZ; Slater, CA; Visvesvara, GS1
Berman, JD; Grogl, M; Soto-Mancipe, J1
Berti, E; Girgenti, V; Recalcati, S; Venegoni, L; Veraldi, S; Vezzoli, P1
Escobar, P; Salazar-Villamizar, ME1

Reviews

4 review(s) available for ketoconazole and pentamidine

ArticleYear
Recently reported biological activities of pyrazole compounds.
    Bioorganic & medicinal chemistry, 2017, 11-01, Volume: 25, Issue:21

    Topics: Analgesics; Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Antifungal Agents; Antineoplastic Agents; Antiviral Agents; Humans; Pyrazoles

2017
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
[Treatment of localized cutaneous leishmaniasis].
    Annales de dermatologie et de venereologie, 1994, Volume: 121, Issue:6-7

    Topics: Amphotericin B; Antimony Sodium Gluconate; Antiprotozoal Agents; Humans; Itraconazole; Ketoconazole; Leishmaniasis, Cutaneous; Meglumine; Meglumine Antimoniate; Organometallic Compounds; Pentamidine

1994
Diagnosis and treatment of kala-azar.
    Indian pediatrics, 1994, Volume: 31, Issue:6

    Topics: Allopurinol; Amphotericin B; Antimony Sodium Gluconate; Child; Combined Modality Therapy; Humans; Ketoconazole; Leishmaniasis, Visceral; Pentamidine; Predictive Value of Tests; Reproducibility of Results; Sensitivity and Specificity; Splenectomy

1994

Trials

1 trial(s) available for ketoconazole and pentamidine

ArticleYear
Evaluation of pentamidine for the treatment of cutaneous leishmaniasis in Colombia.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 1993, Volume: 16, Issue:3

    Topics: Administration, Oral; Adolescent; Adult; Antifungal Agents; Colombia; Follow-Up Studies; Humans; Injections, Intramuscular; Itraconazole; Ketoconazole; Leishmaniasis, Cutaneous; Male; Meglumine; Pentamidine; Treatment Outcome

1993

Other Studies

20 other study(ies) available for ketoconazole and pentamidine

ArticleYear
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Increased glycolytic ATP synthesis is associated with tafenoquine resistance in Leishmania major.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:3

    Topics: Adenosine Triphosphate; Aminoquinolines; Antiprotozoal Agents; Drug Resistance; Glycolysis; Leishmania major; Pyruvate Kinase

2011
Synthesis and antileishmanial evaluation of 1-aryl-4-(4,5-dihydro-1H-imidazol-2-yl)-1H-pyrazole derivatives.
    Bioorganic & medicinal chemistry letters, 2011, Dec-15, Volume: 21, Issue:24

    Topics: Animals; Antiprotozoal Agents; Imidazoles; Leishmania; Leishmaniasis; Mice; Pyrazoles; Structure-Activity Relationship

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Synthesis and antifungal evaluation of head-to-head and head-to-tail bisamidine compounds.
    Bioorganic & medicinal chemistry, 2015, Sep-01, Volume: 23, Issue:17

    Topics: Antifungal Agents; Candida; Cryptococcus neoformans; DNA-Binding Proteins; Furans; Humans

2015
Maintenance itraconazole for visceral leishmaniasis in HIV infection.
    The American journal of medicine, 1992, Volume: 92, Issue:4

    Topics: Adult; Antifungal Agents; Female; HIV Infections; Humans; Itraconazole; Ketoconazole; Leishmaniasis, Visceral; Opportunistic Infections; Pentamidine

1992
Ketoconazole in the treatment of antimony- and pentamidine-resistant kala-azar.
    The Journal of infectious diseases, 1992, Volume: 166, Issue:1

    Topics: Antimony; Drug Resistance; Humans; Ketoconazole; Leishmaniasis, Visceral; Pentamidine

1992
Effects of pentamidine alone and in combination with ketoconazole or itraconazole on the growth of Candida albicans.
    Antimicrobial agents and chemotherapy, 1990, Volume: 34, Issue:12

    Topics: Acquired Immunodeficiency Syndrome; Antifungal Agents; Candida albicans; Candidiasis; Drug Resistance, Microbial; Humans; Itraconazole; Ketoconazole; Microbial Sensitivity Tests; Pentamidine

1990
Semiautomated assessment of in vitro activity of potential antileishmanial drugs.
    Antimicrobial agents and chemotherapy, 1985, Volume: 28, Issue:6

    Topics: Aminoquinolines; Amphotericin B; Antimony Sodium Gluconate; Antiprotozoal Agents; Automation; Azure Stains; Drug Evaluation, Preclinical; Formycins; Humans; In Vitro Techniques; Ketoconazole; Leishmania tropica; Macrophages; Pentamidine; Tritium; Uracil

1985
Activity of antileishmanial agents against amastigotes in human monocyte-derived macrophages and in mouse peritoneal macrophages.
    The Journal of parasitology, 1984, Volume: 70, Issue:2

    Topics: Aminoquinolines; Animals; Antimony Sodium Gluconate; Antiprotozoal Agents; Ascitic Fluid; Cells, Cultured; Drug Evaluation, Preclinical; Gluconates; Humans; Ketoconazole; Leishmania; Macrophages; Mice; Mice, Inbred BALB C; Monocytes; Pentamidine; Primaquine

1984
In vitro susceptibility of antimony-resistant Leishmania to alternative drugs.
    The Journal of infectious diseases, 1982, Volume: 145, Issue:2

    Topics: Amphotericin B; Anti-Bacterial Agents; Antibiotics, Antineoplastic; Antimony; Formycins; Humans; Imidazoles; Ketoconazole; Leishmaniasis; Pentamidine; Piperazines

1982
Fine-structural alterations in Leishmania tropica within human macrophages exposed to antileishmanial drugs in vitro.
    The Journal of protozoology, 1983, Volume: 30, Issue:3

    Topics: Aminoquinolines; Amphotericin B; Animals; Antimony Sodium Gluconate; Antiprotozoal Agents; Cell Membrane; Formycins; Humans; Intracellular Membranes; Ketoconazole; Leishmania; Macrophages; Organoids; Pentamidine

1983
Drugs for AIDS and associated infections.
    The Medical letter on drugs and therapeutics, 1995, Oct-13, Volume: 37, Issue:959

    Topics: Acquired Immunodeficiency Syndrome; AIDS-Related Opportunistic Infections; Amphotericin B; Antifungal Agents; Antiprotozoal Agents; Antiviral Agents; Atovaquone; Candidiasis, Oral; Clindamycin; Clotrimazole; Cryptosporidiosis; Cytomegalovirus Infections; Dapsone; Didanosine; Drug Combinations; Drug Therapy, Combination; Fluconazole; Flucytosine; Folic Acid Antagonists; Foscarnet; Glucuronates; Herpes Simplex; Herpes Zoster; Humans; Isoniazid; Itraconazole; Ketoconazole; Lamivudine; Mycobacterium avium-intracellulare Infection; Naphthoquinones; Nystatin; Pentamidine; Pneumocystis Infections; Pneumonia, Pneumocystis; Prednisone; Primaquine; Reverse Transcriptase Inhibitors; Stavudine; Syphilis; Toxoplasmosis; Trimetrexate; Tuberculosis; Zalcitabine; Zidovudine

1995
Brief report: successful treatment of disseminated acanthamoeba infection in an immunocompromised patient.
    The New England journal of medicine, 1994, Jul-14, Volume: 331, Issue:2

    Topics: Acanthamoeba; Adult; Amebiasis; Animals; Antiparasitic Agents; Chlorhexidine; Humans; Immunocompromised Host; Ketoconazole; Male; Pentamidine

1994
Cutaneous lymphoid hyperplasia associated with Leishmania panamensis infection.
    Acta dermato-venereologica, 2010, Volume: 90, Issue:4

    Topics: Administration, Oral; Aged; Antiprotozoal Agents; Female; Humans; Infusions, Intravenous; Ketoconazole; Leishmania guyanensis; Leishmaniasis, Mucocutaneous; Pentamidine; Pseudolymphoma; Treatment Outcome

2010
In vitro selection of ketoconazole-pentamidine-resistant Leishmania (Viannia) braziliensis strains.
    Experimental parasitology, 2022, Volume: 233

    Topics: Analysis of Variance; Animals; Antiprotozoal Agents; Drug Resistance; Drug Therapy, Combination; Female; Humans; Inhibitory Concentration 50; Ketoconazole; Leishmania braziliensis; Leishmaniasis, Cutaneous; Male; Mice; Mice, Inbred BALB C; Pentamidine; THP-1 Cells

2022